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Giovanna Pescatore

Discovery of Raltegravir, a Potent, Selective Orally Bioavailable HIV-Integrase Inhibitor for the Treatment of HIV-AIDS Infection
2008 · Vincenzo Summa, Alessia Petrocchi, et al. · Journal of Medicinal Chemistry · 653
Tetrazole thioacetanilides: Potent non-nucleoside inhibitors of WT HIV reverse transcriptase and its K103N mutant
2006 · Ester Muraglia, Olaf D. Kinzel, et al. · Bioorganic & Medicinal Chemistry Letters · 90
Discovery and Synthesis of HIV Integrase Inhibitors: Development of Potent and Orally Bioavailable N-Methyl Pyrimidones
2007 · Cristina Gardelli, Emanuela Nizi, et al. · Journal of Medicinal Chemistry · 67
A Novel Series of Potent and Selective Ketone Histone Deacetylase Inhibitors with Antitumor Activity in Vivo
2008 · Philip Jones, Sergio Altamura, et al. · Journal of Medicinal Chemistry · 59
Design and Synthesis of Bicyclic Pyrimidinones as Potent and Orally Bioavailable HIV-1 Integrase Inhibitors
2008 · Ester Muraglia, Olaf Kinzel, et al. · Journal of Medicinal Chemistry · 53
Discovery of a Potent Class I Selective Ketone Histone Deacetylase Inhibitor with Antitumor Activity in Vivo and Optimized Pharmacokinetic Properties
2009 · Olaf Kinzel, Laura Llauger-Bufi, et al. · Journal of Medicinal Chemistry · 46
A study on the chelation control in the regioselective opening of 2,3-bifunctionalized epoxides
2001 · Giuliana Righi, Giovanna Pescatore, et al. · Tetrahedron · 29
New stereoselective synthesis of the peptidic aminopeptidase inhibitors bestatin, phebestin and probestin
2003 · Giuliana Righi, Claudia D'Achille, et al. · Tetrahedron Letters · 28
Identification and SAR of novel pyrrolo[1,2-a]pyrazin-1(2H)-one derivatives as inhibitors of poly(ADP-ribose) polymerase-1 (PARP-1)
2009 · Giovanna Pescatore, Danila Branca, et al. · Bioorganic & Medicinal Chemistry Letters · 21
A novel base-mediated intramolecular hydroamination to build fused heteroaryl pyrazinones
2008 · Laura Llauger, Costanza Bergami, et al. · Tetrahedron Letters · 14
Dihydroxy-pyrimidine and N-methylpyrimidone HIV-integrase inhibitors: Improving cell based activity by the quaternarization of a chiral center
2009 · Emanuela Nizi, Maria Vittoria Orsale, et al. · Bioorganic & Medicinal Chemistry Letters · 12
Optimization of a series of potent and selective ketone histone deacetylase inhibitors
2008 · Giovanna Pescatore, Olaf Kinzel, et al. · Bioorganic & Medicinal Chemistry Letters · 12
The synthesis of tetrahydropyridopyrimidones as a new scaffold for HIV-1 integrase inhibitors
2007 · Olaf D. Kinzel, Edith Monteagudo, et al. · Tetrahedron Letters · 11
ChemInform Abstract: A Study on the Chelation Control in the Regioselective Opening of 2,3‐Bifunctionalized Epoxides.
2001 · Giuliana Righi, Giovanna Pescatore, et al. · ChemInform · 1
ChemInform Abstract: Identification and SAR of Novel Pyrrolo[1,2‐a]pyrazin‐1(2H)‐one Derivatives as Inhibitors of Poly(ADP‐Ribose) Polymerase‐1 (PARP‐1).
2010 · Giovanna Pescatore, et al. et al. · ChemInform
ChemInform Abstract: A Novel Base‐Mediated Intramolecular Hydroamination to Build Fused Heteroaryl Pyrazinones.
2009 · Laura Llauger, Costanza Bergami, et al. · ChemInform
New Stereoselective Synthesis of the Peptidic Aminopeptidase Inhibitors Bestatin, Phebestin and Probestin.
2003 · Giuliana Righi, Claudia D'Achille, et al. · ChemInform
Works count: 17
Citation count: 1,096
H-index: 12
I10-index: 13
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