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Hélène Adihou

New Modalities for Challenging Targets in Drug Discovery
2017 · Eric Valeur, Stéphanie M. Guéret, et al. · Angewandte Chemie International Edition · 384
TEAD–YAP Interaction Inhibitors and MDM2 Binders from DNA‐Encoded Indole‐Focused Ugi Peptidomimetics
2020 · Verena B. K. Kunig, Marco Potowski, et al. · Angewandte Chemie International Edition · 81
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Discovery of Covalent Inhibitors Targeting the Transcriptional Enhanced Associate Domain Central Pocket
2020 · Hacer Karatas, Mohammad Akbarzadeh, et al. · Journal of Medicinal Chemistry · 66
A straightforward method for automated Fmoc-based synthesis of bio-inspired peptide crypto-thioesters
2015 · Victor P. Terrier, Hélène Adihou, et al. · Chemical Science · 61
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Highly efficient solid phase synthesis of large polypeptides by iterative ligations of bis(2-sulfanylethyl)amido (SEA) peptide segments
2013 · Laurent Raibaut, Hélène Adihou, et al. · Chemical Science · 60
A protein tertiary structure mimetic modulator of the Hippo signalling pathway
2020 · Hélène Adihou, Ranganath Gopalakrishnan, et al. · Nature Communications · 58
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Selective Fluorescent Nonpeptidic Antagonists For Vasopressin V2GPCR: Application To Ligand Screening and Oligomerization Assays.
2012 · Stéphanie Loison, Martin Cottet, et al. · Journal of Medicinal Chemistry · 57
Structure, Biosynthesis, and Occurrence of Bacterial Pyrrolizidine Alkaloids
2015 · Olivia Schimming, Victoria L. Challinor, et al. · Angewandte Chemie International Edition · 50
Neue Modalitäten für schwierige Zielstrukturen in der Wirkstoffentwicklung
2017 · Eric Valeur, Stéphanie M. Guéret, et al. · Angewandte Chemie · 40
Biosynthesis of the Antibiotic Nematophin and Its Elongated Derivatives in Entomopathogenic Bacteria
2017 · Xiaofeng Cai, Victoria L. Challinor, et al. · Organic Letters · 34
Structure Based Design of Bicyclic Peptide Inhibitors of RbAp48
2020 · Peter 't Hart, Pascal Hommen, et al. · Angewandte Chemie International Edition · 31
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Biochemical Investigation of the Interaction of pICln, RioK1 and COPR5 with the PRMT5–MEP50 Complex
2021 · Adrian Krzyzanowski, Raphael Gasper, et al. · ChemBioChem · 29
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Robust Prediction of Relative Binding Energies for Protein–Protein Complex Mutations Using Free Energy Perturbation Calculations
2024 · Jared M. Sampson, Daniel A. Cannon, et al. · Journal of Molecular Biology · 24
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Molecular mechanism of polyketide shortening in anthraquinone biosynthesis of Photorhabdus luminescens
2019 · Qiuqin Zhou, Alois Bräuer, et al. · Chemical Science · 23
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Synthesis of Peptides by Reactive Extrusion. Application to the Continuous and Solventless Preparation of Aspartame.
2024 · Tharwat Mohy El‐Dine, Matthieu Lavayssiere, et al. · ChemistryEurope · 18
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Solid‐Phase Enrichment and Analysis of Azide‐Labeled Natural Products: Fishing Downstream of Biochemical Pathways
2015 · Alexander J. Pérez, Frank Wesche, et al. · Chemistry - A European Journal · 15
TEAD–YAP Interaction Inhibitors and MDM2 Binders from DNA‐Encoded Indole‐Focused Ugi Peptidomimetics
2020 · Verena B. K. Kunig, Marco Potowski, et al. · Angewandte Chemie · 13
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Structure, Biosynthesis, and Occurrence of Bacterial Pyrrolizidine Alkaloids
2015 · Olivia Schimming, Victoria L. Challinor, et al. · Angewandte Chemie · 11
Lipidated Stapled Peptides Targeting the Acyl Binding Protein UNC119
2019 · Philipp M. Cromm, Hélène Adihou, et al. · ChemBioChem · 10
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Combined Approach of Backbone Amide Linking and On-Resin N-Methylation for the Synthesis of Bioactive and Metabolically Stable Peptides
2018 · Frank Wesche, Hélène Adihou, et al. · Journal of Medicinal Chemistry · 7
Hot-spot guided design of macrocyclic inhibitors of the LSD1-CoREST1 interaction
2019 · Peter ‘T Hart, Joseph Openy, et al. · Tetrahedron · 6
Combining Real-Time Monitoring Using Raman Spectroscopy, Rotating-Bed Reactors, and Green Solvents to Improve Sustainability in Solid-Phase Peptide Synthesis
2024 · Eugenie Fournier, Arjun Vijeta, et al. · ACS Sustainable Chemistry & Engineering · 4
Synthesis and SAR of the antistaphylococcal natural product nematophin from Xenorhabdus nematophila
2019 · Frank Wesche, Hélène Adihou, et al. · Beilstein Journal of Organic Chemistry · 4
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Structure Based Design of Bicyclic Peptide Inhibitors of RbAp48
2020 · Peter 't Hart, Pascal Hommen, et al. · Angewandte Chemie · 2
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Cover Feature: Lipidated Stapled Peptides Targeting the Acyl Binding Protein UNC119 (ChemBioChem 24/2019)
2019 · Philipp M. Cromm, Hélène Adihou, et al. · ChemBioChem · 1
Works count: 33
Citation count: 1,093
H-index: 15
I10-index: 19
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