Get started
Author

Abdellah Yamani

Observed name: A. Yamani
ORCID: 0009-0006-9516-9387
Observed ORCID: 0009-0006-9516-9387
OpenAlex ID: A5001779027
Trypanothione as a Target in the Design of Antitrypanosomal and Antileishmanial Agents
2001 · K. Augustyns, K. Amssoms, et al. · Current Pharmaceutical Design · 70
β-Secretase inhibitors: Modification at the P4 position and improvement of inhibitory activity in cultured cells
2006 · Yoshio Hamada, Naoto Igawa, et al. · Bioorganic & Medicinal Chemistry Letters · 51
Discovery and optimization of novel pyrazole-benzimidazole CPL304110, as a potent and selective inhibitor of fibroblast growth factor receptors FGFR (1–3)
2020 · Abdellah Yamani, Daria Zdżalik-Bielecka, et al. · European Journal of Medicinal Chemistry · 49
Novel non-peptidic and small-sized BACE1 inhibitors
2008 · Yoshio Hamada, Hiroko Ohta, et al. · Bioorganic & Medicinal Chemistry Letters · 44
BACE1 inhibitors: Optimization by replacing the P1′ residue with non-acidic moiety
2008 · Yoshio Hamada, Hamdy Abdel-Rahman, et al. · Bioorganic & Medicinal Chemistry Letters · 38
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1
2012 · Sabrina Castellano, Astrid Spannhoff, et al. · Journal of Medicinal Chemistry · 37
Significance of interactions of BACE1–Arg235 with its ligands and design of BACE1 inhibitors with P2 pyridine scaffold
2009 · Yoshio Hamada, Hiroko Ohta, et al. · Bioorganic & Medicinal Chemistry Letters · 36
Design of pentapeptidic BACE1 inhibitors with carboxylic acid bioisosteres at P1′ and P4 positions
2010 · Harichandra D. Tagad, Yoshio Hamada, et al. · Bioorganic & Medicinal Chemistry · 35
Views on Amyloid Hypothesis and Secretase Inhibitors for Treating Alzheimers Disease: Progress and Problems
2006 · Jeffrey-Tri Nguyen, Abdellah Yamani, et al. · Current Pharmaceutical Design · 35
Glutathione-like tripeptides as inhibitors of glutathionylspermidine synthetase. Part 1: Substitution of the glycine carboxylic acid group
2002 · Katie Amssoms, Sandra L Oza, et al. · Bioorganic & Medicinal Chemistry Letters · 22
PDF
Glutathione-like tripeptides as inhibitors of glutathionylspermidine synthetase. Part 2: Substitution of the glycine part
2002 · Katie Amssoms, Sandra L Oza, et al. · Bioorganic & Medicinal Chemistry Letters · 17
An Efficient Synthesis of Orthogonally Protected Spermidine
2002 · K. Amssoms, K. Augustyns, et al. · Synthetic Communications · 9
Preclinical characterization of CPL304110 as a potent and selective inhibitor of fibroblast growth factor receptors 1, 2, and 3 for gastric, bladder, and squamous cell lung cancer
2024 · Delfina Popiel, Aleksandra Stańczak, et al. · Frontiers in Oncology · 7
Identification of pyrrolo[2,3-d]pyrimidine-based dual MERTK and FLT3 inhibitor: Hit-to-lead, machine learning, modeling, synthesis, and biological evaluation
2026 · Abdellah Yamani, Paweł Maliszewski, et al. · European Journal of Pharmaceutical Sciences · 2
550P Preclinical characterization of CPL304110 as a potential selective inhibitor of fibroblast growth factors 1/2/3 in solid cancers
2020 · D. Popiel, A. Mikołajczyk, et al. · Annals of Oncology · 2
Corrigendum to “Significance of interactions of BACE1–Arg235 with its ligands and design of BACE1 inhibitors with P2 pyridine scaffold” [Bioorg. Med. Chem. Lett. 19 (2009) 2435]
2009 · Yoshio Hamada, Hiroko Ohta, et al. · Bioorganic & Medicinal Chemistry Letters · 2
Fast Claisen condensation reaction optimization in a continuous flow reactor
2023 · Stanisław Michałek, Antoni Powała, et al. · Monatshefte für Chemie - Chemical Monthly · 1
PDF
Preclinical evaluation of CPL423: a novel potent small-molecule inhibitor of TAM family and FLT3 kinase for cancer therapy
2026 · Agata Mikołajczyk, Delfina Popiel, et al. · Frontiers in Pharmacology
PDF
Significance of interaction of BACE1-Arg235 with its ligands and design of BACE1 inhibitors
2009 · Y. Hamada, Hiroko Ohta, et al. · Peptide science : proceedings of the ... Japanese Peptide Symposium
SAR study of BACE1 inhibitors containing pyridine derivatives
2009 · Hiroko Ohta, Y. Hamada, et al. · Peptide science : proceedings of the ... Japanese Peptide Symposium
Structure-Activity Relationship Study of BACE1 Inhibitors Containing Chelidonamide
2008 · Ryoji Yamaguchi, Y. Hamada, et al. · Peptide science : proceedings of the ... Japanese Peptide Symposium
Novel BACE1 Inhibitors : Design Approach Focused on Inhibitor's Conformer
2008 · Y. Hamada, Ryoji Yamaguchi, et al. · Peptide science : proceedings of the ... Japanese Peptide Symposium
Design of BACE1 Inhibitors : Replacing the P_1' Residue with Non-Acidic Moiety
2007 · Y. Hamada, Abdel-Rahman Hamdy, et al. · Peptide science : proceedings of the ... Japanese Peptide Symposium
ChemInform Abstract: An Efficient Synthesis of Orthogonally Protected Spermidine.
2002 · K. Amssoms, K. Augustyns, et al. · ChemInform
Works count: 24
Citation count: 457
H-index: 11
I10-index: 11
Year
Topic
Type