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Masato Yoshikawa
Observed names:
M. YOSHIKAWA,
Masato YOSHIKAWA,
Yoshikawa, Masato
Institution:
Takeda (Japan)
Observed institutions:
Tokyo University of Science,
Kyoto University,
Himeji University,
Hoshi University,
Takeda (Japan),
The University of Tokyo
show all 6
ORCID:
0000-0002-7175-1173
Observed ORCID:
0000-0002-7175-1173
OpenAlex ID:
A5031824022
Ruthenium‐Catalyzed Propargylic Substitution Reactions of Propargylic Alcohols with Oxygen‐, Nitrogen‐, and Phosphorus‐Centered Nucleophiles
2005
·
Yoshiaki Nishibayashi
, Marilyn Daisy Milton
, et al.
·
Chemistry - A European Journal
·
184
Novel Ruthenium‐ and Platinum‐Catalyzed Sequential Reactions: Synthesis of Tri‐ and Tetrasubstituted Furans and Pyrroles from Propargylic Alcohols and Ketones
2003
·
Yoshiaki Nishibayashi
, Masato Yoshikawa
, et al.
·
Angewandte Chemie International Edition
·
182
Ruthenium-Catalyzed Propargylation of Aromatic Compounds with Propargylic Alcohols
2002
·
Yoshiaki Nishibayashi
, Masato Yoshikawa
, et al.
·
Journal of the American Chemical Society
·
165
Propargylation of Aromatic Compounds with Propargylic Alcohols Catalyzed by a Cationic Diruthenium Complex
2003
·
Yoshiaki Nishibayashi
, Youichi Inada
, et al.
·
Angewandte Chemie International Edition
·
150
Discovery of 7-Oxo-2,4,5,7-tetrahydro-6 H -pyrazolo[3,4- c ]pyridine Derivatives as Potent, Orally Available, and Brain-Penetrating Receptor Interacting Protein 1 (RIP1) Kinase Inhibitors: Analysis of Structure–Kinetic Relationships
2018
·
Masato Yoshikawa
, Morihisa Saitoh
, et al.
·
Journal of Medicinal Chemistry
·
118
Ruthenium- and Platinum-Catalyzed Sequential Reactions: Selective Synthesis of Fused Polycyclic Compounds from Propargylic Alcohols and Alkenes
2004
·
Yoshiaki Nishibayashi
, Masato Yoshikawa
, et al.
·
Journal of the American Chemical Society
·
89
Soticlestat, a novel cholesterol 24-hydroxylase inhibitor shows a therapeutic potential for neural hyperexcitation in mice
2020
·
Toshiya Nishi
, Shinichi Kondo
, et al.
·
Scientific Reports
·
76
PDF
Ruthenium‐Catalyzed Propargylation of Aromatic Compounds with Propargylic Alcohols
2006
·
Youichi Inada
, Masato Yoshikawa
, et al.
·
European Journal of Organic Chemistry
·
76
Ruthenium-Catalyzed Cycloaddition between Propargylic Alcohols and Cyclic 1,3-Dicarbonyl Compounds via an Allenylidene Intermediate
2004
·
Yoshiaki Nishibayashi
, Masato Yoshikawa
, et al.
·
The Journal of Organic Chemistry
·
75
Discovery of 1-[2-Fluoro-4-(1 H -pyrazol-1-yl)phenyl]-5-methoxy-3-(1-phenyl-1 H -pyrazol-5-yl)pyridazin-4(1 H )-one (TAK-063), a Highly Potent, Selective, and Orally Active Phosphodiesterase 10A (PDE10A) Inhibitor
2014
·
Jun Kunitomo
, Masato Yoshikawa
, et al.
·
Journal of Medicinal Chemistry
·
64
Design and biological evaluation of imidazo[1,2-a]pyridines as novel and potent ASK1 inhibitors
2012
·
Yoshito Terao
, Hideo Suzuki
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
64
TAK-676: A Novel Stimulator of Interferon Genes (STING) Agonist Promoting Durable IFN-dependent Antitumor Immunity in Preclinical Studies
2022
·
Elizabeth Carideo Cunniff
, Yosuke Sato
, et al.
·
Cancer Research Communications
·
62
Diastereo-differentiating cyclopropanation of a chiral enol ether: a simple method for the preparation of optically pure cyclopropyl ethers
1990
·
Takashi Sugimura
, Masato Yoshikawa
, et al.
·
Tetrahedron
·
59
Diastereo-differentiating Simmons-Smith reaction using a new chiral auxiliary
1989
·
Takashi Sugimura
, Tohru Futagawa
, et al.
·
Tetrahedron Letters
·
58
CETSA quantitatively verifies in vivo target engagement of novel RIPK1 inhibitors in various biospecimens
2017
·
Tsuyoshi Ishii
, Takuro Okai
, et al.
·
Scientific Reports
·
48
PDF
Discovery of Soticlestat, a Potent and Selective Inhibitor for Cholesterol 24-Hydroxylase (CH24H)
2021
·
Tatsuki Koike
, Masato Yoshikawa
, et al.
·
Journal of Medicinal Chemistry
·
45
PDF
Novel Ruthenium‐ and Platinum‐Catalyzed Sequential Reactions: Synthesis of Tri‐ and Tetrasubstituted Furans and Pyrroles from Propargylic Alcohols and Ketones
2003
·
Yoshiaki Nishibayashi
, Masato Yoshikawa
, et al.
·
Angewandte Chemie
·
45
Propargylation of Aromatic Compounds with Propargylic Alcohols Catalyzed by a Cationic Diruthenium Complex
2003
·
Yoshiaki Nishibayashi
, Youichi Inada
, et al.
·
Angewandte Chemie
·
43
Ruthenium-Catalyzed Dienyne Formation from Propargylic Alcohols and 1,3-Conjugated Dienes
2008
·
Masaki Daini
, Masato Yoshikawa
, et al.
·
Organometallics
·
41
Design and synthesis of a novel 2-oxindole scaffold as a highly potent and brain-penetrant phosphodiesterase 10A inhibitor
2015
·
Masato Yoshikawa
, Haruhi Kamisaki
, et al.
·
Bioorganic & Medicinal Chemistry
·
34
A novel Na+‐Independent alanine‐serine‐cysteine transporter 1 inhibitor inhibits both influx and efflux of D‐Serine
2016
·
Katsuya Sakimura
, Kenji Nakao
, et al.
·
Journal of Neuroscience Research
·
26
Preparation of streochemically pure sex pheromone components of the pine sawfly (Neodiprion sertifer) and field tests of the synthetic compounds.
1990
·
Akira TAI
, Naotake MORIMOTO
, et al.
·
Agricultural and Biological Chemistry
·
23
PDF
Hydroxy direction of zinc carbenoid addition to a remote olefin. Analysis and improvement of 2,4-pentanediol tethered Furukawa cyclopropanation
2001
·
Takashi Sugimura
, Tohru Futagawa
, et al.
·
Tetrahedron
·
17
Structure-based rational design of staurosporine-based fluorescent probe with broad-ranging kinase affinity for kinase panel application
2019
·
Yoshihiko Hirozane
, Masashi Toyofuku
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
16
Preparation of Optically Pure (3S,5S)- and (3R,5R)-2,6-Dimethyl-3,5-heptanediol
1990
·
Takashi Sugimura
, Masato Yoshikawa
, et al.
·
Bulletin of the Chemical Society of Japan
·
14
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Works count:
65
Citation count:
1,874
H-index:
22
I10-index:
29
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