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Gabriele Amari

CHF6001 I: A Novel Highly Potent and Selective Phosphodiesterase 4 Inhibitor with Robust Anti-Inflammatory Activity and Suitable for Topical Pulmonary Administration
2015 · Nadia Moretto, Paola Caruso, et al. · Journal of Pharmacology and Experimental Therapeutics · 77
Novel Class of Benzoic Acid Ester Derivatives as Potent PDE4 Inhibitors for Inhaled Administration in the Treatment of Respiratory Diseases
2014 · Elisabetta Armani, Gabriele Amari, et al. · Journal of Medicinal Chemistry · 47
Structural Determinants of Torpedo c alifornica Acetylcholinesterase Inhibition by the Novel and Orally Active Carbamate Based Anti-Alzheimer Drug Ganstigmine (CHF-2819)
2006 · Cecilia Bartolucci, Mariacristina Siotto, et al. · Journal of Medicinal Chemistry · 47
Bronchodilator Activity of (3R)-3-[[[(3-fluorophenyl)[(3,4,5-trifluorophenyl)methyl]amino] carbonyl]oxy]-1-[2-oxo-2-(2-thienyl)ethyl]-1-azoniabicyclo[2.2.2]octane bromide (CHF5407), a Potent, Long-Acting, and Selective Muscarinic M3 Receptor Antagonist
2010 · G. Villetti, F. Pastore, et al. · Journal of Pharmacology and Experimental Therapeutics · 28
Discovery of Diaryl Imidazolidin-2-one Derivatives, a Novel Class of Muscarinic M3 Selective Antagonists (Part 1)
2007 · Ilaria Peretto, Roberto Forlani, et al. · Journal of Medicinal Chemistry · 26
Synthesis, pharmacological evaluation, and structure–activity relationships of benzopyran derivatives with potent SERM activity
2004 · Gabriele Amari, Elisabetta Armani, et al. · Bioorganic & Medicinal Chemistry · 24
Discovery and Optimization of Thiazolidinyl and Pyrrolidinyl Derivatives as Inhaled PDE4 Inhibitors for Respiratory Diseases
2017 · Laura Carzaniga, Gabriele Amari, et al. · Journal of Medicinal Chemistry · 22
Discovery of Diaryl Imidazolidin-2-one Derivatives, a Novel Class of Muscarinic M3 Selective Antagonists (Part 2)
2007 · Ilaria Peretto, Claudia Fossati, et al. · Journal of Medicinal Chemistry · 16
Discovery of M3 Antagonist-PDE4 Inhibitor Dual Pharmacology Molecules for the Treatment of Chronic Obstructive Pulmonary Disease
2021 · Elisabetta Armani, Andrea Rizzi, et al. · Journal of Medicinal Chemistry · 12
Novel Basic Isoflavones as Inhibitors of Bone Resorption
2001 · Maurizio Delcanale, Gabriele Amari, et al. · Helvetica Chimica Acta · 12
Effects of 3-Phenyl-4-[[4-[2-(1-piperidinyl)ethoxy]phenyl]methyl]- 2 H-1-benzopyran-7-ol (CHF 4056), a Novel Nonsteroidal Estrogen Agonist/Antagonist, on Reproductive and Nonreproductive Tissue
2002 · Elisabetta Galbiati, Paola Lorenza Caruso, et al. · Journal of Pharmacology and Experimental Therapeutics · 11
Discovery of a Potent, Selective, and Orally Bioavailable Tool Compound for Probing the Role of Lysophosphatidic Acid Type 2 Receptor Antagonists in Fibrotic Disorders
2023 · Elisabetta Armani, Andrea Rizzi, et al. · Journal of Medicinal Chemistry · 10
The Molecular Structure and Crystal Organization Of Rac -terfenadine/β-cyclodextrin/tartaric Acid Multicomponent Inclusion Complex
2002 · Alessia Bacchi, Giancarlo Pelizzi, et al. · Supramolecular chemistry · 10
Pharmacological Actions of a Novel, Potent, Tissue-Selective Benzopyran Estrogen
2002 · Elisabetta Galbiati, Paola Lorenza Caruso, et al. · Journal of Pharmacology and Experimental Therapeutics · 10
The Crystal Structure of the Inclusion Complex of the Sodium Salt of Piroxicam with β-cyclodextrin
1998 · Angiola Chiesi-villa, Corrado Rizzoli, et al. · Supramolecular chemistry · 9
Erythroid differentiation ability of butyric acid analogues: Identification of basal chemical structures of new inducers of foetal haemoglobin
2015 · Nicoletta Bianchi, Cristiano Chiarabelli, et al. · European Journal of Pharmacology · 8
New method for the resolution of the enantiomers of 5,6-Dihydroxy-2-Methyl-Aminotetralin by selective derivatization and HPLC analysis: Application to biological fluids
1996 · Ivano Rondelli, Roberto Corsaletti, et al. · Chirality · 8
Solution‐ and Solid‐state Structures of the (—)‐n‐Heptylcarbamate of Geneseroline and Its Hydrochloride Salt
1995 · Enrico Redenti, Maurizio Delcanale, et al. · Journal of Pharmaceutical Sciences · 7
Optimization of M3 Antagonist–PDE4 Inhibitor (MAPI) Dual Pharmacology Molecules for the Treatment of COPD
2023 · Andrea Rizzi, Gabriele Amari, et al. · Journal of Medicinal Chemistry · 6
Synthesis of glycose carbamides and evaluation of the induction of erythroid differentiation of human erythroleukemic K562 cells
2008 · Martina Landi, Giorgio Catelani, et al. · European Journal of Medicinal Chemistry · 6
Differentiation of diastereomeric aminotetralins by metastable ion spectra of 2‐oxazolidinone derivatives upon electron‐impact ionization
1992 · Antonio Selva, Enrico Redenti, et al. · Organic Mass Spectrometry · 6
Geneserine hydrochloride
1994 · A. Bacchi, G. Pelizzi, et al. · Acta Crystallographica Section C Crystal Structure Communications · 2
Selective method for plasma quantitation of the stereoisomers of a new aminotetralin by high-performance liquid chromatography with electrochemical detection
1993 · Ivano Rondelli, Fabrizia Mariotti, et al. · Journal of Chromatography B Biomedical Sciences and Applications · 2
The soluble tris(acetylacetonato)vanadium/dialkylaluminium chloride system for alkene polymerization. Enhancement of activity by the use of dimethylaluminium chloride
1987 · Antonino Giarrusso, Gabriele Amari, et al. · Die Makromolekulare Chemie Rapid Communications · 2
Corrigendum to “Synthesis, pharmacological evaluation, and structure–activity relationships of benzopyran derivatives with potent SERM activity” [Bioorg. Med. Chem. 12 (2004) 3763]
2004 · Gabriele Amari, Elisabetta Armani, et al. · Bioorganic & Medicinal Chemistry · 1
Works count: 34
Citation count: 410
H-index: 11
I10-index: 14
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