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Jacek Stalewski

GnRH Antagonists: A New Generation of Long Acting Analogues Incorporatingp-Ureido-phenylalanines at Positions 5 and 6
2000 · Guangcheng Jiang, Jacek Stalewski, et al. · Journal of Medicinal Chemistry · 109
Novel d-amino acid tetrapeptides produce potent antinociception by selectively acting at peripheral κ-opioid receptors,
2008 · Todd W. Vanderah, Tally Largent-Milnes, et al. · European Journal of Pharmacology · 104
Synthesis of 7,8-Dimethoxy-2-oxo-1,3,4,5-tetrahydropyrrolo[4,3,2-de]quinoline: A Key Intermediate en Route to Makaluvamines, Discorhabdin C and Other Marine Alkaloids of this Group via Vicarious Nucleophilic Substitution of Hydrogen
1997 · Mieczysław Mąkosza, Jacek Stalewski, et al. · Synthesis · 30
Synthesis of 1,3,4,5-tetrahydropyrrolo-[4,3,2-de]quinolines via the vicarious nucleophilic sybstitution of hydrogen
1995 · Mieczysław Ma̧kosza, Jacek Stalewski · Tetrahedron · 22
Synthesis of a 1,3,4,5-tetrahydrobenz[cd]indole via the Vicarious Nucleophilic substitution of hydrogen
1997 · Mieczysa̵w Ma̧jkosza, Jacek Stalewski, et al. · Tetrahedron · 15
The vicarious nucleophilic substitution of hydrogen and related reactions in nitrobenzoxazoles
1995 · Mieczysław Ma̧kosza, Jacek Stalewski · Tetrahedron · 13
Reactions of organic anions, 182. Vicarious nucleophilic substitution of a hydrogen atom in 1‐fluoro‐2,4‐dinitrobenzene (Sanger's Reagent)
1991 · Mieczyslaw Mąkosza, Jacek Stalewski · Liebigs Annalen der Chemie · 12
pH Dependence of a GPR4 Selective Antagonist Hampers Its Therapeutic Potential
2023 · Jacek Stalewski, Amy Y. Shih, et al. · Journal of Pharmacology and Experimental Therapeutics · 9
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Metabolite Profiles of Degarelix, a New Gonadotropin-Releasing Hormone Receptor Antagonist, in Rat, Dog, and Monkey
2011 · Anders Sonesson, Wolfgang Koechling, et al. · Drug Metabolism and Disposition · 8
The vicarious nucleophilic substitution of hydrogen proceeding via a cyclopropane ring-opening
1998 · Jacek Stalewski · Tetrahedron Letters · 8
Additive effect of simultaneous continuous administration of degarelix and TAK-448 on LH suppression in a castrated rat model
2018 · Jacek Stalewski, Diane M. Hargrove, et al. · European Journal of Pharmacology · 2
Novel, water soluble and long acting GnRH antagonists
2006 · Guangcheng Jiang, Jacek Stalewski, et al. · Kluwer Academic Publishers eBooks · 2
Identification of an Induced Orthosteric Pocket in IL-23: A New Avenue for Non-biological Therapeutic Targeting
2025 · Fabien C. Lecomte, Jeremiah S. Joseph, et al. · ACS Chemical Biology
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Abstract 588: Characterization of oncolytic peptides for local bladder cancer therapy
2020 · Amy Klova, Hiroe Tariga, et al. · Cancer Research
58. A peptide antagonist in a genetic rat angiotensinogen × renin model of preeclampsia
2018 · Nadine Haase, Kristin Kräker, et al. · Pregnancy Hypertension
ChemInform Abstract: The Vicarious Nucleophilic Substitution of Hydrogen Proceeding via a Cyclopropane Ring‐Opening.
1999 · Jacek Stalewski · ChemInform
ChemInform Abstract: Synthesis of 7,8‐Dimethoxy‐2‐oxo‐1,3,4,5‐tetrahydropyrrolo[4,3,2‐de]quinoline: A Key Intermediate en route to Makaluvamines, Discorhabdin C and Other Marine Alkaloids of this Group via Vicarious Nucleophilic Substitution of Hydrogen.
1998 · M. MAKOSZA, J. STALEWSKI, et al. · ChemInform
ChemInform Abstract: Synthesis of a 1,3,4,5‐Tetrahydrobenz(cd)indole via the Vicarious Nucleophilic Substitution of Hydrogen.
1997 · M. MAKOSZA, J. STALEWSKI, et al. · ChemInform
ChemInform Abstract: Synthesis of 1,3,4,5‐Tetrahydropyrrolo(4,3,2‐de)quinolines via the Vacarious Nucleophilic Substitution of Hydrogen.
1995 · M. MAKOSZA, J. STALEWSKI · ChemInform
ChemInform Abstract: The Vicarious Nucleophilic Substitution of Hydrogen and Related Reactions in Nitrobenzoxazoles.
1995 · M. MAKOSZA, J. STALEWSKI · ChemInform
Works count: 22
Citation count: 339
H-index: 8
I10-index: 7
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