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Alessandro Deplano

Observed names: A. Deplano, DEPLANO, ALESSANDRO, Deplano A., Deplano, A, Deplano, Alessandro
Observed institutions: Universitat Autònoma de Barcelona, University of Cagliari, American University, University of Ferrara, Istituto Superiore di Sanità, Aptuit (Italy), Parc Científic de Barcelona, Sapienza University of Rome, Evotec (United States)
ORCID: 0000-0002-8451-5831
Observed ORCID: 0000-0002-8451-5831
OpenAlex ID: A5023339313
Potent Nematicidal Activity of Maleimide Derivatives on Meloidogyne incognita
2016 · Kodjo Eloh, Monica Demurtas, et al. · Journal of Agricultural and Food Chemistry · 46
Computationally driven discovery of SARS-CoV-2 M pro inhibitors: from design to experimental validation
2022 · Léa El Khoury, Zhifeng Jing, et al. · Chemical Science · 45
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Design, Synthesis and Evaluation of Antiproliferative Activity of New Benzimidazolehydrazones
2016 · Valentina Onnis, Monica Demurtas, et al. · Molecules · 45
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Design, synthesis and antiviral evaluation of novel heteroarylcarbothioamide derivatives as dual inhibitors of HIV-1 reverse transcriptase-associated RNase H and RDDP functions
2017 · Angela Corona, Valentina Onnis, et al. · Pathogens and Disease · 40
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Structure-activity relationship with pyrazoline-based aromatic sulfamates as carbonic anhydrase isoforms I, II, IX and XII inhibitors: Synthesis and biological evaluation
2019 · Davide Moi, Alessio Nocentini, et al. · European Journal of Medicinal Chemistry · 39
A new convenient synthetic method and preliminary pharmacological characterization of triazinediones as prokineticin receptor antagonists
2014 · Cenzo Congiu, Valentina Onnis, et al. · European Journal of Medicinal Chemistry · 38
Synthesis of sulfonamides incorporating piperazinyl-ureido moieties and their carbonic anhydrase I, II, IX and XII inhibitory activity
2015 · Cenzo Congiu, Valentina Onnis, et al. · Bioorganic & Medicinal Chemistry Letters · 31
In Vitro Nematicidal Activity of Aryl Hydrazones and Comparative GC-MS Metabolomics Analysis
2015 · Kodjo Eloh, Monica Demurtas, et al. · Journal of Agricultural and Food Chemistry · 25
Appliance of the piperidinyl-hydrazidoureido linker to benzenesulfonamide compounds: Synthesis, in vitro and in silico evaluation of potent carbonic anhydrase II, IX and XII inhibitors
2020 · Davide Moi, Alessio Nocentini, et al. · Bioorganic Chemistry · 22
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Development and Validation of Molecular Overlays Derived from Three-Dimensional Hydrophobic Similarity with PharmScreen
2018 · Javier Vázquez, Alessandro Deplano, et al. · Journal of Chemical Information and Modeling · 22
Exploring the fatty acid amide hydrolase and cyclooxygenase inhibitory properties of novel amide derivatives of ibuprofen
2020 · Alessandro Deplano, Jessica Karlsson, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 20
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Sulfonamide/sulfamate switch with a series of piperazinylureido derivatives: Synthesis, kinetic and in silico evaluation as carbonic anhydrase isoforms I, II, IV, and IX inhibitors
2019 · Alessio Nocentini, Davide Moi, et al. · European Journal of Medicinal Chemistry · 20
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Synthesis and carbonic anhydrase I, II, IX and XII inhibitory activity of sulfamates incorporating piperazinyl-ureido moieties
2015 · Cenzo Congiu, Valentina Onnis, et al. · Bioorganic & Medicinal Chemistry · 20
Homology modeling of a Class A GPCR in the inactive conformation: A quantitative analysis of the correlation between model/template sequence identity and model accuracy
2016 · Stefano Costanzi, Matthew Skorski, et al. · Journal of Molecular Graphics and Modelling · 17
Assessing the Performance of Mixed Strategies To Combine Lipophilic Molecular Similarity and Docking in Virtual Screening
2020 · Javier Vazquez, Alessandro Deplano, et al. · Journal of Chemical Information and Modeling · 16
Synthesis and in vitro evaluation of piperazinyl-ureido sulfamates as steroid sulfatase inhibitors
2019 · Davide Moi, Paul A. Foster, et al. · European Journal of Medicinal Chemistry · 16
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Benzylamides and piperazinoarylamides of ibuprofen as fatty acid amide hydrolase inhibitors
2019 · Alessandro Deplano, Mariateresa Cipriano, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 15
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Interaction of the N-(3-Methylpyridin-2-yl)amide Derivatives of Flurbiprofen and Ibuprofen with FAAH: Enantiomeric Selectivity and Binding Mode
2015 · Jessica Karlsson, Carmine M. Morgillo, et al. · PLoS ONE · 15
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Characterisation of (R)-2-(2-Fluorobiphenyl-4-yl)-N-(3-Methylpyridin-2-yl)Propanamide as a Dual Fatty Acid Amide Hydrolase: Cyclooxygenase Inhibitor
2015 · Sandra Gouveia-Figueira, Jessica Karlsson, et al. · PLoS ONE · 15
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Novel propanamides as fatty acid amide hydrolase inhibitors
2017 · Alessandro Deplano, Carmine Marco Morgillo, et al. · European Journal of Medicinal Chemistry · 12
The fatty acid amide hydrolase and cyclooxygenase-inhibitory properties of novel amide derivatives of carprofen
2020 · Alessandro Deplano, Jessica Karlsson, et al. · Bioorganic Chemistry · 9
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Synthesis of Sulfonamides Incorporating Piperidinyl-Hydrazidoureido and Piperidinyl-Hydrazidothioureido Moieties and Their Carbonic Anhydrase I, II, IX and XII Inhibitory Activity
2022 · Davide Moi, Alessandro Deplano, et al. · Molecules · 8
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Design, synthesis and in vitro and in vivo biological evaluation of flurbiprofen amides as new fatty acid amide hydrolase/cyclooxygenase-2 dual inhibitory potential analgesic agents
2021 · Alessandro Deplano, Jessica Karlsson, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 8
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Molecular Basis for Non-Covalent, Non-Competitive FAAH Inhibition
2022 · Carmine Marco Morgillo, Antonio Lupia, et al. · International Journal of Molecular Sciences · 7
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Inhibitory effect of positively charged triazine antagonists of prokineticin receptors on the transient receptor vanilloid type-1 (TRPV1) channel
2015 · Luciano De Petrocellis, Aniello Schiano Moriello, et al. · Pharmacological Research · 7
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Works count: 47
Citation count: 565
H-index: 16
I10-index: 20
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