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Masahiro Sakaitani

dl-threo-β-Benzyloxyaspartate, A Potent Blocker of Excitatory Amino Acid Transporters
1998 · Keiko Shimamoto, Bruno Lebrun, et al. · Molecular Pharmacology · 547
Syntheses and reactions of silyl carbamates. 1. Chemoselective transformation of amino protecting groups via tert-butyldimethylsilyl carbamates
1990 · Masahiro Sakaitani, Yasufumi Ohfune · The Journal of Organic Chemistry · 275
Molecular studies on enzymes in chorismate metabolism and the enterobactin biosynthetic pathway
1990 · Christopher T. Walsh, Jun Liu, et al. · Chemical Reviews · 214
Biosynthesis of the Escherichia coli siderophore enterobactin: sequence of the entF gene, expression and purification of EntF, and analysis of covalent phosphopantetheine
1991 · Frank Rusnak, Masahiro Sakaitani, et al. · Biochemistry · 147
Selective transformation of N--butoxycarbonyl group into n-alkoxy-carbonyl group n-carboxylate ion equivalent
1985 · Masahiro Sakaitani, Yasufumi Ohfune · Tetrahedron Letters · 103
Design, synthesis and antifungal activity of a novel water soluble prodrug of antifungal triazole
2003 · Jun Ohwada, Masao Tsukazaki, et al. · Bioorganic & Medicinal Chemistry Letters · 87
New β-Hydroxyaspartate Derivatives Are Competitive Blockers for the Bovine Glutamate/Aspartate Transporter
1997 · Bruno Lebrun, Masahiro Sakaitani, et al. · Journal of Biological Chemistry · 72
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Pavoninins: Shark-Repelling Ichthyotoxins from the Defense Secretion of the Pacific Sole
1984 · Kazuo Tachibana, Masahiro Sakaitani, et al. · Science · 70
An efficient route to 1,3-amino hydroxyl system via electrophilic lactonization of 2-amino-4-pentenoic acid derivatives. Stereoselective synthesis of (−)-bulgecinine
1986 · Yasufumi Ohfune, Keiko Hori, et al. · Tetrahedron Letters · 69
Pavoninins, shark-repelling and ichthyotoxic steroid n-acetylglucosaminides from the defense secretion of the sole pardachirus pavoninus (soleidae)
1985 · Kazuo Tachibana, Masahiro Sakaitani, et al. · Tetrahedron · 68
One-pot conversion of N-benzyloxycarbonyl group into N-tert-butoxycarbonyl group
1988 · Masahiro Sakaitani, Keiko Hori, et al. · Tetrahedron Letters · 65
Syntheses and reactions of silyl carbamates. 2. A new mode of cyclic carbamate formation from tert-butyldimethylsilyl carbamate
1990 · Masahiro Sakaitani, Yasufumi Ohfune · Journal of the American Chemical Society · 62
Synthesis of riccardin B by nickel-catalyzed intramolecular cyclization
1985 · Masahiko Iyoda, Masahiro Sakaitani, et al. · Tetrahedron Letters · 48
Characterization of EntF as a serine‐activating enzyme
1992 · Janice Reichert, Masahiro Sakaitani, et al. · Protein Science · 45
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Suramin, screened from an approved drug library, inhibits HuR functions and attenuates malignant phenotype of oral cancer cells
2018 · Wataru Kakuguchi, Takao Nomura, et al. · Cancer Medicine · 44
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Mechanistic studies on trans-2,3-dihydro-2,3-dihydroxybenzoate dehydrogenase (Ent A) in the biosynthesis of the iron chelator enterobactin
1990 · Masahiro Sakaitani, Frank Rusnak, et al. · Biochemistry · 44
Synthesis and structure–activity relationships of novel benzofuran farnesyltransferase inhibitors
2009 · Kohsuke Asoh, Masami Kohchi, et al. · Bioorganic & Medicinal Chemistry Letters · 41
N-carboxylate ion equivalent. II. Novel transformations of N-benzyloxycarbonyl (Z) group and N-allyloxycarbonyl group into N--butyldimethylsilyloxycarbonyl intermediate
1986 · Masahiro Sakaitani, Natsuko Kurokawa, et al. · Tetrahedron Letters · 40
Fluorine Scanning by Nonselective Fluorination: Enhancing Raf/MEK Inhibition while Keeping Physicochemical Properties
2013 · Ikumi Hyohdoh, Noriyuki Furuichi, et al. · ACS Medicinal Chemistry Letters · 39
A new mode of cyclic carbamate formation via tert-butyldimethylsilyl carbamate. Stereoselective syntheses of statine and its analogue
1987 · Masahiro Sakaitani, Yasufumi Ohfune · Tetrahedron Letters · 38
Piperazine Propanol Derivative as a Novel Antifungal Targeting 1,3-.BETA.-D-Glucan Synthase
2005 · Osamu Kondoh, Yukiko Inagaki, et al. · Biological and Pharmaceutical Bulletin · 31
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Optimizing the Physicochemical Properties of Raf/MEK Inhibitors by Nitrogen Scanning
2014 · Toshihiro Aoki, Ikumi Hyohdoh, et al. · ACS Medicinal Chemistry Letters · 26
New and efficient dehalogenative coupling and reduction of α-haloketones with active nickel complex. Facile syntheses of 1,4-diketones and bicyclo[4.2.O]oct-3-ene-2,5-diones
1985 · Masahiko Iyoda, Masahiro Sakaitani, et al. · Tetrahedron Letters · 26
Cloning and expression of a bovine glutamate transporter
1995 · Kiyoshi Inoue, Masahiro Sakaitani, et al. · Molecular Brain Research · 22
The sulfamide moiety affords higher inhibitory activity and oral bioavailability to a series of coumarin dual selective RAF/MEK inhibitors
2013 · Toshihiro Aoki, Ikumi Hyohdoh, et al. · Bioorganic & Medicinal Chemistry Letters · 21
Works count: 48
Citation count: 2,318
H-index: 23
I10-index: 28
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