Author

Marc Capet

Observed names: Capet, Marc, M. CAPET, M. Capet

Observed institutions: Western University, Centre National de la Recherche Scientifique, Université de Haute-Alsace, École Normale Supérieure - PSL, Bioprojet (France), Université Rennes 1, Université de Rennes

ORCID: 0000-0003-4826-0736

Observed ORCID: 0000-0003-4826-0736

OpenAlex ID: A5070569366

Histamine and tele-methylhistamine quantification in cerebrospinal fluid from narcoleptic subjects by liquid chromatography tandem mass spectrometry with precolumn derivatization

2010 · Mikaël Croyal, Yves Dauvilliers, et al. · Analytical Biochemistry · 45

Congo Red protects against toxicity of β-amyloid peptides on rat hippocampal neurones

1994 · Marie-Claude Burgevin, Marylène Passat, et al. · Neuroreport · 44

Refined Docking as a Valuable Tool for Lead Optimization: Application to Histamine H3 Receptor Antagonists

2008 · Nicolas Levoin, Thierry Calmels, et al. · Archiv der Pharmazie · 38

Psychopharmacological Agents

2000 · Marie-Christine Dubroeucq, Jean-Marie Stutzmann, et al. · Ullmann's Encyclopedia of Industrial Chemistry · 37

Pharmacological properties of ureido-acetamides, new potent and selective non-peptide CCKB/gastrin receptor antagonists

1994 · Philippe Bertrand, G.Andrees Böhme, et al. · European Journal of Pharmacology · 36

Unexpected Formation of Aryl Ketones by Palladium-Catalyzed Coupling of Aryl Bromides with Vinylic Acetates

2007 · Mickaël Jean, Jacques Renault, et al. · Organic Letters · 32

Fluorinated non-imidazole histamine H3 receptor antagonists

2009 · K. Isensee, M. Amon, et al. · Bioorganic & Medicinal Chemistry Letters · 29

Homology Model Versus X-ray Structure in Receptor-based Drug Design: A Retrospective Analysis with the Dopamine D3 Receptor

2011 · Nicolas Levoin, Thierry Calmels, et al. · ACS Medicinal Chemistry Letters · 22

Interaction of brain cannabinoid receptors with guanine nucleotide binding protein

1997 · François Petitet, Bernadette Jeantaud, et al. · Biochemical Pharmacology · 22

Syntheses with sulfones L: Preparation of β-hydroxysulfones through the combined oxidative desulfonylation/condensation reaction of sulfonyl anions. Application to terpene synthesis.

1987 · M. Capet, T. Cuvigny, et al. · Tetrahedron Letters · 22

Exploring occupancy of the histamine H3 receptor by pitolisant in humans using PET

2020 · Pablo Rusjan, Pamela Sabioni, et al. · British Journal of Pharmacology · 21

Novel and highly potent histamine H3 receptor ligands. Part 1: withdrawing of hERG activity

2011 · Nicolas Levoin, Olivier Labeeuw, et al. · Bioorganic & Medicinal Chemistry Letters · 21

Parallel synthesis and dopamine D3/D2 receptor screening of novel {4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}carboxamides

2005 · Philipp Heidler, Vida Zohrabi-Kalantari, et al. · Bioorganic & Medicinal Chemistry · 15

Determination of the binding mode and interacting amino-acids for dibasic H3 receptor antagonists

2013 · Nicolas Levoin, Olivier Labeeuw, et al. · Bioorganic & Medicinal Chemistry · 13

Discovery of nanomolar ligands with novel scaffolds for the histamine H4 receptor by virtual screening

2016 · Nicolas Levoin, Olivier Labeeuw, et al. · European Journal of Medicinal Chemistry · 11

Novel and highly potent histamine H3 receptor ligands. Part 3: An alcohol function to improve the pharmacokinetic profile

2013 · Olivier Labeeuw, Nicolas Levoin, et al. · Bioorganic & Medicinal Chemistry Letters · 10

A Two-Step Synthesis of Camphosultam

1995 · M. Capet, F. David, et al. · Synthetic Communications · 10

The Ureidoacetamides, a Novel Family of Non‐peptide CCK‐B/Gastrin Antagonists

1994 · G. A. BÖHME, P. BERTRAND, et al. · Annals of the New York Academy of Sciences · 10

Synthesis and evaluation of a 2-benzothiazolylphenylmethyl ether class of histamine H4 receptor antagonists

2016 · Olivier Labeeuw, Nicolas Levoin, et al. · Bioorganic & Medicinal Chemistry Letters · 9

Novel and highly potent histamine H3 receptor ligands. Part 2: Exploring the cyclohexylamine-based series

2011 · Olivier Labeeuw, Nicolas Levoin, et al. · Bioorganic & Medicinal Chemistry Letters · 9

Synthesis and evaluation of amides surrogates of dopamine D3 receptor ligands

2010 · Mickaël Jean, Jacques Renault, et al. · Bioorganic & Medicinal Chemistry Letters · 8

Improving selectivity of dopamine D3 receptor ligands

2015 · Marc Capet, Thierry Calmels, et al. · Bioorganic & Medicinal Chemistry Letters · 7

Determination of the absolute configuration of fasidotril, a potent dual ACE/NEP inhibitor

2003 · V. Grosset, D. Danvy, et al. · Tetrahedron Asymmetry · 4

Novel pyrrolidinone derivative lacks claimed histamine H3 receptor stimulation in receptor binding and functional studies

2020 · David Reiner, Aleksandra Zivkovic, et al. · European Journal of Medicinal Chemistry · 3

A solid phase parallel synthesis of diverse amides as dopamine D3receptor ligands

2008 · Mickaël Jean, Jacques Renault, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 3

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Works count: 39

Citation count: 485

H-index: 13

I10-index: 18