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Benedict‐Tilman Berger

Observed names: B.-T. Berger, B.T. Berger, Benedict Tilman Berger, Benedict-Tilman Berger, Benedict-Tilmann Berger, Berger Benedict-Tilman, Berger, Benedict-Tilman, Berger, Benedict-Tilman (author), Tillman-Berger, Benedict
ORCID: 0000-0002-3314-2617
Observed ORCID: 0000-0002-3314-2617
OpenAlex ID: A5028720772
Quantitative, Wide-Spectrum Kinase Profiling in Live Cells for Assessing the Effect of Cellular ATP on Target Engagement
2017 · James D. Vasta, Cesear R. Corona, et al. · Cell chemical biology · 270
CDK11 regulates pre-mRNA splicing by phosphorylation of SF3B1
2022 · Milan Hluchý, Pavla Gajdušková, et al. · Nature · 94
Chemical proteomics reveals the target landscape of 1,000 kinase inhibitors
2023 · Maria Reinecke, Paul Brear, et al. · Nature Chemical Biology · 91
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Binding Kinetics Survey of the Drugged Kinome
2018 · Victoria Georgi, Felix Schiele, et al. · Journal of the American Chemical Society · 85
Structure-kinetic relationship reveals the mechanism of selectivity of FAK inhibitors over PYK2
2021 · Benedict-Tilman Berger, Marta Amaral, et al. · Cell chemical biology · 76
Mutation in Abl kinase with altered drug-binding kinetics indicates a novel mechanism of imatinib resistance
2021 · Agatha Lyczek, Benedict-Tilman Berger, et al. · Proceedings of the National Academy of Sciences · 69
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Quantifying Target Occupancy of Small Molecules Within Living Cells
2020 · M.B. Robers, R. Friedman-Ohana, et al. · Annual Review of Biochemistry · 66
SGC-GAK-1: A Chemical Probe for Cyclin G Associated Kinase (GAK)
2019 · Christopher R. M. Asquith, Benedict-Tilman Berger, et al. · Journal of Medicinal Chemistry · 65
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Development, Optimization, and Structure–Activity Relationships of Covalent-Reversible JAK3 Inhibitors Based on a Tricyclic Imidazo[5,4-d]pyrrolo[2,3-b]pyridine Scaffold
2018 · Michael Forster, Apirat Chaikuad, et al. · Journal of Medicinal Chemistry · 61
Furo[3,2‐b]pyridine: A Privileged Scaffold for Highly Selective Kinase Inhibitors and Effective Modulators of the Hedgehog Pathway
2018 · Václav Němec, Michaela Hylsová, et al. · Angewandte Chemie International Edition · 55
Optimization of pyrazolo[1,5-a]pyrimidines lead to the identification of a highly selective casein kinase 2 inhibitor
2020 · Andreas Krämer, Christian Georg Kurz, et al. · European Journal of Medicinal Chemistry · 51
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Characterization of a dual BET / HDAC inhibitor for treatment of pancreatic ductal adenocarcinoma
2020 · Xin Zhang, Tim Zegar, et al. · International Journal of Cancer · 50
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Design of a “Two-in-One” Mutant-Selective Epidermal Growth Factor Receptor Inhibitor That Spans the Orthosteric and Allosteric Sites
2021 · Florian Wittlinger, David E. Heppner, et al. · Journal of Medicinal Chemistry · 45
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Controlling the Covalent Reactivity of a Kinase Inhibitor with Light
2021 · Martin Reynders, Apirat Chaikuad, et al. · Angewandte Chemie International Edition · 45
Structure-Based Design of Selective Salt-Inducible Kinase Inhibitors
2021 · Roberta Tesch, Marcel Rak, et al. · Journal of Medicinal Chemistry · 42
Identification of molecular targets for the targeted treatment of gastric cancer using dasatinib
2020 · Raquel Carvalho Montenegro, Alison Howarth, et al. · Oncotarget · 42
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Single tracer-based protocol for broad-spectrum kinase profiling in live cells with NanoBRET
2021 · Matthew B. Robers, Jennifer M. Wilkinson, et al. · STAR Protocols · 37
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Highly selective inhibitors of protein kinases CLK and HIPK with the furo[3,2-b]pyridine core
2021 · Václav Němec, Lukáš Maier, et al. · European Journal of Medicinal Chemistry · 33
Development and Characterization of Type I, Type II, and Type III LIM-Kinase Chemical Probes
2022 · Thomas Hanke, Sebastian Mathea, et al. · Journal of Medicinal Chemistry · 32
Fast Iterative Synthetic Approach toward Identification of Novel Highly Selective p38 MAP Kinase Inhibitors
2019 · Sandra Röhm, Benedict-Tilman Berger, et al. · Journal of Medicinal Chemistry · 28
Novel, highly potent PROTACs targeting AURORA-A kinase
2022 · Jelena Bozilovic, Lorenz Eing, et al. · Current Research in Chemical Biology · 27
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Selective targeting of the αC and DFG-out pocket in p38 MAPK
2020 · Sandra Röhm, Martin Schröder, et al. · European Journal of Medicinal Chemistry · 27
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NVP‐BHG712: Effects of Regioisomers on the Affinity and Selectivity toward the EPHrin Family
2018 · Alix Tröster, Stephanie Heinzlmeir, et al. · ChemMedChem · 27
Illuminating the Dark: Highly Selective Inhibition of Serine/Threonine Kinase 17A with Pyrazolo[1,5- a ]pyrimidine-Based Macrocycles
2022 · Christian G. Kurz, Franziska Preuss, et al. · Journal of Medicinal Chemistry · 25
A Toolbox for the Generation of Chemical Probes for Baculovirus IAP Repeat Containing Proteins
2022 · Martin P. Schwalm, Lena M. Berger, et al. · Frontiers in Cell and Developmental Biology · 22
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Works count: 72
Citation count: 1,762
H-index: 24
I10-index: 39
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