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Author

Takafumi Yukawa

Observed name: Yukawa, Takafumi
ORCID: 0000-0003-2685-2909
Observed ORCID: 0000-0003-2685-2909
OpenAlex ID: A5065791689
Catalytic Asymmetric Aza-Morita−Baylis−Hillman Reaction of Methyl Acrylate: Role of a Bifunctional La(O-iPr)3/Linked-BINOL Complex
2010 · Takafumi Yukawa, Bianca Seelig, et al. · Journal of the American Chemical Society · 79
Lewis Base Assisted Brønsted Base Catalysis: Bidentate Phosphine Oxides as Activators and Modulators of Brønsted Basic Lanthanum–Aryloxides
2008 · Hiroyuki Morimoto, Tatsuhiko Yoshino, et al. · Angewandte Chemie International Edition · 58
Development of a Highly Selective Plasmodium falciparum Proteasome Inhibitor with Anti‐malaria Activity in Humanized Mice
2021 · Wenhu Zhan, Hao Zhang, et al. · Angewandte Chemie International Edition · 46
Discovery and optimization of 1,7-disubstituted-2,2-dimethyl-2,3-dihydroquinazolin-4(1H)-ones as potent and selective PKCθ inhibitors
2016 · Taisuke Katoh, Takafumi Takai, et al. · Bioorganic & Medicinal Chemistry · 29
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Design, Synthesis, and Optimization of Macrocyclic Peptides as Species-Selective Antimalaria Proteasome Inhibitors
2022 · Hao Zhang, John Ginn, et al. · Journal of Medicinal Chemistry · 25
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Direct and Regioselective Monofluorination of N-Protected Pyridone Derivatives using N-Fluorobenzenesulfonimide (NFSI)
2019 · Fumie Sakurai, Takafumi Yukawa, et al. · Organic Letters · 24
Macrocyclic Peptides that Selectively Inhibit the Mycobacterium tuberculosis Proteasome
2021 · Hao Zhang, Hao-Chi Hsu, et al. · Journal of Medicinal Chemistry · 19
Structure–Activity Relationship Studies of Antimalarial Plasmodium Proteasome Inhibitors─Part II
2023 · Hao Zhang, John Ginn, et al. · Journal of Medicinal Chemistry · 18
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Lewis Base Assisted Brønsted Base Catalysis: Bidentate Phosphine Oxides as Activators and Modulators of Brønsted Basic Lanthanum–Aryloxides
2008 · Hiroyuki Morimoto, Tatsuhiko Yoshino, et al. · Angewandte Chemie · 15
Discovery of 1,8-naphthyridin-2-one derivative as a potent and selective sphingomyelin synthase 2 inhibitor
2020 · Takafumi Yukawa, Takashi Nakahata, et al. · Bioorganic & Medicinal Chemistry · 11
Discovery of Pyrazolo[1,5-a]pyrazin-4-ones as Potent and Brain Penetrant GluN2A-Selective Positive Allosteric Modulators Reducing AMPA Receptor Binding Activity
2021 · Fumie Sakurai, Takafumi Yukawa, et al. · Bioorganic & Medicinal Chemistry · 9
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Development of a Highly Selective Plasmodium falciparum Proteasome Inhibitor with Anti‐malaria Activity in Humanized Mice
2021 · Wenhu Zhan, Hao Zhang, et al. · Angewandte Chemie · 6
2 H -Thiazolo[4,5- d ][1,2,3]triazole: synthesis, functionalization, and application in scaffold-hopping
2024 · Ryuya Miyazaki, Fumito Takada, et al. · Chemical Science · 4
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Design and synthesis of 6-methylpyridin-2-one derivatives as novel and potent GluN2A positive allosteric modulators for the treatment of cognitive impairment
2022 · Takafumi Yukawa, Tohru Yamashita, et al. · Bioorganic & Medicinal Chemistry · 2
Structure–Activity Relationship Study of Antimalarial Asparagine-Derived Proteasome Inhibitors
2026 · Hao Zhang, Daqiang Li, et al. · ACS Omega
CCDC 2120146: Experimental Crystal Structure Determination
2021 · Sakurai, Fumie, Yukawa, Takafumi, et al. · The Cambridge Structural Database
CCDC 1968615: Experimental Crystal Structure Determination
2020 · Yukawa, Takafumi, Nakahata, Takashi, et al. · The Cambridge Structural Database
ChemInform Abstract: Catalytic Asymmetric Aza‐Morita—Baylis—Hillman Reaction of Methyl Acrylate: Role of a Bifunctional La(OiPr)3/Linked BINOL Complex.
2011 · Takafumi Yukawa, Bianca Seelig, et al. · ChemInform
ChemInform Abstract: Lewis Base Assisted Broensted Base Catalysis: Bidentate Phosphine Oxides as Activators and Modulators of Broensted Basic Lanthanum—Aryloxides.
2009 · Hiroyuki Morimoto, Tatsuhiko Yoshino, et al. · ChemInform
Works count: 21
Citation count: 345
H-index: 10
I10-index: 10
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