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Nora R. Vail

Observed names: N.R. Vail, Nora R. Vail, Nora Vail, Vail, Nora
OpenAlex ID: A5059564608
4-Methyl-1,2,3-Triazoles as N -Acetyl-Lysine Mimics Afford Potent BET Bromodomain Inhibitors with Improved Selectivity
2021 · Huarui Cui, Angela S. Carlson, et al. · Journal of Medicinal Chemistry · 37
Efficacy and Toxicity Analysis of Selective BET Bromodomain Inhibitors in Models of Inflammatory Liver Disease
2025 · Luke C. Doskey, Cole R. Scholtz, et al. · Journal of Medicinal Chemistry · 7
Design, synthesis, and evaluation of transition-state analogs as inhibitors of the bacterial quorum sensing autoinducer synthase CepI
2021 · Erin L. Higgins, Julian S. Kellner-Rogers, et al. · Bioorganic & Medicinal Chemistry Letters · 7
Development of cell-active BRD4-D1 selective inhibitors to decode the role of BET proteins in LPS-mediated liver inflammation
2025 · Cole R. Scholtz, Luke C. Doskey, et al. · European Journal of Medicinal Chemistry · 3
BET Bromodomain Pan-D1-Biased Inhibitors with Improved Drug-Like Properties and hERG Profiles as Therapies for Inflammatory Liver Injury
2026 · Nora R. Vail, Luke C. Doskey, et al. · ChemRxiv
Development of Cell-Active BRD4-D1 Selective Inhibitors to Decode the Role of BET Proteins in LPS-Mediated Liver Inflammation
2025 · William Pomerantz, Cole R. Scholtz, et al. · SSRN Electronic Journal
CCDC 2000389: Experimental Crystal Structure Determination
2022 · Porter, Matthew R., Xiao, Haiyan, et al. · The Cambridge Structural Database
CCDC 2000390: Experimental Crystal Structure Determination
2022 · Porter, Matthew R., Xiao, Haiyan, et al. · The Cambridge Structural Database
X-ray crystal structure of human BRD4(D1) in complex with 2-(4-{5-[6-(2,5-dibromophenoxy)pyridin-2-yl]-4-methyl-1H-1,2,3-triazol-1-yl}piperidin-1-yl)-N,N-dimethylethan-1-amine (compound 26)
2021 · H. Cui, J.A. Johnson, et al. · Worldwide Protein Data Bank
Enhanced Affinity for 3-Amino-Chromane-Derived σ1 Receptor Ligands
2020 · Matthew R. Porter, Haiyan Xiao, et al. · ACS Omega
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Works count: 10
Citation count: 54
H-index: 3
I10-index: 1
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