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Author

Gianfranco Battistuzzi

Observed names: Battistuzzi, Gianfranco, G. Battistuzzi
Institution: Alfasigma (Italy)
ORCID: 0000-0001-9538-7516
Observed ORCID: 0000-0001-9538-7516
OpenAlex ID: A5015947111
The Aminopalladation/Reductive Elimination Domino Reaction in the Construction of Functionalized Indole Rings
2002 · Gianfranco Battistuzzi, Sandro Cacchi, et al. · European Journal of Organic Chemistry · 245
An Efficient Palladium-Catalyzed Synthesis of Cinnamaldehydes from Acrolein Diethyl Acetal and Aryl Iodides and Bromides
2003 · Gianfranco Battistuzzi, Sandro Cacchi, et al. · Organic Letters · 150
An Efficient Palladium‐Catalyzed Synthesis of Cinnamaldehydes from Acrolein Diethyl Acetal and Aryl Iodides and Bromides.
2003 · Gianfranco Battistuzzi, Sandro Cacchi, et al. · ChemInform · 114
4‐Aryl‐2‐quinolones through a Pseudo‐Domino Heck/Buchwald–Hartwig Reaction in a Molten Tetrabutylammonium Acetate/ Tetrabutylammonium Bromide Mixture
2007 · Gianfranco Battistuzzi, Roberta Bernini, et al. · Advanced Synthesis & Catalysis · 75
Non-Natural Macrocyclic Inhibitors of Histone Deacetylases: Design, Synthesis, and Activity
2010 · Luciana Auzzas, Andreas Larsson, et al. · Journal of Medicinal Chemistry · 66
Synthesis of Coumarins in a Molten n‐Bu4NOAc/n‐Bu4NBr Mixture through a Domino Heck Reaction/Cyclization Process
2005 · Gianfranco Battistuzzi, Sandro Cacchi, et al. · Advanced Synthesis & Catalysis · 53
12-Acylindolo[1,2-c]quinazolines by Palladium-Catalyzed Cyclocarbonylation of o-Alkynyltrifluoroacetanilides
2002 · Gianfranco Battistuzzi, Sandro Cacchi, et al. · Organic Letters · 53
Exploring bis-(indolyl)methane moiety as an alternative and innovative CAP group in the design of histone deacetylase (HDAC) inhibitors
2009 · Giuseppe Giannini, Mauro Marzi, et al. · Bioorganic & Medicinal Chemistry Letters · 52
Epoxidation of chromones and flavonoids in ionic liquids
2003 · Roberta Bernini, Enrico Mincione, et al. · Tetrahedron · 49
ST7612AA1, a Thioacetate-ω(γ-lactam carboxamide) Derivative Selected from a Novel Generation of Oral HDAC Inhibitors
2014 · Giuseppe Giannini, Loredana Vesci, et al. · Journal of Medicinal Chemistry · 48
Hydroxamic acid based histone deacetylase inhibitors with confirmed activity against the malaria parasite
2014 · Giuseppe Giannini, Gianfranco Battistuzzi, et al. · Bioorganic & Medicinal Chemistry Letters · 45
N-Hydroxy-(4-oxime)-cinnamide: A versatile scaffold for the synthesis of novel histone deacetilase (HDAC) inhibitors
2009 · Giuseppe Giannini, Mauro Marzi, et al. · Bioorganic & Medicinal Chemistry Letters · 42
Antibody drug conjugates (ADCs) charged with HDAC inhibitor for targeted epigenetic modulation
2018 · Elena Cini, Valentina Faltoni, et al. · Chemical Science · 39
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Novel PARP-1 inhibitors based on a 2-propanoyl-3H-quinazolin-4-one scaffold
2013 · Giuseppe Giannini, Gianfranco Battistuzzi, et al. · Bioorganic & Medicinal Chemistry Letters · 37
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Novel Benzazole Derivatives Endowed with Potent Antiheparanase Activity
2018 · Valentina Noemi Madia, Antonella Messore, et al. · Journal of Medicinal Chemistry · 35
A Molten n-Bu4NOAc/n-Bu4NBr Mixture as an Efficient Medium for the Stereoselective Synthesis of (E)- and (Z)-3,3-Diarylacrylates
2002 · Gianfranco Battistuzzi, Sandro Cacchi, et al. · Synlett · 30
Novel Symmetrical Benzazolyl Derivatives Endowed with Potent Anti-Heparanase Activity
2018 · Antonella Messore, Valentina Noemi Madia, et al. · Journal of Medicinal Chemistry · 25
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Lactam based 7-amino suberoylamide hydroxamic acids as potent HDAC inhibitors
2013 · Maurizio Taddei, Elena Cini, et al. · Bioorganic & Medicinal Chemistry Letters · 25
Human inhalable antibody fragments neutralizing SARS-CoV-2 variants for COVID-19 therapy
2022 · Olga Minenkova, Daniela Santapaola, et al. · Molecular Therapy · 24
ErbB2 Targeted Epigenetic Modulation: Anti-tumor Efficacy of the ADC Trastuzumab-HDACi ST8176AA1
2020 · Ferdinando Maria Milazzo, Loredana Vesci, et al. · Frontiers in Oncology · 20
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Antibody drug conjugates with hydroxamic acid cargos for histone deacetylase (HDAC) inhibition
2021 · Claudio Cianferotti, Valentina Faltoni, et al. · Chemical Communications · 18
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Exploring in vitro and in vivo Hsp90 inhibitors activity against human protozoan parasites
2014 · Giuseppe Giannini, Gianfranco Battistuzzi · Bioorganic & Medicinal Chemistry Letters · 17
4,5,6,7-Tetrahydro-isoxazolo-[4,5-c]-pyridines as a new class of cytotoxic Hsp90 inhibitors
2014 · Riccardo Baruchello, Daniele Simoni, et al. · European Journal of Medicinal Chemistry · 17
New classes of potent heparanase inhibitors from ligand-based virtual screening
2020 · Daniele Pala, Laura Scalvini, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 15
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New retinoid derivatives as back-ups of Adarotene
2012 · Giuseppe Giannini, Tiziana Brunetti, et al. · Bioorganic & Medicinal Chemistry · 14
Works count: 52
Citation count: 1,375
H-index: 20
I10-index: 28
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