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Author

Antonio Quotadamo

Observed names: A. Quotadamo, Quotadamo, Antonio
Institution: IRBM
ORCID: 0000-0002-0357-3504
Observed ORCID: 0000-0002-0357-3504
OpenAlex ID: A5001825823
Computational and biological profile of boronic acids for the detection of bacterial serine- and metallo-β-lactamases
2017 · Matteo Santucci, Francesca Spyrakis, et al. · Scientific Reports · 44
Aryl thiosemicarbazones for the treatment of trypanosomatidic infections
2018 · Pasquale Linciano, Carolina B. Moraes, et al. · European Journal of Medicinal Chemistry · 41
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Enhancement of Benzothiazoles as Pteridine Reductase-1 Inhibitors for the Treatment of Trypanosomatidic Infections
2019 · Pasquale Linciano, Cecilia Pozzi, et al. · Journal of Medicinal Chemistry · 40
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X-ray Crystallography Deciphers the Activity of Broad-Spectrum Boronic Acid β-Lactamase Inhibitors
2019 · Laura Cendron, Antonio Quotadamo, et al. · ACS Medicinal Chemistry Letters · 39
Comparative mapping of on-targets and off-targets for the discovery of anti-trypanosomatid folate pathway inhibitors
2017 · Joanna Panecka-Hofman, Ina Pöhner, et al. · Biochimica et Biophysica Acta (BBA) - General Subjects · 30
Multitarget, Selective Compound Design Yields Potent Inhibitors of a Kinetoplastid Pteridine Reductase 1
2022 · Ina Pöhner, Antonio Quotadamo, et al. · Journal of Medicinal Chemistry · 25
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Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform
2019 · Carolina B. Moraes, Gesa Witt, et al. · SLAS DISCOVERY · 24
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An Improved Synthesis of CENTA, a Chromogenic Substrate for β-Lactamases
2016 · Maria Costi, Alberto Venturelli, et al. · Synlett · 18
Human Thymidylate Synthase Inhibitors Halting Ovarian Cancer Growth
2018 · Stefania Ferrari, Leda Severi, et al. · Vitamins and hormones · 17
High-Throughput Phenotypic Screening and Machine Learning Methods Enabled the Selection of Broad-Spectrum Low-Toxicity Antitrypanosomatidic Agents
2023 · Pasquale Linciano, Antonio Quotadamo, et al. · Journal of Medicinal Chemistry · 15
Destabilizers of the thymidylate synthase homodimer accelerate its proteasomal degradation and inhibit cancer growth
2022 · Luca Costantino, Stefania Ferrari, et al. · eLife · 15
New Insights into Bioactive Compounds from the Medicinal Plant Spathodea campanulata P. Beauv. and Their Activity against Helicobacter pylori
2020 · Corinne Raïssa Ngnameko, Lucia Marchetti, et al. · Antibiotics · 15
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First virtual screening and experimental validation of inhibitors targeting GES-5 carbapenemase
2019 · Francesca Spyrakis, Pierangelo Bellio, et al. · Journal of Computer-Aided Molecular Design · 15
Chapter Two - Scaffolds and Biological Targets Avenue to Fight Against Drug Resistance in Leishmaniasis
2018 · Chiara Borsari, Antonio Quotadamo, et al. · Annual reports in medicinal chemistry · 8
Structure–Property Optimization of a Series of Imidazopyridines for Visceral Leishmaniasis
2023 · Maria Dichiara, Quillon J. Simpson, et al. · ACS Infectious Diseases · 7
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An allosteric inhibitor of the Zika virus NS2B-NS3 protease with oral efficacy in mouse models
2026 · Jesus M. Ontoria, Esther Torrente, et al. · Nature Communications · 6
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Open Source Antibiotics: Simple Diarylimidazoles Are Potent against Methicillin-Resistant Staphylococcus aureus
2023 · Dana M. Klug, Edwin G. Tse, et al. · ACS Infectious Diseases · 6
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Optimization of N ‐alkylation in the Synthesis of Methotrexate and Pteridine‐based Derivatives Under Microwave‐Irradiation
2019 · Antonio Quotadamo, Pasquale Linciano, et al. · ChemistrySelect · 6
Scaffolds and Biological Targets Avenue to Fight Against Drug Resistance in Leishmaniasis
2018 · Chiara Borsari, Antonio Quotadamo, et al. · Annual reports in medicinal chemistry · 6
Pharmacophore Identification and Structure–Activity Relationship Analysis of a Series of Substituted Azaindoles as Inhibitors of Trypanosoma brucei
2024 · Lori Ferrins, Rosario Diaz, et al. · Journal of Medicinal Chemistry · 5
Identification of novel anti-amoebic pharmacophores from kinase inhibitor chemotypes
2023 · Lori Ferrins, Melissa J. Buskes, et al. · Frontiers in Microbiology · 4
Diastereoselective Synthesis of (1,3‐Dioxan‐4‐yl)pyrimidine and Purin Nucleoside Analogues
2015 · Umberto M. Battisti, Claudia Sorbi, et al. · European Journal of Organic Chemistry · 4
Corrigendum: Identification of novel anti-amoebic pharmacophores from kinase inhibitor chemotypes
2023 · Lori Ferrins, Melissa J. Buskes, et al. · Frontiers in Microbiology · 2
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Discovery and Optimization of IRBM-Z-2, an Allosteric Zika Virus NS2B-NS3 Protease Inhibitor Exhibiting In Vivo Efficacy
2026 · Esther Torrente, Antonio Quotadamo, et al. · Journal of Medicinal Chemistry
Author response: Destabilizers of the thymidylate synthase homodimer accelerate its proteasomal degradation and inhibit cancer growth
2022 · Luca Costantino, Stefania Ferrari, et al. · eLife
Works count: 34
Citation count: 392
H-index: 13
I10-index: 13
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