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Tim J. Luker

Observed names: Luker, T., Luker, Timothy Jon, T. J. Luker, T. LUKER, T. Luker, Tim J Luker, Tim Luker, Timothy J. Luker, Timothy Luker
OpenAlex ID: A5026898037
Molybdenum-Mediated Carbonylation of Aryl Halides with Nucleophiles Using Microwave Irradiation
2010 · Bryan Roberts, David Liptrot, et al. · Organic Letters · 110
Discovery of Potent and Selective Adamantane-Based Small-Molecule P2X7Receptor Antagonists/Interleukin-1β Inhibitors
2007 · Mark Furber, Lilian Alcaraz, et al. · Journal of Medicinal Chemistry · 60
Strategies to improve in vivo toxicology outcomes for basic candidate drug molecules
2011 · Tim Luker, Lilian Alcaraz, et al. · Bioorganic & Medicinal Chemistry Letters · 59
Palladium catalysed amination of electron deficient halothiophenes
2000 · Tim J Luker, Haydn G Beaton, et al. · Tetrahedron Letters · 52
Synthesis and Further Reactivity of Functionalized Lactam-Derived Enol Triflates
1997 · Tim Luker, Henk Hiemstra, et al. · The Journal of Organic Chemistry · 51
Total Synthesis of Desoxoprosophylline: Application of a Lactam-Derived Enol Triflate to Natural Product Synthesis
1997 · Tim Luker, Henk Hiemstra, et al. · The Journal of Organic Chemistry · 51
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Permanganate Oxidation of 1,5,9-Trienes: Stereoselective Synthesis of Tetrahydrofuran-Containing Fragments
2002 · Richard C. D. Brown, Carole J. Bataille, et al. · The Journal of Organic Chemistry · 50
Michael Additions to (R)-1-Acetyl-5-isopropoxy-3-pyrrolin-2-one and Subsequent N-Acyliminium Ion Generation: Synthesis of Enantiopure 1-Azabicycles and Preparation of an Intermediate for a Projected Synthesis of Roseophilin
1998 · Tim Luker, Wim-Jan Koot, et al. · The Journal of Organic Chemistry · 47
Enantioselective Formal Total Synthesis of Roseophilin
2000 · Samantha J. Bamford, Tim Luker, et al. · Organic Letters · 45
Molybdenum-mediated synthesis of quinazolin-4(3H)-ones via cyclocarbonylation using microwave irradiation
2011 · Bryan Roberts, David Liptrot, et al. · Tetrahedron Letters · 40
Tandem reactions on a zirconocene template
1997 · S. F. Fillery, G. J. Gordon, et al. · Pure and Applied Chemistry · 39
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Substituted indole-1-acetic acids as potent and selective CRTh2 antagonists—discovery of AZD1981
2011 · Tim Luker, Roger Bonnert, et al. · Bioorganic & Medicinal Chemistry Letters · 38
Organozirconium methods for the efficient construction of the bicyclo[9.3.0]tetradecane dolabellane skeleton
1996 · Tim Luker, Richard J. Whitby · Tetrahedron Letters · 34
Formation of medium-size bridged ring systems via ring-closing metathesis of 2,5-disubstituted-2,3-dihydro-1H-pyrroles
2000 · Samantha J. Bamford, Kees Goubitz, et al. · Journal of the Chemical Society Perkin Transactions 1 · 32
Elaboration of zirconacyclopentanes by sequential insertion of lithium chloroallylide and ketones or aldehydes
1994 · Tim Luker, Richard J. Whitby · Tetrahedron Letters · 32
The Regiochemistry of Carbenoid Insertion into Zirconacycles
2000 · George J. Gordon, Tim Luker, et al. · Tetrahedron · 30
Insertion of phenyl azide and diphenyldiazomethane into bis(cyclopentadienyl)zirconacyclopentanes. Crystal structure of an 18-electron alkyl zirconocene triazenido complex
1995 · Tim Luker, Richard J. Whitby, et al. · Journal of Organometallic Chemistry · 30
Prediction of Efficacious Inhalation Lung Doses via the Use of In Silico Lung Retention Quantitative Structure-Activity Relationship Models and In Vitro Potency Screens
2010 · Anne Cooper, Tim Potter, et al. · Drug Metabolism and Disposition · 27
trans-2-Tritylcyclohexanol as a Chiral Auxiliary in Permanganate-Mediated Oxidative Cyclization of 2-Methylenehept-5-enoates: Application to the Synthesis of trans-(+)-Linalool Oxide
2014 · Ali M. Al Hazmi, Nadeem S. Sheikh, et al. · Organic Letters · 26
The discovery of novel, potent and highly selective inhibitors of inducible nitric oxide synthase (iNOS)
2010 · David R. Cheshire, Anders Åberg, et al. · Bioorganic & Medicinal Chemistry Letters · 26
Synthesis and reactivity of pyrrolidinone- and piperidinone-derived enol triflates
1996 · Tim Luker, Henk Hiemstra, et al. · Tetrahedron Letters · 23
Deferitazole, a new orally active iron chelator
2015 · Robert C. Hider, Xiaole Kong, et al. · Dalton Transactions · 19
Lipophilicity of acidic compounds: Impact of ion pair partitioning on drug design
2011 · Mark C. Wenlock, Patrick Barton, et al. · Bioorganic & Medicinal Chemistry Letters · 17
The tandem insertion of lithium chloroallylide and various electrophiles into zirconacyclopentanes
1995 · Tim Luker, Richard J. Whitby · Tetrahedron Letters · 15
Enantioselective Formal Synthesis of Eurylene: Synthesis of the cis- and trans-THF Fragments Using Oxidative Cyclization
2010 · Nadeem S. Sheikh, Carole J. Bataille, et al. · Organic Letters · 14
Works count: 54
Citation count: 1,031
H-index: 21
I10-index: 29
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