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Ester Colarusso
Observed names:
Colarusso, Ester,
E Colarusso
Institution:
University of Salerno
Observed institution:
University of Salerno
ORCID:
0000-0002-4193-1659
Observed ORCID:
0000-0002-4193-1659
OpenAlex ID:
A5058505465
Targeting mPGES-1 by a Combinatorial Approach: Identification of the Aminobenzothiazole Scaffold to Suppress PGE2 Levels
2020
·
Maria G. Chini
, Assunta Giordano
, et al.
·
ACS Medicinal Chemistry Letters
·
25
Essential Oils of Laurus nobilis L.: From Chemical Analysis to In Silico Investigation of Anti-Inflammatory Activity by Soluble Epoxide Hydrolase (sEH) Inhibition
2024
·
Francesca Fantasma
, Vadym Samukha
, et al.
·
Foods
·
22
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders
2022
·
Ester Colarusso
, Sara Ceccacci
, et al.
·
European Journal of Medicinal Chemistry
·
15
Identification and Development of BRD9 Chemical Probes
2024
·
Ester Colarusso
, Maria Giovanna Chini
, et al.
·
Pharmaceuticals
·
14
PDF
Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9
2023
·
Erica Gazzillo
, Martina Pierri
, et al.
·
Bioorganic Chemistry
·
14
6‐Methylquinazolin‐4(3H)‐one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis
2022
·
Ester Colarusso
, Erica Gazzillo
, et al.
·
European Journal of Organic Chemistry
·
11
PDF
5‐methyl‐2‐carboxamidepyrrole‐based novel dual mPGES‐1/sEH inhibitors as promising anticancer candidates
2024
·
Ester Colarusso
, Gianluigi Lauro
, et al.
·
Archiv der Pharmazie
·
10
PDF
Thiazolidin-4-one-based compounds interfere with the eicosanoid biosynthesis pathways by mPGES-1/sEH/5-LO multi-target inhibition
2022
·
Ester Colarusso
, Marianna Potenza
, et al.
·
European Journal of Medicinal Chemistry Reports
·
10
PDF
Chemical Profiling of Polar Lipids and the Polyphenolic Fraction of Commercial Italian Phaseolus Seeds by UHPLC-HRMS and Biological Evaluation
2024
·
Vadym Samukha
, Francesca Fantasma
, et al.
·
Biomolecules
·
8
PDF
Repositioning of Small Molecules through the Inverse Virtual Screening in silico Tool: Case of Benzothiazole‐Based Inhibitors of Soluble Epoxide Hydrolase (sEH)
2024
·
Erica Gazzillo
, Ester Colarusso
, et al.
·
ChemPlusChem
·
8
PharmaCore: The Automatic Generation of 3D Structure-Based Pharmacophore Models from Protein/Ligand Complexes
2024
·
Simona De Vita
, Ester Colarusso
, et al.
·
Journal of Chemical Information and Modeling
·
7
Marine Natural Products in Preclinical Cancer Studies: Ten Years of Advanced Total Synthesis
2025
·
Ester Colarusso
, Assunta Giordano
, et al.
·
Marine Drugs
·
5
PDF
In Silico Design, Chemical Synthesis, Biophysical and in Vitro Evaluation for the Identification of 1‐Ethyl‐1H‐Pyrazolo[3,4‐b]Pyridine‐Based BRD9 Binders
2024
·
Ester Colarusso
, Erica Gazzillo
, et al.
·
ChemPlusChem
·
4
Identification of Novel Bromodomain-Containing Protein 4 (BRD4) Binders through 3D Pharmacophore-Based Repositioning Screening Campaign
2024
·
Ester Colarusso
, Erica Gazzillo
, et al.
·
Molecules
·
3
PDF
Potential Nutraceutical Properties of Vicia faba L: LC-ESI-HR-MS/MS-Based Profiling of Ancient Faba Bean Varieties and Their Biological Activity
2026
·
Francesca Fantasma
, Gilda D’Urso
, et al.
·
Molecules
·
2
PDF
Unveiling New Triazoloquinoxaline‐Based PROTACs Designed for the Selective Degradation of the ncBAF Chromatin Remodeling Subunit BRD9
2025
·
Martina Pierri
, Guglielmo Bove
, et al.
·
Chemistry - A European Journal
·
2
PDF
2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines
2023
·
Simona De Vita
, Sara Meninno
, et al.
·
Bioorganic & Medicinal Chemistry
·
2
Phytochemical analysis of Laurus nobilis L. leaves essential oil: rationalization of antioxidant and anti-inflammatory activities by combined in vitro and in silico approach
2025
·
Francesca Fantasma
, Vadym Samukha
, et al.
·
Phytochemistry Letters
·
1
Untargeted Diversity-Oriented Synthesis for the Discovery of New Antitumor Agents: An Integrated Approach of Inverse Virtual Screening, Bioinformatics, and Omics for Target Deconvolution
2025
·
Tania Ciaglia
, Valeria Napolitano
, et al.
·
Journal of Medicinal Chemistry
·
1
Anti-Inflammatory Activity of Monoterpene Phenol Dimers from Satureja bachtiarica
2026
·
Simone Di Micco
, Milena Masullo
, et al.
·
ACS Omega
PDF
Exploring the Anti-Inflammatory Potential of Daucus carota L. subsp. carota Seed Extracts: Phytochemical Profiling, In Vitro Antioxidant Activity and Modulation of the Arachidonic Acid Cascade
2026
·
Monica Maio
, Gilda D’Urso
, et al.
·
Plants
PDF
Repositioning of 3-(isoxazol-3-yl)thiazolidin-4-one-based compounds via Inverse Virtual Screening: discovery of new ERα inhibitors with in vitro activity in breast cancer models
2026
·
Ester Colarusso
, Simona De Vita
, et al.
·
European Journal of Medicinal Chemistry
Biological assessment and phytochemical investigation of commercial bean varieties by NMR and LC-ESI-HR-MS analysis
2026
·
G D’Urso
, F Fantasma
, et al.
·
Planta Medica
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Works count:
24
Citation count:
164
H-index:
8
I10-index:
8
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