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Kasiram Katneni

Observed names: K. Katneni, Katneni Kasiram, Katneni, Kasiram
Institution: Monash University
OpenAlex ID: A5029502805
Structure-Guided Lead Optimization of Triazolopyrimidine-Ring Substituents Identifies PotentPlasmodium falciparumDihydroorotate Dehydrogenase Inhibitors with Clinical Candidate Potential
2011 · Jose M. Coteron, María Marco, et al. · Journal of Medicinal Chemistry · 290
Endochin-like quinolones are highly efficacious against acute and latent experimental toxoplasmosis
2012 · J. Stone Doggett, Aaron Nilsen, et al. · Proceedings of the National Academy of Sciences · 189
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An in vitro toolbox to accelerate anti-malarial drug discovery and development
2020 · Susan A. Charman, Alice Andreu, et al. · Malaria Journal · 150
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3,5-Diaryl-2-aminopyridines as a Novel Class of Orally Active Antimalarials Demonstrating Single Dose Cure in Mice and Clinical Candidate Potential
2012 · Yassir Younis, Frederic Douelle, et al. · Journal of Medicinal Chemistry · 133
Discovery, Synthesis, and Optimization of Antimalarial 4(1 H )-Quinolone-3-Diarylethers
2014 · Aaron Nilsen, Galen P. Miley, et al. · Journal of Medicinal Chemistry · 123
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Comparative Antimalarial Activities and ADME Profiles of Ozonides (1,2,4-trioxolanes) OZ277, OZ439, and Their 1,2-Dioxolane, 1,2,4-Trioxane, and 1,2,4,5-Tetraoxane Isosteres
2013 · Xiaofang Wang, Yuxiang Dong, et al. · Journal of Medicinal Chemistry · 89
Novel phthalazinone and benzoxazinone containing thiazolidinediones as antidiabetic and hypolipidemic agents
2001 · Gurram R Madhavan, Ranjan Chakrabarti, et al. · European Journal of Medicinal Chemistry · 89
Discovery and Structure–Activity Relationships of Pyrrolone Antimalarials
2013 · Dinakaran Murugesan, Alka Mital, et al. · Journal of Medicinal Chemistry · 81
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Permeability assessment of poorly water‐soluble compounds under solubilizing conditions: The reciprocal permeability approach
2006 · Kasiram Katneni, Susan A. Charman, et al. · Journal of Pharmaceutical Sciences · 63
A Prodrug Approach Toward Cancer-Related Carbonic Anhydrase Inhibition
2013 · Cindy J. Carroux, Gregory M. Rankin, et al. · Journal of Medicinal Chemistry · 60
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3-Alkylthio-1,2,4-triazine dimers with potent antimalarial activity
2010 · Kung Ban, Sandra Duffy, et al. · Bioorganic & Medicinal Chemistry Letters · 59
Novel Euglycemic and Hypolipidemic Agents. 4. Pyridyl- and Quinolinyl-Containing Thiazolidinediones
1999 · B. B. Lohray, Vidya Bhushan, et al. · Journal of Medicinal Chemistry · 59
Drug Transport Across the Blood-Brain Barrier and the Impact of Breast Cancer Resistance Protein (ABCG2)
2009 · Joseph Nicolazzo, Kasiram Katneni · Current Topics in Medicinal Chemistry · 57
Potent Antimalarials with Development Potential Identified by Structure-Guided Computational Optimization of a Pyrrole-Based Dihydroorotate Dehydrogenase Inhibitor Series
2021 · Michael J. Palmer, Xiaoyi Deng, et al. · Journal of Medicinal Chemistry · 49
Impact of Cremophor-EL and Polysorbate-80 on Digoxin Permeability across Rat Jejunum: Delineation of Thermodynamic and Transporter Related Events Using the Reciprocal Permeability Approach
2006 · Kasiram Katneni, Susan A. Charman, et al. · Journal of Pharmaceutical Sciences · 49
Discovery of Benzoylsulfonohydrazides as Potent Inhibitors of the Histone Acetyltransferase KAT6A
2019 · David J. Leaver, Benjamin Cleary, et al. · Journal of Medicinal Chemistry · 45
Insights Into Drug Repurposing, as Well as Specificity and Compound Properties of Piperidine-Based SARS-CoV-2 PLpro Inhibitors
2022 · Dale J. Calleja, Nathan Kuchel, et al. · Frontiers in Chemistry · 44
A novel PLpro inhibitor improves outcomes in a pre-clinical model of long COVID
2025 · Stefanie M. Bader, Dale J. Calleja, et al. · Nature Communications · 40
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Discovery and Structure–Activity Relationships of Quinazolinone-2-carboxamide Derivatives as Novel Orally Efficacious Antimalarials
2021 · Benoît Laleu, Yuichiro Akao, et al. · Journal of Medicinal Chemistry · 40
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Intestinal Lymph Flow, and Lipid and Drug Transport Scale Allometrically From Pre-clinical Species to Humans
2020 · Natalie L. Trevaskis, Given Lee, et al. · Frontiers in Physiology · 39
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Lead Optimization of a Pyrrole-Based Dihydroorotate Dehydrogenase Inhibitor Series for the Treatment of Malaria
2020 · Sreekanth Kokkonda, Xiaoyi Deng, et al. · Journal of Medicinal Chemistry · 39
Discovery of Acylsulfonohydrazide-Derived Inhibitors of the Lysine Acetyltransferase, KAT6A, as Potent Senescence-Inducing Anti-Cancer Agents
2020 · Daniel L. Priebbenow, David J. Leaver, et al. · Journal of Medicinal Chemistry · 38
Structure–Activity Relationship Studies of Orally Active Antimalarial 3,5-Substituted 2-Aminopyridines
2012 · Diego González Cabrera, Frederic Douelle, et al. · Journal of Medicinal Chemistry · 38
DNDI-6174 is a preclinical candidate for visceral leishmaniasis that targets the cytochrome bc 1
2023 · Stéphanie Braillard, Martine Keenan, et al. · Science Translational Medicine · 31
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Pharmacological and pharmacokinetic evaluation of celecoxib prodrugs in rats
2002 · Rao N.V.S. Mamidi, Ramesh Mullangi, et al. · Biopharmaceutics & Drug Disposition · 31
Works count: 60
Citation count: 2,231
H-index: 25
I10-index: 41
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