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Andrea Trabocchi

Observed names: A Trabocchi, A. Trabocchi, Andrea Trabocchi., TRABOCCHI, ANDREA, Trabocchi Andrea, Trabocchi, A., Trabocchi, Andrea, Trabocchi, Andrea; Menchi, Gloria; Guarna, Francesco; Machetti, Fabrizio; Scarpi, Dina; Guarna, Antonio:
Observed institutions: University of Milan, University of Oxford, Menarini Group (Italy), Florence (Netherlands), Institute for the Chemistry of OrganoMetallic Compounds, University of Florence, University of California, Berkeley
ORCID: 0000-0003-1774-9301
Observed ORCID: 0000-0003-1774-9301
OpenAlex ID: A5041407933
Peptidomimetic toolbox for drug discovery
2020 · Elena Lenci, Andrea Trabocchi · Chemical Society Reviews · 334
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A New Family of Cinchona-Derived Amino Phosphine Precatalysts: Application to the Highly Enantio- and Diastereoselective Silver-Catalyzed Isocyanoacetate Aldol Reaction
2011 · Filippo Sladojevich, Andrea Trabocchi, et al. · Journal of the American Chemical Society · 261
AI is a viable alternative to high throughput screening: a 318-target study
2024 · The Atomwise AIMS Program, Izhar Wallach, et al. · Scientific Reports · 149
Occurrence of Morpholine in Central Nervous System Drug Discovery
2021 · Elena Lenci, Lorenzo Calugi, et al. · ACS Chemical Neuroscience · 100
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Exploring the chemical space and the bioactivity profile of lactams: a chemoinformatic study
2019 · Fernanda I. Saldívar-González, Elena Lenci, et al. · RSC Advances · 87
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Suzuki Reaction of Vinyl Triflates from Six- and Seven-Membered N-Alkoxycarbonyl Lactams with Boronic Acids and Esters
2001 · Ernesto G. Occhiato, Andrea Trabocchi, et al. · The Journal of Organic Chemistry · 80
Peptidomimetics in Organic and Medicinal Chemistry: The Art of Transforming Peptides in Drugs
2014 · Andrea Trabocchi, Antonio Guarna · Wiley eBooks · 74
Structural diversity of bicyclic amino acids
2007 · A. Trabocchi, D. Scarpi, et al. · Amino Acids · 73
γ- and δ-Amino Acids: Synthetic Strategies and Relevant Applications
2005 · A. Trabocchi, F. Guarna, et al. · Current Organic Chemistry · 72
Diversity‐Oriented Synthesis: Basics and Applications in Organic Synthesis, Drug Discovery, and Chemical Biology
2013 · TRABOCCHI, ANDREA, CAVALIERI, DUCCIO, et al. · Wiley eBooks · 66
Synthesis and Conformational Analysis of Small Peptides Containing 6-Endo-BT(t)L Scaffolds as Reverse Turn Mimetics
2002 · Andrea Trabocchi, Ernesto G. Occhiato, et al. · The Journal of Organic Chemistry · 55
Carbohydrates in diversity-oriented synthesis: challenges and opportunities
2015 · E. Lenci, G. Menchi, et al. · Organic & Biomolecular Chemistry · 50
Click-Chemistry-Derived Triazole Ligands of Arginine−Glycine−Aspartate (RGD) Integrins with a Broad Capacity To Inhibit Adhesion of Melanoma Cells and Both in Vitro and in Vivo Angiogenesis
2010 · Andrea Trabocchi, Gloria Menchi, et al. · Journal of Medicinal Chemistry · 48
Bicyclic acetals: biological relevance, scaffold analysis, and applications in diversity-oriented synthesis
2018 · Elena Lenci, Gloria Menchi, et al. · Organic & Biomolecular Chemistry · 43
Synthesis and Reactivity of Bicycles Derived from Tartaric Acid and α-Amino Acids: A Novel Class of Conformationally Constrained Dipeptide Isosteres Based upon Enantiopure 3-Aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxylic Acid
1999 · Antonio Guarna, Antonio Guidi, et al. · The Journal of Organic Chemistry · 40
Novel matrix metalloproteinase inhibitors: an updated patent review (2014 - 2020)
2021 · Elena Lenci, Lucrezia Cosottini, et al. · Expert Opinion on Therapeutic Patents · 38
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Diversity‐Oriented Synthesis of Morpholine‐Containing Molecular Scaffolds
2009 · Claudia Lalli, Andrea Trabocchi, et al. · Chemistry - A European Journal · 37
Diversity-Oriented Synthesis and Chemoinformatic Analysis of the Molecular Diversity of sp3-Rich Morpholine Peptidomimetics
2018 · Elena Lenci, Riccardo Innocenti, et al. · Frontiers in Chemistry · 36
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Convenient Route to Enantiopure Fmoc-Protected Morpholine-3-carboxylic Acid
2007 · Filippo Sladojevich, Andrea Trabocchi, et al. · The Journal of Organic Chemistry · 35
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Development of a GC-376 Based Peptidomimetic PROTAC as a Degrader of 3-Chymotrypsin-like Protease of SARS-CoV-2
2024 · Deborah Grifagni, Elena Lenci, et al. · ACS Medicinal Chemistry Letters · 34
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Multilayered Bioorthogonal SERS Nanoprobes Selectively Aggregating in Human Fluids: A Smart Optical Assay for β-Amyloid Peptide Quantification
2023 · Caterina Dallari, Elena Lenci, et al. · ACS Sensors · 34
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Diversity‐Oriented Synthesis and Chemoinformatics: A Fruitful Synergy towards Better Chemical Libraries
2022 · Elena Lenci, Andrea Trabocchi · European Journal of Organic Chemistry · 33
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Diversity-Oriented Synthesis as a Tool for Chemical Genetics
2014 · Elena Lenci, Antonio Guarna, et al. · Molecules · 33
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Diversity-oriented synthesis as a tool to expand the chemical space of DNA-encoded libraries
2021 · Elena Lenci, Lorenzo Baldini, et al. · Bioorganic & Medicinal Chemistry · 32
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Stereoselective cyclopropanation of serine- and threonine-derived oxazines to access new morpholine-based scaffolds
2008 · Filippo Sladojevich, Andrea Trabocchi, et al. · Organic & Biomolecular Chemistry · 32
Works count: 213
Citation count: 3,113
H-index: 29
I10-index: 86
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