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Adeline Palisse
Observed names:
Palisse, Adeline,
Palisse, Adeline 1985-
Institution:
Galapagos (Belgium)
Observed institutions:
University of Wuppertal,
AstraZeneca (Netherlands),
Acerta Pharma BV (Netherlands),
Technical University of Munich,
Galapagos (Belgium)
ORCID:
0000-0001-8944-9565
Observed ORCID:
0000-0001-8944-9565
OpenAlex ID:
A5029877832
Metal-free reactions of alkynes via electrophilic iodocarbocyclizations
2012
·
Adeline Palisse
, Stefan F. Kirsch
·
Organic & Biomolecular Chemistry
·
73
Domino Reactions Consisting of Heterocyclization and 1,2‐Migration—Redox‐Neutral and Oxidative Transition‐Metal Catalysis
2011
·
Klaus‐Daniel Umland
, Adeline Palisse
, et al.
·
Angewandte Chemie International Edition
·
44
Discovery of the S1P2 Antagonist GLPG2938 (1-[2-Ethoxy-6-(trifluoromethyl)-4-pyridyl]-3-[[5-methyl-6-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]pyridazin-3-yl]methyl]urea), a Preclinical Candidate for the Treatment of Idiopathic Pulmonary Fibrosis
2021
·
Oscar Mammoliti
, Adeline Palisse
, et al.
·
Journal of Medicinal Chemistry
·
34
Discovery and Optimization of Orally Bioavailable Phthalazone and Cinnolone Carboxylic Acid Derivatives as S1P2 Antagonists against Fibrotic Diseases
2021
·
Oscar Mammoliti
, Koen Jansen
, et al.
·
Journal of Medicinal Chemistry
·
22
Synthesis of Furans through Silver‐Catalyzed Propargyl–Claisen Rearrangement Followed by Cyclocondensation
2014
·
Adeline Palisse
, Stefan F. Kirsch
·
European Journal of Organic Chemistry
·
20
Dominoreaktionen bestehend aus Heterocyclisierung und 1,2‐Verschiebung – redoxneutrale und oxidative Übergangsmetallkatalyse im Vergleich
2011
·
Klaus‐Daniel Umland
, Adeline Palisse
, et al.
·
Angewandte Chemie
·
15
Discovery of GLPG2737, a Potent Type 2 Corrector of CFTR for the Treatment of Cystic Fibrosis in Combination with a Potentiator and a Type 1 Co-corrector
2024
·
Mathieu Pizzonero
, Rhalid Akkari
, et al.
·
Journal of Medicinal Chemistry
·
13
Structure-Based Optimization of a Series of Covalent, Cell Active Bfl-1 Inhibitors
2024
·
Simon C. C. Lucas
, J. Henry Blackwell
, et al.
·
Journal of Medicinal Chemistry
·
10
Design of a potent and selective dual JAK1/TYK2 inhibitor
2024
·
Oscar Mammoliti
, Christel Menet
, et al.
·
Bioorganic & Medicinal Chemistry
·
5
Structure-Based Discovery of a Series of Covalent, Orally Bioavailable, and Selective BFL1 Inhibitors
2024
·
Adeline Palisse
, Tony Cheung
, et al.
·
Journal of Medicinal Chemistry
·
4
HBsAg Suppression by a New Series of HBV RNA Destabilizers: Discovery and Effects on In Vitro Neurite Outgrowth
2026
·
Jacques Huck
, Caroline Joannesse
, et al.
·
Journal of Medicinal Chemistry
·
3
Discovery and Characterization of GLPG3808, a PAPD5/7 Inhibitor for Suppression of Hepatitis B Viral Infections
2026
·
Oscar Mammoliti
, Adeline Palisse
, et al.
·
Journal of Medicinal Chemistry
·
2
Identification of novel, potent, and selective JAK2V617F inhibitors
2025
·
Fazal Hadi
, Peter Linders
, et al.
·
Blood
·
1
PDF
Optimization and Chemoproteomic Profiling of a Selective, Covalent Bfl-1-Targeting Cellular Tool
2025
·
J. Henry Blackwell
, Simon C. C. Lucas
, et al.
·
Journal of Medicinal Chemistry
CCDC 2122384: Experimental Crystal Structure Determination
2021
·
Mammoliti, Oscar
, Jansen, Koen
, et al.
·
The Cambridge Structural Database
CCDC 2122349: Experimental Crystal Structure Determination
2021
·
Mammoliti, Oscar
, Jansen, Koen
, et al.
·
The Cambridge Structural Database
Cascade Reactions Initiated by ᴨ - Activation. A Flexible Way to Heterocycles & Studies toward the Total Synthesis of Melohenine B
2018
·
Adeline Palisse
ChemInform Abstract: Synthesis of Furans Through Silver‐Catalyzed Propargyl‐Claisen Rearrangement Followed by Cyclocondensation.
2015
·
Adeline Palisse
, Stefan F. Kirsch
·
ChemInform
ChemInform Abstract: Metal‐Free Reactions of Alkynes via Electrophilic Iodocarbocyclizations
2013
·
Adeline Palisse
, Stefan F. Kirsch
·
ChemInform
ChemInform Abstract: Domino Reactions Consisting of Heterocyclization and 1,2‐Migration—Redox‐Neutral and Oxidative Transition‐Metal Catalysis.
2012
·
Klaus‐Daniel Umland
, Adeline Palisse
, et al.
·
ChemInform
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Works count:
21
Citation count:
246
H-index:
8
I10-index:
8
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