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Pablo García‐Losada

Observed names: García-Losada, Pablo, P. Garcia‐Losada, Pablo Garcia Losada, Pablo Garcia-Losada, Pablo Garcia‐Losada, Pablo García-Losada, Pablo García Losada, Pablo García-Losada
ORCID: 0000-0002-8307-0033
Observed ORCID: 0000-0002-8307-0033
OpenAlex ID: A5015541674
The Evolution of High-Throughput Experimentation in Pharmaceutical Development and Perspectives on the Future
2019 · Steven M. Mennen, Carolina Alhambra, et al. · Organic Process Research & Development · 542
Decatungstate‐Mediated C(sp3)–H Heteroarylation via Radical‐Polar Crossover in Batch and Flow
2021 · Ting Wan, Luca Capaldo, et al. · Angewandte Chemie International Edition · 113
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The Merger of Benzophenone HAT Photocatalysis and Silyl Radical-Induced XAT Enables Both Nickel-Catalyzed Cross-Electrophile Coupling and 1,2-Dicarbofunctionalization of Olefins
2022 · Alberto Luridiana, Daniele Mazzarella, et al. · ACS Catalysis · 76
Accelerated and Scalable C(sp 3 )–H Amination via Decatungstate Photocatalysis Using a Flow Photoreactor Equipped with High-Intensity LEDs
2021 · Ting Wan, Zhenghui Wen, et al. · ACS Central Science · 75
Electrochemical Nickel-Catalyzed C(sp3)–C(sp3) Cross-Coupling of Alkyl Halides with Alkyl Tosylates
2023 · Malek Y. S. Ibrahim, Graham R. Cumming, et al. · Journal of the American Chemical Society · 67
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Continuous stirred-tank reactor cascade platform for self-optimization of reactions involving solids
2022 · Kakasaheb Y. Nandiwale, Travis Hart, et al. · Reaction Chemistry & Engineering · 49
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2-Chloro-4-[[(1R,2R)-2-hydroxy-2-methyl-cyclopentyl]amino]-3-methyl-benzonitrile: A Transdermal Selective Androgen Receptor Modulator (SARM) for Muscle Atrophy
2015 · Ashraf Saeed, Grant M. Vaught, et al. · Journal of Medicinal Chemistry · 39
Discovery and Early Clinical Development of LY3202626, a Low-Dose, CNS-Penetrant BACE Inhibitor
2021 · David L. McKinzie, Leonard L. Winneroski, et al. · Journal of Medicinal Chemistry · 31
Development of a selective androgen receptor modulator for transdermal use in hypogonadal patients
2018 · V. Krishnan, N. J. Patel, et al. · Andrology · 22
Preparation and biological evaluation of BACE1 inhibitors: Leveraging trans-cyclopropyl moieties as ligand efficient conformational constraints
2019 · Leonard L. Winneroski, Jon A. Erickson, et al. · Bioorganic & Medicinal Chemistry · 19
Preparation and biological evaluation of conformationally constrained BACE1 inhibitors
2015 · Leonard L. Winneroski, Matthew A. Schiffler, et al. · Bioorganic & Medicinal Chemistry · 18
Large-Scale Continuous Flow Transformation of Oximes into Fused-Bicyclic Isoxazolidines: An Example of Process Intensification
2015 · Juan A. Rincón, Carlos Mateos, et al. · Organic Process Research & Development · 18
Synthesis of new fluorophores derived from monoazacrown ethers and coumarin nucleus
2002 · Ernesto Brunet, Pablo García-Losada, et al. · Canadian Journal of Chemistry · 18
Scale-up of N -alkylation reaction using phase-transfer catalysis with integrated separation in flow
2018 · María José Nieves-Remacha, Myriam Torres, et al. · Reaction Chemistry & Engineering · 13
Synthesis, Optimization, and Large-Scale Preparation of the Low-Dose Central Nervous System-Penetrant BACE1 Inhibitor LY3202626 via a [3 + 2] Nitrone Cycloaddition
2020 · Pablo Garcia-Losada, Amy C. DeBaillie, et al. · Organic Process Research & Development · 12
Continuous-Flow Supercritical CO 2 Platform for In-Situ Synthesis and Purification of Small Molecules for Drug Discovery
2023 · Sergio Alcalde, Raúl Porcar, et al. · Organic Process Research & Development · 11
Synthesis of a novel series of 4,4-disubstituted 2,3,4,7-tetrahydroazepines
2005 · Mario Barberis, Pablo García-Losada, et al. · Tetrahedron Letters · 11
An Integrated 12 C/ 13 C Exchange Platform for Accessing Isotopically-Labeled Ketones via Dual Catalytic C–C Bond-Functionalization
2025 · Hui-Qing Geng, Álvaro Velasco-Rubio, et al. · ACS Catalysis · 10
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Practical Asymmetric Fluorination Approach to the Scalable Synthesis of New Fluoroaminothiazine BACE Inhibitors
2018 · Pablo Garcia-Losada, Mario Barberis, et al. · Organic Process Research & Development · 10
Practical Manufacture of 4-Alkyl-4-aminocyclohexylalcohols Using Ketoreductases
2017 · Susana García-Cerrada, Laura Redondo-Gallego, et al. · Organic Process Research & Development · 10
Design of Experiments-Based Optimization of an Electrochemical Decarboxylative Alkylation Using a Spinning Cylinder Electrode Reactor
2024 · Nikola Petrović, Graham R. Cumming, et al. · Organic Process Research & Development · 8
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Multigram Synthesis of Chiral Cyclopropane Carboxylic Acids via Tandem Diastereoselective Wadsworth–Emmons Cyclopropanation-Hydrolysis in Continuous Flow
2024 · Carlos Mateos, Susana García-Cerrada, et al. · Organic Process Research & Development · 5
Decatungstate‐Mediated C(sp3)–H Heteroarylation via Radical‐Polar Crossover in Batch and Flow
2021 · Ting Wan, Luca Capaldo, et al. · Angewandte Chemie · 5
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Flow photochemical Giese reaction via silane-mediated activation of alkyl bromides
2023 · Fabiola Fanini, Alberto Luridiana, et al. · Tetrahedron Letters · 4
Evolution of Synthetic Strategies for Lilly’s Clinical BACE Inhibitors: From Discovery Concepts to Manufacturing-Ready Routes
2026 · Michael O. Frederick, Pablo Garcia-Losada, et al. · Organic Process Research & Development
Works count: 31
Citation count: 1,186
H-index: 13
I10-index: 20
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