Author

Davide Graziani

Observed names: D Graziani, D. Graziani

Observed institutions: Recordati (Italy), Dompé (Italy)

ORCID: 0000-0003-1826-5392

Observed ORCID: 0000-0003-1826-5392

OpenAlex ID: A5043805284

Discovery of a Novel Class of Selective Non-Peptide Antagonists for the Human Neurokinin-3 Receptor. 2. Identification of (S)-N-(1-Phenylpropyl)-3-hydroxy-2- phenylquinoline-4-carboxamide (SB 223412)

1999 · Giuseppe A. M. Giardina, Luca F. Raveglia, et al. · Journal of Medicinal Chemistry · 62

Selective δ opioid receptor agonists for inflammatory and neuropathic pain

2001 · Giulio Dondio, Silvano Ronzoni, et al. · Il Farmaco · 33

Replacement of the quinoline system in 2-phenyl-4-quinolinecarboxamide NK-3 receptor antagonists

1999 · G.A.M Giardina, M Artico, et al. · Il Farmaco · 21

Insights into the interaction of negative allosteric modulators with the metabotropic glutamate receptor 5: Discovery and computational modeling of a new series of ligands with nanomolar affinity

2015 · Andrew Anighoro, Davide Graziani, et al. · Bioorganic & Medicinal Chemistry · 17

Evaluation of Amides, Carbamates, Sulfonamides, and Ureas of 4-Prop-2-ynylidenecycloalkylamine as Potent, Selective, and Bioavailable Negative Allosteric Modulators of Metabotropic Glutamate Receptor 5

2019 · Davide Graziani, Silvia Caligari, et al. · Journal of Medicinal Chemistry · 14

The Approach of Conformational Chimeras to Model the Role of Proline‐Containing Helices on GPCR Mobility: the Fertile Case of Cys‐LTR1

2011 · Ilaria Bettinelli, Davide Graziani, et al. · ChemMedChem · 11

Transformation of a Potent C9-Substituted Phenylmorphan into MOR Partial Agonists with Improvement of Metabolic Stability: An In Vitro, In Vivo, and In Silico Study

2025 · Delmis E. Hernandez, Dan Luo, et al. · ACS Chemical Neuroscience · 2

Novel 5-Phenylmorphans as Opioid Receptor Antagonists: Synthesis, Structure-Activity Relationship, Biological Evaluation and Computational Modeling

2026 · Zahra Hasanpour, Dan Luo, et al. · Molecules

Beyond the Exscalate4CoV Project: LIGATE and REMEDI4ALL Projects

2023 · Carmine Talarico, Andrea R. Beccari, et al. · SpringerBriefs in applied sciences and technology

ChemInform Abstract: Selective δ Opioid Receptor Agonists for Inflammatory and Neuropathic Pain.

2001 · Giulio Dondio, Silvano Ronzoni, et al. · ChemInform

Works count: 11

Citation count: 160

H-index: 6

I10-index: 6