Author

Francesco Saccoliti

Observed names: Saccoliti F, Saccoliti, F., Saccoliti, Francesco

Observed institutions: Italian Institute of Technology, Istituto Pasteur, Link Campus University, Sapienza University of Rome

ORCID: 0000-0002-2907-5503

Observed ORCID: 0000-0002-2907-5503

OpenAlex ID: A5061072881

Structure–Activity Relationship of Pyrrolyl Diketo Acid Derivatives as Dual Inhibitors of HIV-1 Integrase and Reverse Transcriptase Ribonuclease H Domain

2015 · Giuliana Cuzzucoli Crucitti, Mathieu Métifiot, et al. · Journal of Medicinal Chemistry · 83

Inhibition of Leishmania infantum trypanothione reductase by diaryl sulfide derivatives

2017 · Francesco Saccoliti, Gabriella Angiulli, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 76

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Comparison of different methods for the extraction of cannabinoids from cannabis

2019 · Daniela De Vita, Valentina Noemi Madia, et al. · Natural Product Research · 53

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N-Substituted Quinolinonyl Diketo Acid Derivatives as HIV Integrase Strand Transfer Inhibitors and Their Activity against RNase H Function of Reverse Transcriptase

2015 · Luca Pescatori, Mathieu Métifiot, et al. · Journal of Medicinal Chemistry · 53

Investigation of Commiphora myrrha (Nees) Engl. Oil and Its Main Components for Antiviral Activity

2021 · Valentina Noemi Madia, Marta De Angelis, et al. · Pharmaceuticals · 47

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Pyrrolyl Pyrazoles as Non-Diketo Acid Inhibitors of the HIV-1 Ribonuclease H Function of Reverse Transcriptase

2020 · Antonella Messore, Angela Corona, et al. · ACS Medicinal Chemistry Letters · 42

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Design, Synthesis and Biological Evaluation of New Pyrimidine Derivatives as Anticancer Agents

2021 · Valentina Noemi Madia, Alice Nicolai, et al. · Molecules · 37

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Design, Synthesis, and Biological Evaluation of New 1-(Aryl-1H-pyrrolyl)(phenyl)methyl-1H-imidazole Derivatives as Antiprotozoal Agents

2019 · Francesco Saccoliti, Valentina Noemi Madia, et al. · Journal of Medicinal Chemistry · 36

Effect of heparanase inhibitor on tissue factor overexpression in platelets and endothelial cells induced by anti‐β2‐GPI antibodies

2021 · Antonella Capozzi, Gloria Riitano, et al. · Journal of Thrombosis and Haemostasis · 35

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Tegaserod for the Treatment of Irritable Bowel Syndrome

2019 · Valentina Noemi Madia, Antonella Messore, et al. · Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry · 35

Novel Benzazole Derivatives Endowed with Potent Antiheparanase Activity

2018 · Valentina Noemi Madia, Antonella Messore, et al. · Journal of Medicinal Chemistry · 35

Recent Advancement in the Search of Innovative Antiprotozoal Agents Targeting Trypanothione Metabolism

2020 · Francesco Saccoliti, Roberto Di Santo, et al. · ChemMedChem · 33

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Structure-guided approach to identify a novel class of anti-leishmaniasis diaryl sulfide compounds targeting the trypanothione metabolism

2019 · Gianni Colotti, Francesco Saccoliti, et al. · Amino Acids · 29

Biological evaluation and structure-activity relationships of imidazole-based compounds as antiprotozoal agents

2018 · Francesco Saccoliti, Valentina Noemi Madia, et al. · European Journal of Medicinal Chemistry · 29

Inhibition of Polycomb Repressive Complex 2 activity reduces trimethylation of H3K27 and affects development in Arabidopsis seedlings

2019 · Veronica Ruta, Chiara Longo, et al. · BMC Plant Biology · 27

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Novel Symmetrical Benzazolyl Derivatives Endowed with Potent Anti-Heparanase Activity

2018 · Antonella Messore, Valentina Noemi Madia, et al. · Journal of Medicinal Chemistry · 25

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Discovery of a pyrimidine compound endowed with antitumor activity

2019 · Ludovica Taglieri, Francesco Saccoliti, et al. · Investigational New Drugs · 23

New Thiazolidine-4-One Derivatives as SARS-CoV-2 Main Protease Inhibitors

2024 · Antonella Messore, Paolo Malune, et al. · Pharmaceuticals · 20

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Analytical Characterization of an Inulin-Type Fructooligosaccharide from Root-Tubers of Asphodelusramosus L

2021 · Valentina Noemi Madia, Daniela De Vita, et al. · Pharmaceuticals · 19

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Discovery of N-aryl-naphthylamines as in vitro inhibitors of the interaction between HIV integrase and the cofactor LEDGF/p75

2015 · Giuliana Cuzzucoli Crucitti, Luca Pescatori, et al. · European Journal of Medicinal Chemistry · 19

Miconazole-like Scaffold is a Promising Lead for Naegleria fowleri-Specific CYP51 Inhibitors

2023 · Vandna Sharma, Valentina Noemi Madia, et al. · Journal of Medicinal Chemistry · 18

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Quinolinonyl Non-Diketo Acid Derivatives as Inhibitors of HIV-1 Ribonuclease H and Polymerase Functions of Reverse Transcriptase

2021 · Antonella Messore, Angela Corona, et al. · Journal of Medicinal Chemistry · 17

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Inhibition of Leishmania infantum Trypanothione Reductase by New Aminopropanone Derivatives Interacting with the NADPH Binding Site

2023 · Valentina Noemi Madia, Davide Ialongo, et al. · Molecules · 15

In Vitro Antiviral Activity of New Oxazoline Derivatives as Potent Poliovirus Inhibitors

2018 · Valentina Noemi Madia, Antonella Messore, et al. · Journal of Medicinal Chemistry · 15

Small-molecule Inhibitors of HIV-1 Reverse Transcriptase-Associated Ribonuclease H Function: Challenges and Recent Developments

2021 · Valentina Noemi Madia, Antonella Messore, et al. · Current Medicinal Chemistry · 12

Works count: 47

Citation count: 874

H-index: 19

I10-index: 26