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Val S. Goodfellow
Observed names:
Goodfellow, V.S.,
Goodfellow, Val S.,
V. Goodfellow,
V. S. Goodfellow,
V.S. Goodfellow,
VAL S. GOODFELLOW,
Val Goodfellow,
Val S Goodfellow
show all 8
Observed institutions:
University of Michigan,
University of Rochester Medicine,
Bristol-Myers Squibb (United States),
Califia Bio (United States),
University of Rochester,
Neurocrine Biosciences (United States)
show all 6
OpenAlex ID:
A5074490683
Mixed lineage kinase 3 mediates release of C‐X‐C motif ligand 10–bearing chemotactic extracellular vesicles from lipotoxic hepatocytes
2015
·
Samar H. Ibrahim
, Petra Hirsova
, et al.
·
Hepatology
·
232
Discovery, Synthesis, and Characterization of an Orally Bioavailable, Brain Penetrant Inhibitor of Mixed Lineage Kinase 3
2013
·
Val S. Goodfellow
, Colin J. Loweth
, et al.
·
Journal of Medicinal Chemistry
·
86
The New Small-Molecule Mixed-Lineage Kinase 3 Inhibitor URMC-099 Is Neuroprotective and Anti-Inflammatory in Models of Human Immunodeficiency Virus-Associated Neurocognitive Disorders
2013
·
D. F. Marker
, M.-E. Tremblay
, et al.
·
Journal of Neuroscience
·
66
PDF
Potent imidazole and triazole CB 1 receptor antagonists related to SR141716
2004
·
Brian Dyck
, Val S. Goodfellow
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
66
Aryl piperazine melanocortin MC4 receptor agonists
2003
·
Brian Dyck
, Jessica Parker
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
47
A Thienopyridazinone-Based Melanin-Concentrating Hormone Receptor 1 Antagonist with Potent in Vivo Anorectic Properties
2006
·
Brian Dyck
, Stacy Markison
, et al.
·
Journal of Medicinal Chemistry
·
43
The Melanocortin System and its Role in Obesity and Cachexia
2003
·
Val Goodfellow
, John Saunders
·
Current Topics in Medicinal Chemistry
·
40
Potent and orally active non-peptide antagonists of the human melanocortin-4 receptor based on a series of trans-2-disubstituted cyclohexylpiperazines
2005
·
Fabio C. Tucci
, Nicole S. White
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
32
1-(4-Amino-phenyl)-pyrrolidin-3-yl-amine and 6-(3-amino-pyrrolidin-1-yl)-pyridin-3-yl-amine derivatives as melanin-concentrating hormone receptor-1 antagonists
2005
·
Charles Q. Huang
, Tracy Baker
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
32
The mixed lineage kinase-3 inhibitor URMC-099 improves therapeutic outcomes for long-acting antiretroviral therapy
2015
·
Gang Zhang
, Dongwei Guo
, et al.
·
Nanomedicine Nanotechnology Biology and Medicine
·
31
PDF
Assessment of a small molecule melanocortin-4 receptor-specific agonist on energy homeostasis
2004
·
David Cepoi
, Teresa Phillips
, et al.
·
Brain Research
·
31
Rationally designed non-peptides: Variously substituted piperazine libraries for the discovery of bradykinin antagonists and other G-protein-coupled receptor ligands
1996
·
Val S. Goodfellow
, Chris P. Laudeman
, et al.
·
Molecular Diversity
·
30
Bradykinin Receptor Antagonists Containing N-Substituted Amino Acids: In Vitro and in Vivo B2 and B1 Receptor Antagonist Activity
1996
·
Val S. Goodfellow
, Manoj V. Marathe
, et al.
·
Journal of Medicinal Chemistry
·
29
Body Weight Regulation by Selective MC4 Receptor Agonists and Antagonists
2003
·
ALAN C. FOSTER
, MARGARET JOPPA
, et al.
·
Annals of the New York Academy of Sciences
·
28
MLK3 regulates fMLP-stimulated neutrophil motility
2014
·
Oksana Polesskaya
, Christopher Wong
, et al.
·
Molecular Immunology
·
24
Thienopyrimidinone bis-aminopyrrolidine ureas as potent melanin-concentrating hormone receptor-1 (MCH-R1) antagonists
2007
·
Mingzhu Zhang
, Junko Tamiya
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
22
Bis(aminopyrrolidine)-derived ureas (APUs) as potent MCH1 receptor antagonists
2005
·
Jonathan Grey
, Brian Dyck
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
22
p-Nitrophenyl 3-diazopyruvate and diazopyruvamides, a new family of photoactivatable cross-linking bioprobes
1989
·
Val S. Goodfellow
, Marc Settineri
, et al.
·
Biochemistry
·
20
Substituted chromones and quinolones as potent melanin-concentrating hormone receptor 1 antagonists
2006
·
Brian Dyck
, Liren Zhao
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
17
Synthesis and structure–activity relationships of biarylcarboxamide bis-aminopyrrolidine urea derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1)
2005
·
Martin W. Rowbottom
, Troy D. Vickers
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
16
The second generation mixed lineage kinase-3 (MLK3) inhibitor CLFB-1134 protects against neurotoxin-induced nigral dopaminergic neuron loss
2019
·
Elizabeth M. Kline
, Laura M. Butkovich
, et al.
·
Experimental Neurology
·
13
Differences in antiviral activities for isomers of a fluorinated cyclobutane nucleoside analog
1993
·
G.D. Vite
, J.A. Tino
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
13
Synthesis and structure–activity relationships of retro bis-aminopyrrolidine urea (rAPU) derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1). Part 2
2006
·
Sarah Hudson
, Mehrak Kiankarimi
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
11
Synthesis and structure–activity relationships of spirohydantoin-derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1)
2007
·
Martin W. Rowbottom
, Troy D. Vickers
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
9
Synthesis and structure–activity relationships of retro bis-aminopyrrolidine urea (rAPU) derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1). Part 1
2006
·
Martin W. Rowbottom
, Troy D. Vickers
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
8
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Works count:
39
Citation count:
982
H-index:
18
I10-index:
23
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