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Kevin M. Peese

Observed names: K. Peese, Kevin M Peese, Kevin Peese, Kevin M. Peese, Peese, K.M.
ORCID: 0000-0001-5349-8779
Observed ORCID: 0000-0001-5349-8779
OpenAlex ID: A5062228382
Glutathione S-Transferase Omega 1-1 Is a Target of Cytokine Release Inhibitory Drugs and May Be Responsible for Their Effect on Interleukin-1औ Posttranslational Processing
2003 · Ronald E. Laliberte, David G. Perregaux, et al. · Journal of Biological Chemistry · 213
Efficient Synthetic Access to the Hetisine C20-Diterpenoid Alkaloids. A Concise Synthesis of Nominine via Oxidoisoquinolinium-1,3-Dipolar and Dienamine-Diels−Alder Cycloadditions
2006 · Kevin M. Peese, David Y. Gin · Journal of the American Chemical Society · 120
Asymmetric Synthetic Access to the Hetisine Alkaloids: Total Synthesis of (+)‐Nominine
2007 · Kevin M. Peese, David Y. Gin · Chemistry - A European Journal · 98
New first and second generation inhibitors of human immunodeficiency virus-1 integrase
2011 · Annapurna Pendri, Nicholas A Meanwell, et al. · Expert Opinion on Therapeutic Patents · 55
Enantioselective Approach to the Hetisine Alkaloids. Synthesis of the 3-Methyl-1-aza-tricyclo[5.2.1.03,8]decane Core via Intramolecular Dipolar Cycloaddition
2005 · Kevin M. Peese, David Y. Gin · Organic Letters · 44
5,6,7,8-Tetrahydro-1,6-naphthyridine Derivatives as Potent HIV-1-Integrase-Allosteric-Site Inhibitors
2019 · Kevin M. Peese, Christopher W. Allard, et al. · Journal of Medicinal Chemistry · 38
Tandem Ring-Closing Metathesis/Transfer Hydrogenation: Practical Chemoselective Hydrogenation of Alkenes
2014 · Timothy Connolly, Zhongyu Wang, et al. · Organic Letters · 35
Potent Long-Acting Inhibitors Targeting the HIV-1 Capsid Based on a Versatile Quinazolin-4-one Scaffold
2023 · Eric P. Gillis, Kyle Parcella, et al. · Journal of Medicinal Chemistry · 31
Benzimidazolone p38 inhibitors
2004 · Mark A. Dombroski, Michael A. Letavic, et al. · Bioorganic & Medicinal Chemistry Letters · 30
Structure–activity relationships of triazolopyridine oxazole p38 inhibitors: Identification of candidates for clinical development
2006 · Kim F. McClure, Michael A. Letavic, et al. · Bioorganic & Medicinal Chemistry Letters · 29
General Method for the Preparation of Electron-Deficient Imidazo[1,2-a]pyridines and Related Heterocycles
2015 · Ivar M. McDonald, Kevin M. Peese · Organic Letters · 28
New agents for the treatment of leukemia: discovery of DMAPT (LC-1)
2009 · Kevin Peese · Drug Discovery Today · 26
Exploring HIV-1 Maturation: A New Frontier in Antiviral Development
2024 · Aidan McGraw, Grace Hillmer, et al. · Viruses · 18
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Discovery and Preclinical Profiling of GSK3839919, a Potent HIV-1 Allosteric Integrase Inhibitor
2022 · Kyle Parcella, Tao Wang, et al. · ACS Medicinal Chemistry Letters · 12
Synthesis of (±)-Nominine
2006 · D. Gin, K. Peese · Synfacts · 12
To Market, to Market—2018: Small Molecules
2019 · Erika Araujo, Marie-Gabrielle Braun, et al. · Medicinal chemistry reviews · 11
Heterocycle amide isosteres: An approach to overcoming resistance for HIV-1 integrase strand transfer inhibitors
2019 · Kevin M. Peese, B. Narasimhulu Naidu, et al. · Bioorganic & Medicinal Chemistry Letters · 11
To Market, To Market--2014
2015 · Joanne Bronson, Kevin Peese, et al. · Medicinal chemistry reviews · 9
Scaffold modifications to the 4-(4,4-dimethylpiperidinyl) 2,6-dimethylpyridinyl class of HIV-1 allosteric integrase inhibitors
2022 · Kyle Parcella, Manoj Patel, et al. · Bioorganic & Medicinal Chemistry · 8
Structure-based amelioration of PXR transactivation in a novel series of macrocyclic allosteric inhibitors of HIV-1 integrase
2020 · Prasanna Sivaprakasam, Zhongyu Wang, et al. · Bioorganic & Medicinal Chemistry Letters · 8
To Market, To Market--2015
2016 · Joanne Bronson, Kevin Peese, et al. · Medicinal chemistry reviews · 8
To Market, to Market–2021: Small Molecules
2022 · Erika Araujo, Ian M. Bell, et al. · Medicinal chemistry reviews · 7
To Market, To Market--2016
2017 · Catherine A. Bolger, T.G. Murali Dhar, et al. · Medicinal chemistry reviews · 5
To Market, to Market–2022: Small Molecules
2023 · Erika Araujo, Ian M. Bell, et al. · Medicinal chemistry reviews · 4
DNA-Model-Based Design and Execution of Some Fused Benzodiazepine Hybrid Payloads for Antibody–Drug Conjugate Modality
2021 · Prasanna Sivaprakasam, Ivar McDonald, et al. · ACS Medicinal Chemistry Letters · 4
Works count: 42
Citation count: 885
H-index: 13
I10-index: 17
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