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Yuri Bolshan

Observed names: Bolshan, Y., Y. BOLSHAN, Y. Bolshan
ORCID: 0000-0003-4131-2898
Observed ORCID: 0000-0003-4131-2898
OpenAlex ID: A5031380398
Small-molecule inhibition of MLL activity by disruption of its interaction with WDR5
2012 · Guillermo Senisterra, Hong Wu, et al. · Biochemical Journal · 159
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Enamide Synthesis by Copper‐Catalyzed Cross‐Coupling of Amides and Potassium Alkenyltrifluoroborate Salts
2008 · Yuri Bolshan, Robert A. Batey · Angewandte Chemie International Edition · 154
An Allosteric Inhibitor of Protein Arginine Methyltransferase 3
2012 · Alena Siarheyeva, Guillermo Senisterra, et al. · Structure · 101
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A Room-Temperature Protocol for the Rhodium(I)-Catalyzed Addition of Arylboron Compounds to Sulfinimines
2005 · Yuri Bolshan, Robert A. Batey · Organic Letters · 96
Structure-Based Optimization of a Small Molecule Antagonist of the Interaction Between WD Repeat-Containing Protein 5 (WDR5) and Mixed-Lineage Leukemia 1 (MLL1)
2016 · Matthäus Getlik, David Smil, et al. · Journal of Medicinal Chemistry · 89
Nucleophilic Displacement at Benzhydryl Centers: Asymmetric Synthesis of 1,1-Diarylalkyl Derivatives
2003 · Yuri Bolshan, Cheng-yi Chen, et al. · Organic Letters · 74
Synthesis, Optimization, and Evaluation of Novel Small Molecules as Antagonists of WDR5-MLL Interaction
2013 · Yuri Bolshan, Matthäus Getlik, et al. · ACS Medicinal Chemistry Letters · 71
Bromo-deaza-SAH: A potent and selective DOT1L inhibitor
2013 · Wenyu Yu, David Smil, et al. · Bioorganic & Medicinal Chemistry · 67
(R)-β-Lysine-modified Elongation Factor P Functions in Translation Elongation
2012 · Tammy J. Bullwinkle, S. Betty Zou, et al. · Journal of Biological Chemistry · 54
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Metal-Free Synthesis of Ynones from Acyl Chlorides and Potassium Alkynyltrifluoroborate Salts
2013 · Cassandra Taylor, Yuri Bolshan · Organic Letters · 41
Copper-catalyzed cross-coupling of amides and potassium alkenyltrifluoroborate salts: a general approach to the synthesis of enamides
2010 · Yuri Bolshan, Robert A. Batey · Tetrahedron · 39
Metal-free methodology for the preparation of sterically hindered alkynoylphenols and its application to the synthesis of flavones and aurones
2015 · Cassandra Taylor, Yuri Bolshan · Tetrahedron Letters · 36
Enamide Synthesis by Copper‐Catalyzed Cross‐Coupling of Amides and Potassium Alkenyltrifluoroborate Salts
2008 · Yuri Bolshan, Robert A. Batey · Angewandte Chemie · 32
Brønsted Acid-Catalyzed Reactions of Trifluoroborate Salts with Benzhydryl Alcohols
2015 · Kayla M. Fisher, Yuri Bolshan · The Journal of Organic Chemistry · 28
A General Access to Propargylic Ethers through Brønsted Acid Catalyzed Alkynylation of Acetals and Ketals with Trifluoroborates
2015 · Matthew Baxter, Yuri Bolshan · Chemistry - A European Journal · 19
A general Brønsted acid-catalyzed allylation of benzhydryl alcohols
2016 · Ifedi Orizu, Yuri Bolshan · Tetrahedron Letters · 17
Crystal structures of Klebsiella pneumoniae pantothenate kinase in complex with N‐substituted pantothenamides
2013 · Buren Li, Wolfram Tempel, et al. · Proteins Structure Function and Bioinformatics · 16
Thiol on silica as a ‘catch and release’ support for isocyanates to afford ureas
2007 · Yuri Bolshan, Miroslaw J. Tomaszewski, et al. · Tetrahedron Letters · 13
Stereoselective Palladium-Catalyzed Arylation of Exo-Glycals with Aryl Iodides
2021 · Jeffery Regier, Supriya Ghanty, et al. · The Journal of Organic Chemistry · 12
Metal‐Free Alkenylation of Salicylaldehydes with Boronic Acids: Synthesis of Skipped Dienes and 2H‐Chromenes
2020 · Dylan H. Harris, Renata O. Barichello, et al. · European Journal of Organic Chemistry · 12
A Direct Brønsted Acid‐Catalyzed Azidation of Benzhydrols and Carbohydrates
2019 · Jeffery Regier, Robert Maillet, et al. · European Journal of Organic Chemistry · 12
Brønsted Acid-Catalyzed Direct Substitution of 2-Ethoxytetrahydrofuran with Trifluoroborate Salts
2016 · Kayla Fisher, Yuri Bolshan · Catalysts · 6
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Synthesis of C,N-Glycosides via Brønsted Acid-Catalyzed Azidation of exo-Glycals
2023 · Jeffery Regier, Yuri Bolshan · The Journal of Organic Chemistry · 4
Bromination of codeine and its derivatives: Revisiting a 95 year old process
2020 · Samira Barmaki, Arlene Ali, et al. · Tetrahedron Letters · 3
Metal-free Synthesis of Ynones from Acyl Chlorides and Potassium Alkynyltrifluoroborate Salts
2015 · Cassandra L. Taylor, Yuri Bolshan · Journal of Visualized Experiments · 3
Works count: 51
Citation count: 1,164
H-index: 16
I10-index: 21
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