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Chiara Bosetti
Observed names:
BOSETTI, Chiara,
Bosetti, Chiara,
C. Bosetti
Institution:
University of Oulu
Observed institution:
University of Oulu
ORCID:
0000-0003-3809-7533
Observed ORCID:
0000-0003-3809-7533
OpenAlex ID:
A5003025895
An Evolutionary Perspective on the Origin, Conservation and Binding Partner Acquisition of Tankyrases
2022
·
Sven T. Sowa
, Chiara Bosetti
, et al.
·
Biomolecules
·
9
PDF
Substitutions at the C-8 position of quinazolin-4-ones improve the potency of nicotinamide site binding tankyrase inhibitors
2025
·
Chiara Bosetti
, Dionysis Kampasis
, et al.
·
European Journal of Medicinal Chemistry
·
5
Discovery of tankyrase scaffolding inhibitor specifically targeting the ARC4 peptide binding domain
2026
·
Chiara Bosetti
, Albert Galera-Prat
, et al.
·
Structure
·
2
Deconstruction of Dual-Site Tankyrase Inhibitors Provides Insights into Binding Energetics and Suggests Critical Hotspots for Ligand Optimization
2025
·
Sven T. Sowa
, Murat Kücükdisli
, et al.
·
Journal of Medicinal Chemistry
·
2
Optimization of 2,3-dihydrophthalazine-1,4-dione PARP inhibitor scaffold for nanomolar potency and specificity towards human PARP10
2025
·
Juho Alaviuhkola
, Maria Giulia Nizi
, et al.
·
European Journal of Medicinal Chemistry
·
1
Replacement soaking for human tankyrase 2 enables studies on substrate analogues and inhibitors
2026
·
Johan Pääkkönen
, Sven T. Sowa
, et al.
·
Acta Crystallographica Section D Structural Biology
Discovery of Fused Isoquinolinone/Triazole as a Scaffold for Tankyrase and PARP Inhibition
2025
·
Konstantinos A. Ouzounthanasis
, Chiara Bosetti
, et al.
·
Journal of Medicinal Chemistry
PDF
Re‐evaluation of PTEN as an ADP ‐ribosylated tankyrase binding partner
2025
·
Chiara Bosetti
, Albert Galera‐Prat
, et al.
·
FEBS Journal
Tankyrase 2 in complex with a quinazolin-4-one inhibitor
2024
·
C. Bosetti
, L. Lehtio
·
Worldwide Protein Data Bank
Substitutions at the C-8 Position of Quinazolin-4-Ones Improve the Potency of Nicotinamide Site Binding Tankyrase Inhibitors
2024
·
Ioannis K. Kostakis
, Chiara Bosetti
, et al.
·
SSRN Electronic Journal
Substitutions at the C-8 Position of Quinazolin-4-Ones Improve the Potency of Nicotinamide Site Binding Tankyrase Inhibitors
2024
·
Ioannis K. Kostakis
, Chiara Bosetti
, et al.
·
SSRN Electronic Journal
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Works count:
28
Citation count:
19
H-index:
2
I10-index:
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