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Xiao-Yi Xiao

OpenAlex ID: A5055334054
Fluorocyclines. 1. 7-Fluoro-9-pyrrolidinoacetamido-6-demethyl-6-deoxytetracycline: A Potent, Broad Spectrum Antibacterial Agent
2011 · Xiao-Yi Xiao, Diana K. Hunt, et al. · Journal of Medicinal Chemistry · 125
Fluorocyclines. 2. Optimization of the C-9 Side-Chain for Antibacterial Activity and Oral Efficacy
2011 · Roger B. Clark, Diana K. Hunt, et al. · Journal of Medicinal Chemistry · 73
Synthesis and Antibacterial Activity of Pentacyclines: A Novel Class of Tetracycline Analogs
2011 · Cuixiang Sun, Diana K. Hunt, et al. · Journal of Medicinal Chemistry · 64
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Process R&D of Eravacycline: The First Fully Synthetic Fluorocycline in Clinical Development
2013 · Magnus Ronn, Zhijian Zhu, et al. · Organic Process Research & Development · 62
8-Azatetracyclines: Synthesis and Evaluation of a Novel Class of Tetracycline Antibacterial Agents
2011 · Roger B. Clark, Minsheng He, et al. · Journal of Medicinal Chemistry · 41
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Design and synthesis of thiazole-5-hydroxamic acids as novel histone deacetylase inhibitors
2007 · Sampath-Kumar Anandan, John S. Ward, et al. · Bioorganic & Medicinal Chemistry Letters · 30
Design, Synthesis, and Biological Evaluation of Hexacyclic Tetracyclines as Potent, Broad Spectrum Antibacterial Agents
2015 · Cuixiang Sun, Diana K. Hunt, et al. · Journal of Medicinal Chemistry · 17
Heterocyclyl Tetracyclines. 1. 7-Trifluoromethyl-8-Pyrrolidinyltetracyclines: Potent, Broad Spectrum Antibacterial Agents with Enhanced Activity against Pseudomonas aeruginosa
2017 · Yonghong Deng, Cuixiang Sun, et al. · Journal of Medicinal Chemistry · 15
Synthesis and Biological Evaluation of 8-Aminomethyltetracycline Derivatives as Novel Antibacterial Agents
2013 · Roger B. Clark, Minsheng He, et al. · Journal of Medicinal Chemistry · 14
Process Development and Scale-up of Fully Synthetic Tetracycline TP-2758: A Potent Antibacterial Agent with Excellent Oral Bioavailability
2015 · Wu-Yan Zhang, Cuixiang Sun, et al. · Organic Process Research & Development · 12
Fully Synthetic Tetracyclines: Increasing Chemical Diversity to Combat Multidrug-Resistant Bacterial Infections
2017 · Cuixiang Sun, Xiao-Yi Xiao · Topics in medicinal chemistry · 8
Heterocyclyl tetracyclines. 2. 7-Methoxy-8-pyrrolidinyltetracyclines: discovery of TP-2758, a potent, orally efficacious antimicrobial against Gram-negative pathogens
2017 · Cuixiang Sun, Yonghong Deng, et al. · The Journal of Antibiotics · 5
Synthesis Coupled to Scintillation Proximity Affinity Screening
1998 · Zahra Parandoosh, Sue K. Knowles, et al. · SLAS DISCOVERY · 2
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Abstract 3880: In vivo activities of TP-2846: a novel tetracycline antileukemia agent
2019 · Xiao-Yi Xiao, Cuixiang Sun, et al. · Cancer Research
Abstract 4802:In vitrocharacterization of TP-2846: a novel tetracycline antileukemia agent
2019 · Corey Fyfe, Joseph Newman, et al. · Experimental and Molecular Therapeutics
Abstract 3857: Discovery and structure-activity relationship studies of TP-2846: a novel tetracycline antileukemia agent
2019 · Cuixiang Sun, Peng Zhao, et al. · Experimental and Molecular Therapeutics
Abstract 4802: In vitro characterization of TP-2846: a novel tetracycline antileukemia agent
2019 · Corey Fyfe, Joseph Newman, et al. · Cancer Research
Abstract 3857: Discovery and structure-activity relationship studies of TP-2846: a novel tetracycline antileukemia agent
2019 · Cuixiang Sun, Peng Zhao, et al. · Cancer Research
Abstract 3880: In vivo activities of TP-2846: a novel tetracycline antileukemia agent
2019 · Xiao-Yi Xiao, Cuixiang Sun, et al. · Cancer Research
Works count: 19
Citation count: 468
H-index: 10
I10-index: 10
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