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Richard J. Upton

Investigations into the Manzamine Alkaloid Biosynthetic Hypothesis
1998 · Jack E. Baldwin, Timothy D. W. Claridge, et al. · Angewandte Chemie International Edition · 100
NMR quantification using an artificial signal
2010 · Roger D. Farrant, John C. Hollerton, et al. · Magnetic Resonance in Chemistry · 89
Dissociated Nonsteroidal Glucocorticoid Receptor Modulators; Discovery of the Agonist Trigger in a Tetrahydronaphthalene−Benzoxazine Series
2006 · Mike Barker, Margaret Clackers, et al. · Journal of Medicinal Chemistry · 79
A Chemical Probe for the ATAD2 Bromodomain
2016 · Paul Bamborough, Chun‐wa Chung, et al. · Angewandte Chemie International Edition · 77
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The synthesis of cyclic tetrapeptoid analogues of the antiprotozoal natural product apicidin
2001 · Peter J Murray, Michael Kranz, et al. · Bioorganic & Medicinal Chemistry Letters · 77
Improving the passive permeability of macrocyclic peptides: Balancing permeability with other physicochemical properties
2014 · Praew Thansandote, Robert M. Harris, et al. · Bioorganic & Medicinal Chemistry · 64
Use of Calculated Physicochemical Properties to Enhance Quantitative Response When Using Charged Aerosol Detection
2016 · Max W. Robinson, Alan P. Hill, et al. · Analytical Chemistry · 60
Synthesis of Diverse Macrocyclic Peptidomimetics Utilizing Ring-Closing Metathesis and Solid-Phase Synthesis
2004 · Anthony G. M. Barrett, Alan J. Hennessy, et al. · The Journal of Organic Chemistry · 58
Novel extracellular mycobactins, the carboxymycobactins from Mycobacterium avium
1995 · Stephen J Lane, Peter S Marshall, et al. · Tetrahedron Letters · 56
Biosynthetic origin of mycobacterial cell wall arabinosyl residues
1995 · M Scherman, A Weston, et al. · Journal of Bacteriology · 53
Syntheses of trans-5- Oxo-hexahydro-pyrrolo[3,2-b]pyrroles and trans-5-Oxo-hexahydro-furo[3,2-b]pyrroles (Pyrrolidine trans-Lactams and trans-Lactones): New Pharmacophores for Elastase Inhibition
1998 · Simon J. F. Macdonald, David J. Belton, et al. · Journal of Medicinal Chemistry · 43
A Flexible, Practical, and Stereoselective Synthesis of Enantiomerically Pure trans-5-Oxohexahydropyrrolo[3,2-b]pyrroles (Pyrrolidine-trans-lactams), a New Class of Serine Protease Inhibitors, Using Acyliminium Methodology
1999 · Simon J. F. Macdonald, Geoffrey D. E. Clarke, et al. · The Journal of Organic Chemistry · 41
Development of GSK's NMR guides – a tool to encourage the use of more sustainable solvents
2016 · Hugo E. Gottlieb, Grazyna Graczyk-Millbrandt, et al. · Green Chemistry · 30
Isolation and characterization of carboxymycobactins as the second extracellular siderophores in Mycobacterium smegmatis
1998 · Stephen J. Lane, Peter S. Marshall, et al. · BioMetals · 29
Convenient method for the kinetic resolution of β-aminoalcohols
2005 · Béatrice Pelotier, Ghislaine Priem, et al. · Tetrahedron Letters · 27
Solution, solid phase and computational structures of apicidin and its backbone‐reduced analogs
2005 · Michael Kranz, Peter John Murray, et al. · Journal of Peptide Science · 21
Untersuchungen zur Hypothese der Manzaminalkaloid-Biosynthese
1998 · Jack E. Baldwin, Timothy D. W. Claridge, et al. · Angewandte Chemie · 17
A Chemical Probe for the ATAD2 Bromodomain
2016 · Paul Bamborough, Chun‐wa Chung, et al. · Angewandte Chemie · 13
A stereoselective synthesis via a 5-exo-trig cyclisation of trans-2-oxohexahydro-2H-furo[3,2-b]pyrroles (pyrrolidine-trans-lactones)—potent, novel elastase inhibitors
1998 · Simon J. F. Macdonald, Keith Mills, et al. · Journal of the Chemical Society Perkin Transactions 1 · 12
Synthesis of tetrasubstituted bicyclo[3.2.1]octenes as potential inhibitors of influenza virus sialidase
1999 · Paul S. Jones, Paul W. Smith, et al. · Bioorganic & Medicinal Chemistry Letters · 11
Rearrangement of a 16α,17α-Epoxy-16β-methylandrostane-17β-carbothioic Acid to a 17β-Mercapto-16β-methylandrostane-17α,16α-carbolactone
1998 · Brian M. Bain, Gordon H. Phillipps, et al. · The Journal of Organic Chemistry · 7
Pyrrolidine-5,5-trans-lactams 3. Alternative RegiochemicalOutcome of the Acyl-Iminium Coupling Reaction.
2003 · David Andrews, Alan Borthwick, et al. · Synthesis · 1
CCDC 274844: Experimental Crystal Structure Determination
2007 · Kranz, M., Murray, P.J., et al. · The Cambridge Structural Database
Convenient Method for the Kinetic Resolution of β‐Amino Alcohols.
2006 · Beatrice Pelotier, Ghislaine Priem, et al. · ChemInform
CCDC 233388: Experimental Crystal Structure Determination
2004 · Barrett, A.G.M., Hennessy, A.J., et al. · The Cambridge Structural Database
Works count: 30
Citation count: 965
H-index: 17
I10-index: 20
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