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Caroline Joannesse

Observed names: C. Joannesse, Joannesse, C., Joannesse, Caroline
Institution: Galapagos (Belgium)
ORCID: 0000-0002-9548-5439
Observed ORCID: 0000-0002-9548-5439
OpenAlex ID: A5022161528
Isothiourea‐Catalyzed Enantioselective Carboxy Group Transfer
2009 · Caroline Joannesse, Craig P. Johnston, et al. · Angewandte Chemie International Edition · 201
Structure-enantioselectivity effects in 3,4-dihydropyrimido[2,1-b]benzothiazole-based isothioureas as enantioselective acylation catalysts
2010 · Dorine Belmessieri, Caroline Joannesse, et al. · Organic & Biomolecular Chemistry · 103
Discovery ofN-(3-Carbamoyl-5,5,7,7-tetramethyl-5,7-dihydro-4H-thieno[2,3-c]pyran-2-yl)-lH-pyrazole-5-carboxamide (GLPG1837), a Novel Potentiator Which Can Open Class III Mutant Cystic Fibrosis Transmembrane Conductance Regulator (CFTR) Channels to a High Extent
2017 · Steven E. Van der Plas, Hans Kelgtermans, et al. · Journal of Medicinal Chemistry · 65
Nucleophilicities and Lewis Basicities of Isothiourea Derivatives
2011 · Biplab Maji, Caroline Joannesse, et al. · The Journal of Organic Chemistry · 64
Isothiourea‐Catalyzed Enantioselective Carboxy Group Transfer
2009 · Caroline Joannesse, Craig P. Johnston, et al. · Angewandte Chemie · 48
Amidine catalysed O- to C-carboxyl transfer of heterocyclic carbonate derivatives
2008 · Caroline Joannesse, Carmen Simal, et al. · Organic & Biomolecular Chemistry · 40
Isothiourea‐Mediated Asymmetric O‐ to C‐Carboxyl Transfer of Oxazolyl Carbonates: Structure–Selectivity Profiles and Mechanistic Studies
2012 · Caroline Joannesse, Craig P. Johnston, et al. · Chemistry - A European Journal · 36
Discovery of the S1P2 Antagonist GLPG2938 (1-[2-Ethoxy-6-(trifluoromethyl)-4-pyridyl]-3-[[5-methyl-6-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]pyridazin-3-yl]methyl]urea), a Preclinical Candidate for the Treatment of Idiopathic Pulmonary Fibrosis
2021 · Oscar Mammoliti, Adeline Palisse, et al. · Journal of Medicinal Chemistry · 34
Discovery of GLPG2451, a Novel Once Daily Potentiator for the Treatment of Cystic Fibrosis
2021 · Steven E. Van der Plas, Hans Kelgtermans, et al. · Journal of Medicinal Chemistry · 26
Isothiourea-Catalyzed Asymmetric O- to C-Carboxyl Transfer of Furanyl Carbonates
2011 · Andrew Smith, Caroline Joannesse, et al. · Synthesis · 8
Design of a potent and selective dual JAK1/TYK2 inhibitor
2024 · Oscar Mammoliti, Christel Menet, et al. · Bioorganic & Medicinal Chemistry · 5
Regiodivergent Lewis base-promoted O- to C-carboxyl transfer of furanyl carbonates
2015 · Craig D. Campbell, Caroline Joannesse, et al. · Organic & Biomolecular Chemistry · 5
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N-Heterocyclic Carbene Catalysed Oxygen-to-Carbon Carboxyl Transfer of Indolyl and Benzofuranyl Carbonates
2008 · Andrew Smith, Jennifer Thomson, et al. · Synthesis · 5
HBsAg Suppression by a New Series of HBV RNA Destabilizers: Discovery and Effects on In Vitro Neurite Outgrowth
2026 · Jacques Huck, Caroline Joannesse, et al. · Journal of Medicinal Chemistry · 3
Discovery and Characterization of GLPG3808, a PAPD5/7 Inhibitor for Suppression of Hepatitis B Viral Infections
2026 · Oscar Mammoliti, Adeline Palisse, et al. · Journal of Medicinal Chemistry · 2
Abstract C113: Discovery of Best-in-Class FGFR3 small molecule inhibitors with high isoform selectivity and activity against gatekeeper mutations
2025 · Sandrine Vendeville, Lijs Beke, et al. · Molecular Cancer Therapeutics · 1
Correction to “Discovery of GLPG2451, a Novel Once Daily Potentiator for the Treatment of Cystic Fibrosis”
2021 · Steven E. Van der Plas, Hans Kelgtermans, et al. · Journal of Medicinal Chemistry
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Isothiourea-promoted O- to C-carboxyl transfer reactions
2011 · Joannesse, Caroline · St Andrews Research Repository (St Andrews Research Repository)
ChemInform Abstract: Isothiourea‐Catalyzed Asymmetric O‐ to C‐Carboxyl Transfer of Furanyl Carbonates.
2011 · Caroline Joannesse, Louis C. Morrill, et al. · ChemInform
CCDC 822214: Experimental Crystal Structure Determination
2011 · Joannesse, C., Morrill, L.C., et al. · The Cambridge Structural Database
CCDC 822213: Experimental Crystal Structure Determination
2011 · Joannesse, C., Morrill, L.C., et al. · The Cambridge Structural Database
ChemInform Abstract: Isothiourea‐Catalyzed Enantioselective Carboxy Group Transfer.
2010 · Caroline Joannesse, Craig P. Johnston, et al. · ChemInform
Enantioselective Steglich Rearrangement Using Isothiourea Catalysts
2009 · C. Joannesse, C. P. Johnston, et al. · Synfacts
CCDC 683088: Experimental Crystal Structure Determination
2009 · Thomson, J.E., Kyle, A.F., et al. · The Cambridge Structural Database
CCDC 683085: Experimental Crystal Structure Determination
2009 · Thomson, J.E., Kyle, A.F., et al. · The Cambridge Structural Database
Works count: 34
Citation count: 646
H-index: 9
I10-index: 9
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