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Setshaba D. Khanye

Observed names: David S. Khanye, Khanye, S.D., Khanye, Setshaba D., S. D. Khanye, Setshaba D Khanye, Setshaba David Khanye, Setshaba Khanye
Institution: Rhodes University
ORCID: 0000-0003-0725-5738
Observed ORCID: 0000-0003-0725-5738
OpenAlex ID: A5042779104
Isomerization and ring-closing metathesis for the synthesis of 6-, 7- and 8-membered benzo- and pyrido-fused N,N-, N,O- and N,S-heterocycles
2004 · Willem A.L. van Otterlo, Garreth L. Morgans, et al. · Tetrahedron Letters · 73
Synthesis and in vitro evaluation of gold(I) thiosemicarbazone complexes for antimalarial activity
2010 · Setshaba D. Khanye, Gregory S. Smith, et al. · Journal of Inorganic Biochemistry · 72
Application of the Morita-Baylis-Hillman reaction in the synthesis of 3-[( N -cycloalkylbenzamido)methyl]-2-quinolones as potential HIV-1 integrase inhibitors
2017 · Khethobole C. Sekgota, Swarup Majumder, et al. · Bioorganic Chemistry · 58
Ferrocenylthiosemicarbazones conjugated to a poly(propyleneimine) dendrimer scaffold: Synthesis and in vitro antimalarial activity
2011 · Setshaba D. Khanye, Jiri Gut, et al. · Journal of Organometallic Chemistry · 48
Synthesis and in vitro antimalarial and antitubercular activity of gold(III) complexes containing thiosemicarbazone ligands
2011 · Setshaba D. Khanye, Baojie Wan, et al. · Journal of Organometallic Chemistry · 48
Synthesis of unsaturated 1,4-heteroatom-containing benzo-fused heterocycles using a sequential isomerization–ring-closing metathesis strategy
2009 · Garreth L. Morgans, E. Lindani Ngidi, et al. · Tetrahedron · 42
Ferrocenyl and organic novobiocin derivatives: Synthesis and their in vitro biological activity
2017 · Mziyanda Mbaba, Amanda N. Mabhula, et al. · Journal of Inorganic Biochemistry · 36
Quinolone-isoniazid hybrids: synthesis and preliminary in vitro cytotoxicity and anti-tuberculosis evaluation
2019 · Richard M. Beteck, Ronnett Seldon, et al. · MedChemComm · 35
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Novobiocin–ferrocene conjugates possessing anticancer and antiplasmodial activity independent of HSP90 inhibition
2018 · Mziyanda Mbaba, Jo-Anne de la Mare, et al. · JBIC Journal of Biological Inorganic Chemistry · 33
Repurposing a polymer precursor: Synthesis and in vitro medicinal potential of ferrocenyl 1,3-benzoxazine derivatives
2019 · Mziyanda Mbaba, Laura M.K. Dingle, et al. · European Journal of Medicinal Chemistry · 32
Easy-To-Synthesize Spirocyclic Compounds Possess Remarkable in Vivo Activity against Mycobacterium tuberculosis
2018 · Ana Guardia, Jessica Baiget, et al. · Journal of Medicinal Chemistry · 31
Coumarin-Annulated Ferrocenyl 1,3-Oxazine Derivatives Possessing In Vitro Antimalarial and Antitrypanosomal Potency
2021 · Mziyanda Mbaba, Laura M. K. Dingle, et al. · Molecules · 28
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New Quinolone-Based Thiosemicarbazones Showing Activity Against Plasmodium falciparum and Mycobacterium tuberculosis
2019 · Richard M. Beteck, Ronnett Seldon, et al. · Molecules · 25
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Indolyl-3-ethanone-α-thioethers: A promising new class of non-toxic antimalarial agents
2016 · Archibald L. Svogie, Michelle Isaacs, et al. · European Journal of Medicinal Chemistry · 23
Cinnamoyl-Oxaborole Amides: Synthesis and Their in Vitro Biological Activity
2018 · Maureen Gumbo, Richard M. Beteck, et al. · Molecules · 20
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New thiazolidine‐2,4‐dione derivatives combined with organometallic ferrocene: Synthesis, structure and antiparasitic activity
2018 · Ogunyemi O. Oderinlo, Matshawandile Tukulula, et al. · Applied Organometallic Chemistry · 20
Design, synthesis and biological evaluation of mono- and bisquinoline methanamine derivatives as potential antiplasmodial agents
2021 · Fostino R.B. Bokosi, Richard M. Beteck, et al. · Bioorganic & Medicinal Chemistry Letters · 19
Expanding the SAR of Nontoxic Antiplasmodial Indolyl‐3‐ethanone Ethers and Thioethers
2018 · Mayibongwe J. Lunga, Ruramai L. Chisango, et al. · ChemMedChem · 18
Anti-Trypanosomal and Antimalarial Properties of Tetralone Derivatives and Structurally Related Benzocycloalkanones
2019 · Richard M. Beteck, Lesetja J. Legoabe, et al. · Medicina · 17
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Gold(i) derived thiosemicarbazone complexes with rare halogen–halogen interaction–reduction of [Au(damp-C1,N)Cl2]
2010 · Setshaba D. Khanye, Nikoletta B. Báthori, et al. · Dalton Transactions · 16
Synthesis, Structure and In Vitro Anti-Trypanosomal Activity of Non-Toxic Arylpyrrole-Based Chalcone Derivatives
2020 · Ayanda I. Zulu, Ogunyemi O. Oderinlo, et al. · Molecules · 15
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A ring-closing metathesis approach to eight-membered benzannelated scaffolds and subsequent internal alkene isomerizations
2012 · Abu Taher, Blessing A. Aderibigbe, et al. · Tetrahedron · 15
The in Vitro Antiplasmodial and Antiproliferative Activity of New Ferrocene‐Based α‐Aminocresols Targeting Hemozoin Inhibition and DNA Interaction
2020 · Mziyanda Mbaba, Laura M. K. Dingle, et al. · ChemBioChem · 13
Facile synthesis and biological evaluation of assorted indolyl-3-amides and esters from a single, stable carbonyl nitrile intermediate
2015 · Clinton G.L. Veale, Adrienne L. Edkins, et al. · Tetrahedron Letters · 13
Hydrazone‐Tethered 5‐(Pyridin‐4‐yl)‐4H‐1,2,4‐triazole‐3‐thiol Hybrids: Synthesis, Characterisation, in silico ADME Studies, and in vitro Antimycobacterial Evaluation and Cytotoxicity
2023 · Ogunyemi O. Oderinlo, Audrey Jordaan, et al. · ChemMedChem · 12
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Works count: 136
Citation count: 889
H-index: 18
I10-index: 29
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