Get started
Author

Jeffrey C. Pelletier

Observed names: J. C. PELLETIER, Jeffrey C Pelletier, Jeffrey Pelletier, Pelletier Jeffrey C. Pelletier Jeffrey C.
Observed institutions: Northwestern University, DuPont (United States), University of Alabama, Fox Chase Chemical Diversity Center, Wyeth, University of Pennsylvania
ORCID: 0000-0002-0397-0681
Observed ORCID: 0000-0002-0397-0681
OpenAlex ID: A5017508406
Improved Solid-Phase Peptide Synthesis Method Utilizing α-Azide-Protected Amino Acids
2001 · Lundquist, Jeffrey C. Pelletier · Organic Letters · 196
Tricyclic ureas: A new class of HIV-1 protease inhibitors
1998 · Wei Han, Jeffrey C. Pelletier, et al. · Bioorganic & Medicinal Chemistry Letters · 106
Targeting Human Central Nervous System Protein Kinases: An Isoform Selective p38αMAPK Inhibitor That Attenuates Disease Progression in Alzheimer’s Disease Mouse Models
2015 · Saktimayee M. Roy, Valerie L. Grum-Tokars, et al. · ACS Chemical Neuroscience · 100
Substituted 1,2-Dihydrophthalazines: Potent, Selective, and Noncompetitive Inhibitors of the AMPA Receptor
1996 · Jeffrey C. Pelletier, David P. Hesson, et al. · Journal of Medicinal Chemistry · 93
Development of Novel In Vivo Chemical Probes to Address CNS Protein Kinase Involvement in Synaptic Dysfunction
2013 · D. Martin Watterson, Valerie L. Grum-Tokars, et al. · PLoS ONE · 80
PDF
Synthesis, Resolution, and Biological Evaluation of the Four Stereoisomers of 4-Methylglutamic Acid: Selective Probes of Kainate Receptors
1995 · Zi-Qiang Gu, David P. Hesson, et al. · Journal of Medicinal Chemistry · 74
A Selective and Brain Penetrant p38αMAPK Inhibitor Candidate for Neurologic and Neuropsychiatric Disorders That Attenuates Neuroinflammation and Cognitive Dysfunction
2019 · Saktimayee M. Roy, George Minasov, et al. · Journal of Medicinal Chemistry · 60
PDF
Synthesis of the marine alkaloids aaptamine and demethyloxyaaptamine and of the parent structure didemethoxyaaptamine
1987 · Jeffrey C. Pelletier, Michael P. Cava · The Journal of Organic Chemistry · 58
Mitsunobu reaction modifications allowing product isolation without chromatography: application to a small parallel library
2000 · Jeffrey C. Pelletier, Scott Kincaid · Tetrahedron Letters · 57
(1-(4-(Naphthalen-2-yl)pyrimidin-2-yl)piperidin-4-yl)methanamine: A Wingless β-Catenin Agonist That Increases Bone Formation Rate
2009 · Jeffrey C. Pelletier, Joseph T. Lundquist, et al. · Journal of Medicinal Chemistry · 52
Identification of Clinically Viable Quinolinol Inhibitors of Botulinum Neurotoxin A Light Chain
2014 · Dejan Caglič, Michelle C. Krutein, et al. · Journal of Medicinal Chemistry · 49
PDF
A New Tri-Orthogonal Strategy for Peptide Cyclization
2002 · Lundquist, Jeffrey C. Pelletier · Organic Letters · 47
Novel (4-Piperidin-1-yl)-phenyl Sulfonamides as Potent and Selective Human β3 Agonists
2001 · Baihua Hu, John Ellingboe, et al. · Bioorganic & Medicinal Chemistry · 44
Enhanced Parallel Synthesis Efficiency through Tandem Pd-Catalyzed S- and N-Arylation Reactions: Single-Vessel Formation of Aminobenzothiazoles
2007 · Matthew D. Vera, Jeffrey C. Pelletier · Journal of Combinatorial Chemistry · 38
GnRH Agonists and Antagonists in Cancer Therapy
2003 · Murty Chengalvala, Jeffrey Pelletier, et al. · Anti-Cancer Agents in Medicinal Chemistry · 36
Mild and Adaptable Silver Triflate-Assisted Method for Trityl Protection of Alcohols in Solution with Solid-Phase Loading Applications
2006 · Lundquist, Andrew D. Satterfield, et al. · Organic Letters · 34
Riluzole prodrugs for melanoma and ALS: Design, synthesis, and in vitro metabolic profiling
2012 · Mark E. McDonnell, Matthew D. Vera, et al. · Bioorganic & Medicinal Chemistry · 30
Preparation of highly substituted γ-lactam follicle stimulating hormone receptor agonists
2005 · Jeffrey C. Pelletier, John Rogers, et al. · Bioorganic & Medicinal Chemistry · 30
2-Phenyl-4-piperazinylbenzimidazoles: Orally active inhibitors of the gonadotropin releasing hormone (GnRH) receptor
2008 · Jeffrey C. Pelletier, Murty Chengalvala, et al. · Bioorganic & Medicinal Chemistry · 29
7-Azabicycloheptane Carboxylic Acid: A Proline Replacement in a Boroarginine Thrombin Inhibitor
1999 · Wei Han, Jeffrey C. Pelletier, et al. · Organic Letters · 28
The Reaction of 3,4-Dihydroisoquinolines With Malonic Acid and Its Derivatives
1987 · Jeffrey C. Pelletier, Michael P. Cava · Synthesis · 24
Preparation of amides from acids and resin bound azides: Suppression of intramolecular lactam formation
1998 · Zhilian Tang, Jeffrey C. Pelletier · Tetrahedron Letters · 20
Synthesis of aaptamine, a novel marine alkaloid
1985 · Jeffrey C. Pelletier, Michael P. Cava · Tetrahedron Letters · 19
A Mild Preparation of Amino Acid N-Acylsulfonamides
1995 · Jeffrey C. Pelletier, David P. Hesson · Synlett · 18
Dipeptide Prodrugs of the Glutamate Modulator Riluzole
2018 · Jeffrey C. Pelletier, Suzie Chen, et al. · ACS Medicinal Chemistry Letters · 17
Works count: 57
Citation count: 1,461
H-index: 21
I10-index: 29
Year
Topic
Type