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Vladimír Garaj

Observed names: Garaj V, V Garaj, V. Garaj, VLADIMÍR GARAJ, Vladimir Garaj
ORCID: 0000-0002-8229-414X
Observed ORCID: 0000-0002-8229-414X
OpenAlex ID: A5024473336
Carbonic anhydrase inhibitors: Novel sulfonamides incorporating 1,3,5-triazine moieties as inhibitors of the cytosolic and tumour-associated carbonic anhydrase isozymes I, II and IX
2005 · Vladimir Garaj, Luca Puccetti, et al. · Bioorganic & Medicinal Chemistry Letters · 149
Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating 1,2,4-triazine moieties
2004 · Vladimir Garaj, Luca Puccetti, et al. · Bioorganic & Medicinal Chemistry Letters · 106
Sulfonamides incorporating 1,3,5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II: Solution and X-ray crystallographic studies
2011 · Fabrizio Carta, Vladimir Garaj, et al. · Bioorganic & Medicinal Chemistry · 100
Optimal detection of cholinesterase activity in biological samples: Modifications to the standard Ellman’s assay
2014 · Dominika Dingova, Jacqueline Leroy, et al. · Analytical Biochemistry · 83
Novel sulfonamide incorporating piperazine, aminoalcohol and 1,3,5-triazine structural motifs with carbonic anhydrase I, II and IX inhibitory action
2018 · Eva Havránková, Jozef Csöllei, et al. · Bioorganic Chemistry · 40
Small-molecule coumarin fluorescent pH probes for extremely acidic conditions
2019 · Jakub Joniak, Henrieta Stankovičová, et al. · Sensors and Actuators B Chemical · 39
Coumarin phenylsemicarbazones: sensitive colorimetric and fluorescent “turn-on” chemosensors for low-level water content in aprotic organic solvents
2016 · Marek Cigáň, Jan Gašpar, et al. · New Journal of Chemistry · 39
Photoswitching hydrazones based on benzoylpyridine
2019 · Bernard Mravec, Juraj Filo, et al. · Physical Chemistry Chemical Physics · 30
Enantioseparation of citalopram enantiomers by capillary electrophoresis: Method development through experimental design and computational modeling
2020 · Monica Budău, Gabriel Hancu, et al. · Chirality · 27
Novel sulfonamides incorporating 1,3,5-triazine and amino acid structural motifs as inhibitors of the physiological carbonic anhydrase isozymes I, II and IV and tumor-associated isozyme IX
2018 · Peter Mikuš, Dominika Krajčiová, et al. · Bioorganic Chemistry · 23
Isatinphenylsemicarbazones as efficient colorimetric sensors for fluoride and acetate anions – Anions induce tautomerism
2013 · Klaudia Jakusová, Jana Donovalová, et al. · Spectrochimica Acta Part A Molecular and Biomolecular Spectroscopy · 23
7-Dialkylaminocoumarin Oximates: Small Molecule Fluorescent “Turn-On” Chemosensors for Low-Level Water Content in Aprotic Organic Solvents
2017 · Marek Cigáň, Miroslav Horváth, et al. · Molecules · 21
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Synthesis and antimycobacterial evaluation of 5-alkylamino-N-phenylpyrazine-2-carboxamides
2014 · Jan Zitko, Barbora Servusová, et al. · Bioorganic & Medicinal Chemistry · 21
Thermodynamics of binding of Zn2+to carbonic anhydrase inhibitors
2003 · MILAN REMKO, VLADIMÍR GARAJ · Molecular Physics · 19
The inhibitory potency of local anesthetics on NMDA receptor signalling depends on their structural features
2011 · Carsten Gronwald, Vladimir Vegh, et al. · European Journal of Pharmacology · 16
Alkylamino derivatives of N-benzylpyrazine-2-carboxamide: synthesis and antimycobacterial evaluation
2015 · Barbora Servusova-Vanaskova, Ondrej Jandourek, et al. · MedChemComm · 13
Venlafaxine Chiral Separation by Capillary Electrophoresis Using Cyclodextrin Derivatives as Chiral Selector and Experimental Design Method Optimization
2020 · Andreea Milan, Gabriel Hancu, et al. · Symmetry · 11
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Gas phase and solution state stability of complexes L…M, where M = Cu2+, Ni2+, or Zn2+ and L = R−C( O)NHOH (R = H, NH2, CH3, CF3, or Phenyl)
2009 · Július Šille, Martin Šramko, et al. · Journal of Molecular Structure THEOCHEM · 11
Novel 1,3,5-Triazinyl Aminobenzenesulfonamides Incorporating Aminoalcohol, Aminochalcone and Aminostilbene Structural Motifs as Potent Anti-VRE Agents, and Carbonic Anhydrases I, II, VII, IX, and XII Inhibitors
2021 · Eva Havránková, Vladimír Garaj, et al. · International Journal of Molecular Sciences · 10
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Synthesis and Antimicrobial Evaluation of 6‐Alkylamino‐N‐phenylpyrazine‐2‐carboxamides
2015 · Barbora Servusova‐Vanaskova, Pavla Paterova, et al. · Chemical Biology & Drug Design · 10
Thermodynamics of binding of angiotensin-converting enzyme inhibitors to enzyme active site model
2008 · Martin Šramko, Vladimír Garaj, et al. · Journal of Molecular Structure THEOCHEM · 10
Optimization and Comparison of Synthetic Procedures for a Group of Triazinyl-Substituted Benzene-Sulfonamide Conjugates with Amino Acids
2017 · Dominika Krajčiová, Daniel Pecher, et al. · Molecules · 6
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Theoretical Study of Gas-Phase Acidities of Selected Angiotensin-Converting Enzyme Inhibitors
2005 · Martin Šramko, Milan Remko, et al. · Structural Chemistry · 6
New potent N‐hydroxycinnamamide‐based histone deacetylase inhibitors suppress proliferation and trigger apoptosis in THP‐1 leukaemia cells
2025 · Magdalena Onuscakova, Tereza Kauerova, et al. · Archiv der Pharmazie · 4
A simple UHPLC-MS/MS method for determination of SET2, a selective antagonist of TRPV2 receptor, in rat plasma samples
2024 · Linda Bartosova, Peter Balis, et al. · Journal of Chromatography B · 3
Works count: 32
Citation count: 826
H-index: 15
I10-index: 21
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