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Markus Pietsch

Synthesis of Tricyclic 1,3-Oxazin-4-ones and Kinetic Analysis of Cholesterol Esterase and Acetylcholinesterase Inhibition
2005 · Markus Pietsch, Michael Gütschow · Journal of Medicinal Chemistry · 106
2-(Diethylamino)thieno[1,3]oxazin-4-ones as Stable Inhibitors of Human Leukocyte Elastase
1999 · Michael Gütschow, Lars Kuerschner, et al. · Journal of Medicinal Chemistry · 93
Compatible solutes as protectants for zymogens against proteolysis
2006 · Sonja Kolp, Markus Pietsch, et al. · Biochimica et Biophysica Acta (BBA) - Proteins and Proteomics · 77
Calpains: Attractive Targets for the Development of Synthetic Inhibitors
2010 · Markus Pietsch, Krystle Chua, et al. · Current Topics in Medicinal Chemistry · 67
Alternate Substrate Inhibition of Cholesterol Esterase by Thieno[2,3-d][1,3]oxazin-4-ones
2002 · Markus Pietsch, Michael Gütschow · Journal of Biological Chemistry · 64
Activated microglia/macrophage whey acidic protein (AMWAP) inhibits NFκB signaling and induces a neuroprotective phenotype in microglia
2015 · Alexander Aslanidis, Marcus Karlstetter, et al. · Journal of Neuroinflammation · 54
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New cholesterol esterase inhibitors based on rhodanine and thiazolidinedione scaffolds
2011 · Sabrina Heng, William Tieu, et al. · Bioorganic & Medicinal Chemistry · 47
Tissue transglutaminase: An emerging target for therapy and imaging
2013 · Markus Pietsch, Robert Wodtke, et al. · Bioorganic & Medicinal Chemistry Letters · 45
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First Structure of Protein Kinase CK2 Catalytic Subunit with an Effective CK2β-Competitive Ligand
2013 · Jennifer Raaf, Barbara Guerra, et al. · ACS Chemical Biology · 44
Multiple Ligands in Opioid Research
2008 · Steven Ballet, Markus Pietsch, et al. · Protein and Peptide Letters · 41
Chromenones as Multineurotargeting Inhibitors of Human Enzymes
2019 · Carina Lemke, Joscha Christmann, et al. · ACS Omega · 38
Kinetics of inhibition of acetylcholinesterase in the presence of acetonitrile
2009 · Markus Pietsch, Leonie Christian, et al. · FEBS Journal · 37
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Nε-Acryloyllysine Piperazides as Irreversible Inhibitors of Transglutaminase 2: Synthesis, Structure–Activity Relationships, and Pharmacokinetic Profiling
2018 · Robert Wodtke, Christoph Hauser, et al. · Journal of Medicinal Chemistry · 36
Macrocyclic Protease Inhibitors with Reduced Peptide Character
2014 · Krystle C. H. Chua, Markus Pietsch, et al. · Angewandte Chemie International Edition · 33
Regioselective Sulfonylation and N- to O-Sulfonyl Migration of Quinazolin-4(3H)-ones and Analogous Thienopyrimidin-4(3H)-ones
2013 · Matthias D. Mertens, Markus Pietsch, et al. · The Journal of Organic Chemistry · 32
Synthesis and Extended Activity of Triazole‐Containing Macrocyclic Protease Inhibitors
2013 · Ashok D. Pehere, Markus Pietsch, et al. · Chemistry - A European Journal · 30
Selective Inhibitors of Glutathione Transferase P1 with Trioxane Structure as Anticancer Agents
2015 · Maria Bräutigam, Nicole Teusch, et al. · ChemMedChem · 28
2,4,5-Triphenylisothiazol-3(2H)-one 1,1-dioxides as inhibitors of human leukocyte elastase
2005 · Michael Gütschow, Markus Pietsch, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 28
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Development of an 18F-Labeled Irreversible Inhibitor of Transglutaminase 2 as Radiometric Tool for Quantitative Expression Profiling in Cells and Tissues
2021 · Robert Wodtke, Johanna Wodtke, et al. · Journal of Medicinal Chemistry · 27
Unexpected CK2β-antagonistic functionality of bisubstrate inhibitors targeting protein kinase CK2
2020 · Markus Pietsch, Kaido Viht, et al. · Bioorganic Chemistry · 24
The intracellular Ca 2+ -homeostasis influences the frequency-dependent force-generation in man
1999 · K. Brixius, M. Pietsch, et al. · Basic Research in Cardiology · 22
Design of CK2β‐Mimicking Peptides as Tools To Study the CK2α/CK2β Interaction in Cancer Cells
2019 · Dirk Lindenblatt, Mareike Horn, et al. · ChemMedChem · 21
Development of a high-throughput screening-compatible assay to identify inhibitors of the CK2α/CK2β interaction
2014 · Jennifer Hochscherf, Dirk Lindenblatt, et al. · Analytical Biochemistry · 20
Cholesterol esterase action on human high density lipoproteins and inhibition studies: detection by MALDI-TOF MS
2005 · Olaf Zschörnig, Markus Pietsch, et al. · Journal of Lipid Research · 20
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Direct, gabapentin-insensitive interaction of a soluble form of the calcium channel subunit α2δ-1 with thrombospondin-4
2019 · Ehab El-Awaad, Galyna Pryymachuk, et al. · Scientific Reports · 17
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Works count: 103
Citation count: 1,245
H-index: 21
I10-index: 33
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