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Author

Naoki Teno

Observed names: N. TENO, N. Teno, NAOKI TENO, Naoki TENO, Teno, Naoki
Observed institutions: Novartis (Switzerland), The University of Melbourne, Hokkaido University, Kobe Gakuin University, Novartis (Japan), Hiroshima International University, Novartis Institutes for BioMedical Research, Ciba-Geigy Japan Limited (Japan), The University of Osaka
ORCID: 0000-0002-3940-5473
Observed ORCID: 0000-0002-3940-5473
OpenAlex ID: A5034188197
Lysophospholipase I identified as a ghrelin deacylation enzyme in rat stomach
2004 · Yuka Shanado, Motohiko Kometani, et al. · Biochemical and Biophysical Research Communications · 68
N-Alkynyl Imides (Ynimides): Synthesis and Use as a Variant of Highly Labile Ethynamine
2011 · Takuya Sueda, Ayumi Oshima, et al. · Organic Letters · 62
Novel scaffold for cathepsin K inhibitors
2007 · Naoki Teno, Takahiro Miyake, et al. · Bioorganic & Medicinal Chemistry Letters · 43
Discovery of Orally Bioavailable Cathepsin S Inhibitors for the Reversal of Neuropathic Pain
2008 · Osamu Irie, Takatoshi Kosaka, et al. · Journal of Medicinal Chemistry · 41
2-Cyano-pyrimidines: A New Chemotype for Inhibitors of the Cysteine Protease Cathepsin K
2007 · Eva Altmann, Reiner Aichholz, et al. · Journal of Medicinal Chemistry · 36
Ag- and Au-Catalyzed Addition of Alcohols to Ynimides: β-Regioselective Carbonylation and Production of Oxazoles
2013 · Takuya Sueda, Arisa Kawada, et al. · Organic Letters · 33
Synthesis of Novel Farnesoid X Receptor Agonists and Validation of Their Efficacy in Activating Differentiation of Mouse Bone Marrow-Derived Mesenchymal Stem Cells into Osteoblasts
2019 · Ko Fujimori, Yusuke Iguchi, et al. · Molecules · 28
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Conformational Studies on the Specific Cleavage Site of Type I Collagen (α-1) Fragment (157–192) by Cathepsins K and L by Proton NMR Spectroscopy
1999 · Atsuko Y Nosaka, Kenji Kanaori, et al. · Bioorganic & Medicinal Chemistry · 25
Overcoming hERG issues for brain-penetrating cathepsin S inhibitors: 2-Cyanopyrimidines. Part 2
2008 · Osamu Irie, Takatoshi Kosaka, et al. · Bioorganic & Medicinal Chemistry Letters · 24
Discovery of selective and nonpeptidic cathepsin S inhibitors
2008 · Osamu Irie, Takeru Ehara, et al. · Bioorganic & Medicinal Chemistry Letters · 24
Effect of Cathepsin K Inhibitors on Bone Resorption
2008 · Naoki Teno, Keiichi Masuya, et al. · Journal of Medicinal Chemistry · 23
Synthesis of active center-directed peptide inhibitors of plasmin.
1988 · YOSHIO OKADA, YUKO TSUDA, et al. · Chemical and Pharmaceutical Bulletin · 23
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Discovery of Orally Active and Nonsteroidal Farnesoid X Receptor (FXR) Antagonist with Propensity for Accumulation and Responsiveness in Ileum
2021 · Naoki Teno, Yusuke Iguchi, et al. · ACS Medicinal Chemistry Letters · 22
Significant effects of Z-Gln-Val-Val-OMe, common sequences of thiol proteinase inhibitors on thiol proteinases
1987 · N. Teno, S. Tsuboi, et al. · Biochemical and Biophysical Research Communications · 22
Development of Active Center-Directed Plasmin and Plasma Kallikrein Inhibitors and Studies on the Structure-Inhibitory Activity Relationship.
1993 · Naoki TENO, Keiko WANAKA, et al. · Chemical and Pharmaceutical Bulletin · 20
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Nonacidic Chemotype Possessing N-Acylated Piperidine Moiety as Potent Farnesoid X Receptor (FXR) Antagonists
2018 · Naoki Teno, Yukiko Yamashita, et al. · ACS Medicinal Chemistry Letters · 17
New chemotypes for cathepsin K inhibitors
2008 · Naoki Teno, Osamu Irie, et al. · Bioorganic & Medicinal Chemistry Letters · 17
Development of Active Center-Directed Inhibitors against Plasmin.
1991 · Naoki TENO, Keiko WANAKA, et al. · Chemical and Pharmaceutical Bulletin · 17
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IRL 2500: A potent ETB selective endothelin antagonist
1996 · Th. Früh, H. Saika, et al. · Bioorganic & Medicinal Chemistry Letters · 16
Discovery of FXR/PPARγ dual partial agonist
2023 · Yukiko Yamashita, Keigo Gohda, et al. · Bioorganic & Medicinal Chemistry · 14
Synthesis of plasmin substrates and relationship between their structure and plasmin activity
1986 · Yoshio Okada, Yuko Tsuda, et al. · International journal of peptide & protein research · 14
Active site-directed plasmin inhibitors: Extension on the P2 residue
2015 · Koushi Hidaka, Keigo Gohda, et al. · Bioorganic & Medicinal Chemistry · 13
Pyrrolopyrimidine-inhibitors with hydantoin moiety as spacer can explore P4/S4 interaction on plasmin
2014 · Naoki Teno, Keigo Gohda, et al. · Bioorganic & Medicinal Chemistry · 13
N1-Substituted benzimidazole scaffold for farnesoid X receptor (FXR) agonists accompanying prominent selectivity against vitamin D receptor (VDR)
2020 · Arisa Masuda, Keigo Gohda, et al. · Bioorganic & Medicinal Chemistry · 12
Identification of potent farnesoid X receptor (FXR) antagonist showing favorable PK profile and distribution toward target tissues: Comprehensive understanding of structure-activity relationship of FXR antagonists
2019 · Naoki Teno, Yukiko Yamashita, et al. · Bioorganic & Medicinal Chemistry · 12
Works count: 67
Citation count: 825
H-index: 17
I10-index: 31
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