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Thomas Robert

2-Aminophenones, a common precursor to N-aryl isatins and acridines endowed with bioactivities
2018 · Nahida Mokhtari Brikci-Nigassa, Ghenia Bentabed-Ababsa, et al. · Tetrahedron · 39
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Synthesis, biological evaluation and molecular modeling studies of imidazo[1,2- a ]pyridines derivatives as protein kinase inhibitors
2016 · Marie Lawson, Jordi Rodrigo, et al. · European Journal of Medicinal Chemistry · 35
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Structure-based design of novel quinoxaline-2-carboxylic acids and analogues as Pim-1 inhibitors
2018 · Bruno Oyallon, Marie Brachet-Botineau, et al. · European Journal of Medicinal Chemistry · 32
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Identification of a new series of flavopiridol-like structures as kinase inhibitors with high cytotoxic potency
2020 · Nada Ibrahim, Pascal Bonnet, et al. · European Journal of Medicinal Chemistry · 28
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Development of a CDK10/CycM in vitro Kinase Screening Assay and Identification of First Small-Molecule Inhibitors
2020 · Thomas Robert, Jared L. Johnson, et al. · Frontiers in Chemistry · 28
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In vitro identification of imidazo[1,2-a]pyrazine-based antileishmanial agents and evaluation of L. major casein kinase 1 inhibition
2020 · Marc-Antoine Bazin, Sandrine Cojean, et al. · European Journal of Medicinal Chemistry · 27
Betulin, a Newly Characterized Compound in Acacia auriculiformis Bark, Is a Multi-Target Protein Kinase Inhibitor
2021 · Augustine A. Ahmadu, Claire Delehouzé, et al. · Molecules · 25
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New Quinoxaline Derivatives as Dual Pim-1/2 Kinase Inhibitors: Design, Synthesis and Biological Evaluation
2021 · Bruno Oyallon, Marie Brachet-Botineau, et al. · Molecules · 23
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Synthesis and anticancer activity of novel bisindolylhydroxymaleimide derivatives with potent GSK-3 kinase inhibition
2018 · Hannah J. Winfield, Michael M. Cahill, et al. · Bioorganic & Medicinal Chemistry · 20
Imidazo[1,2-a]quinazolines as novel, potent EGFR-TK inhibitors: Design, synthesis, bioactivity evaluation, and in silico studies
2023 · Zaman Hasanvand, Tayebeh Oghabi Bakhshaiesh, et al. · Bioorganic Chemistry · 18
From simple quinoxalines to potent oxazolo[5,4- f ]quinoxaline inhibitors of glycogen-synthase kinase 3 (GSK3)
2019 · Frédéric Lassagne, Camille Duguépéroux, et al. · Organic & Biomolecular Chemistry · 14
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Synthesis, Docking Study and Kinase Inhibitory Activity of a Number of New Substituted Pyrazolo[3,4-c]pyridines
2016 · Meropi Sklepari, Nikolaos Lougiakis, et al. · Chemical and Pharmaceutical Bulletin · 13
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Overexpression of Eimeria tenella Rhoptry Kinase 2 Induces Early Production of Schizonts
2023 · Adeline Ribeiro E. Silva, Mamadou Amadou Diallo, et al. · Microbiology Spectrum · 9
Oxazolo[5,4-f]quinoxaline-type selective inhibitors of glycogen synthase kinase-3α (GSK-3α): Development and impact on temozolomide treatment of glioblastoma cells
2023 · Mohamed Hasyeoui, Frédéric Lassagne, et al. · Bioorganic Chemistry · 9
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Exploration of 7-azaindole-coumaranone hybrids and their analogues as protein kinase inhibitors
2021 · Malikotsi A. Qhobosheane, Richard M. Beteck, et al. · Chemico-Biological Interactions · 9
From benzofuro-, benzothieno- and 10-methylindolo-[2,3- b ]-fused benzothiopyrano[4,3,2- de ]quinolines to the corresponding benzothiopyrano[4,3,2- de ]1,8-naphthyridines: synthesis and properties of these hexacyclic heteroaromatic compounds
2022 · Nicolas Mast, William Erb, et al. · New Journal of Chemistry · 8
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Streptomyces hygroscopicus UFPEDA 3370: A valuable source of the potent cytotoxic agent nigericin and its evaluation against human colorectal cancer cells
2020 · Iza Mirela Rodini Garcia-Princival, Jefferson Luiz Princival, et al. · Chemico-Biological Interactions · 8
Practical approach to N-benzyl derivatives of 2-amino-8-methoxy-4H-chromene-3-carbonitrile by reductive amination: Exploration of their effects against protein kinases and in silico ADME profiling
2022 · Marwa Dhiabi, Ali Bouattour, et al. · Journal of Molecular Structure · 7
Discovery of thiazolidin-4-one analogue as selective GSK-3β inhibitor through structure based virtual screening
2021 · Bhanwar Singh Choudhary, Sukanya, et al. · Bioorganic & Medicinal Chemistry Letters · 7
Regorafenib analogues and their ferrocenic counterparts: synthesis and biological evaluation
2020 · Myron Wilde, Danielle Arzur, et al. · New Journal of Chemistry · 7
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Investigating the C2 Modulation of the Imidazo[1,2‐ a ]pyrazine‐Based Hit Compound CTN1122: Synthesis, in vitro Antileishmanial Activity, Cytotoxicity and Casein Kinase 1 Inhibition
2024 · Lhana Tisseur, Sandrine Cojean, et al. · ChemMedChem · 6
New Fusarochromanone Derivatives from the Marine Fungus Fusarium equiseti UBOCC-A-117302
2024 · Giang Nam Pham, Béatrice Josselin, et al. · Marine Drugs · 6
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Dibenzofuran Derivatives Inspired from Cercosporamide as Dual Inhibitors of Pim and CLK1 Kinases
2021 · Viet Hung Dao, Isabelle Ourliac-Garnier, et al. · Molecules · 6
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Tampering with Cell Division by Using Small‐Molecule Inhibitors of CDK–CKS Protein Interactions
2015 · Amel Hamdi, Aurélien Lesnard, et al. · ChemBioChem · 6
Structure Activity Relationship Studies around DB18, a Potent and Selective Inhibitor of CLK Kinases
2022 · Dabbugoddu Brahmaiah, Anagani Kanaka Durga Bhavani, et al. · Molecules · 5
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Works count: 85
Citation count: 430
H-index: 12
I10-index: 12
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