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Yoshikazu Uto

ORCID: 0000-0002-5170-3297
Observed ORCID: 0000-0002-5170-3297
OpenAlex ID: A5025266325
Synthesis of Functionalized Oxazolines and Oxazoles with DAST and Deoxo-Fluor
2000 · Andrew J. Phillips, Yoshikazu Uto, et al. · Organic Letters · 461
Total Synthesis and Revision of Stereochemistry of the Marine Metabolite Trunkamide A
1999 · Peter Wipf, Yoshikazu Uto · The Journal of Organic Chemistry · 98
Recent progress in the discovery and development of stearoyl CoA desaturase inhibitors
2015 · Yoshikazu Uto · Chemistry and Physics of Lipids · 68
Total Synthesis of a Stereoisomer of Bistramide C and Assignment of Configuration of the Natural Product
2002 · Peter Wipf, Yoshikazu Uto, et al. · Chemistry - A European Journal · 54
Total synthesis of the putative structure of the marine metabolite trunkamide A
1999 · Peter Wipf, Yoshikazu Uto · Tetrahedron Letters · 45
Hypoxia-inducible factor (HIF) inhibitors: a patent survey (2011-2015)
2016 · Hyun Seung Ban, Yoshikazu Uto, et al. · Expert Opinion on Therapeutic Patents · 44
Hypoxia-inducible factor inhibitors: a survey of recent patented compounds (2004 – 2010)
2011 · Hyun Seung Ban, Yoshikazu Uto, et al. · Expert Opinion on Therapeutic Patents · 42
Hypoxia-inducible factor (HIF) inhibitors: a patent survey (2016–2020)
2021 · Hyun Seung Ban, Yoshikazu Uto, et al. · Expert Opinion on Therapeutic Patents · 40
A Novel Inhibitor of Stearoyl-CoA Desaturase-1 Attenuates Hepatic Lipid Accumulation, Liver Injury and Inflammation in Model of Nonalcoholic Steatohepatitis
2013 · Nobuya Kurikawa, Toshiyuki Takagi, et al. · Biological and Pharmaceutical Bulletin · 40
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Synthesis and evaluation of novel stearoyl-CoA desaturase 1 inhibitors: 1′-{6-[5-(pyridin-3-ylmethyl)-1,3,4-oxadiazol-2-yl]pyridazin-3-yl}-3,4-dihydrospiro[chromene-2,4′-piperidine] analogs
2010 · Yoshikazu Uto, Yuko Ueno, et al. · European Journal of Medicinal Chemistry · 32
Novel spiropiperidine-based stearoyl-CoA desaturase-1 inhibitors: Identification of 1′-{6-[5-(pyridin-3-ylmethyl)-1,3,4-oxadiazol-2-yl]pyridazin-3-yl}-5-(trifluoromethyl)-3,4-dihydrospiro[chromene-2,4′-piperidine]
2009 · Yoshikazu Uto, Yohei Kiyotsuka, et al. · Bioorganic & Medicinal Chemistry Letters · 31
Novel benzoylpiperidine-based stearoyl-CoA desaturase-1 inhibitors: Identification of 6-[4-(2-methylbenzoyl)piperidin-1-yl]pyridazine-3-carboxylic acid (2-hydroxy-2-pyridin-3-ylethyl)amide and its plasma triglyceride-lowering effects in Zucker fatty rats
2009 · Yoshikazu Uto, Tsuneaki Ogata, et al. · Bioorganic & Medicinal Chemistry Letters · 28
Novel and potent inhibitors of stearoyl-CoA desaturase-1. Part II: Identification of 4-ethylamino-3-(2-hydroxyethoxy)-N-[5-(3-trifluoromethylbenzyl)thiazol-2-yl]benzamide and its biological evaluation
2009 · Yoshikazu Uto, Tsuneaki Ogata, et al. · Bioorganic & Medicinal Chemistry Letters · 28
Discovery of novel SCD1 inhibitors: 5-Alkyl-4,5-dihydro-3H-spiro[1,5-benzoxazepine-2,4′-piperidine] analogs
2011 · Yoshikazu Uto, Yuko Ueno, et al. · European Journal of Medicinal Chemistry · 24
1, 2-Benzisoxazole: A Privileged Structure with a Potential for Polypharmacology
2016 · Yoshikazu Uto · Current Pharmaceutical Design · 22
Novel and potent inhibitors of stearoyl-CoA desaturase-1. Part I: Discovery of 3-(2-hydroxyethoxy)-4-methoxy-N-[5-(3-trifluoromethylbenzyl)thiazol-2-yl]benzamide
2009 · Yoshikazu Uto, Tsuneaki Ogata, et al. · Bioorganic & Medicinal Chemistry Letters · 22
1,2-Benzisoxazole compounds: a patent review (2009 – 2014)
2015 · Yoshikazu Uto · Expert Opinion on Therapeutic Patents · 19
Imidazo[1,2-a]pyridines as cholesterol 24-hydroxylase (CYP46A1) inhibitors: a patent evaluation (WO2014061676)
2014 · Yoshikazu Uto · Expert Opinion on Therapeutic Patents · 10
Synthesis of Functionalized Oxazolines and Oxazoles with DAST and Deoxo-Fluor
2002 · Andrew J. Phillips, Yoshikazu Uto, et al. · Organic Letters · 7
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Piperidine and pyrrolidine analogs as glycogen synthase activators; a patent evaluation (WO2011058122)
2012 · Yoshikazu Uto · Expert Opinion on Therapeutic Patents · 4
Benzisoxazole analogs as glycogen synthase activators, a patent evaluation (WO2011057956)
2012 · Yoshikazu Uto · Expert Opinion on Therapeutic Patents · 2
ChemInform Abstract: Novel Spiropiperidine‐Based Stearoyl‐CoA Desaturase‐1 Inhibitors: Identification of 1′‐{6‐[5‐(Pyridin‐3‐ylmethyl)‐1,3,4‐oxadiazol‐2‐yl] pyridazin‐3‐yl}‐5‐(trifluoromethyl)‐3,4‐dihydrospiro [chromene‐2,4′‐piperidine].
2010 · Yoshikazu Uto, et al. et al. · ChemInform
ChemInform Abstract: Total Synthesis of a Stereoisomer of Bistramide C and Assignment of Configuration of the Natural Product.
2002 · Peter Wipf, Yoshikazu Uto, et al. · ChemInform
ChemInform Abstract: Synthesis of Functionalized Oxazolines and Oxazoles with DAST and Deoxo‐Fluor.
2000 · Andrew J. Phillips, Yoshikazu Uto, et al. · ChemInform
ChemInform Abstract: Total Synthesis and Revision of Stereochemistry of the Marine Metabolite Trunkamide A.
2000 · Peter Wipf, Yoshikazu Uto · ChemInform
Works count: 26
Citation count: 1,121
H-index: 17
I10-index: 18
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