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Amr Hassan

Observed names: A Q Hassan, A Quamrul Hassan, A. Quamrul Hassan, A. Quamrul Hassan, A. Quamrul Hassan, Asm Quamrul Hassan
ORCID: 0000-0001-6623-2179
Observed ORCID: 0000-0001-6623-2179
OpenAlex ID: A5075196845
The allosteric inhibitor ABL001 enables dual targeting of BCR–ABL1
2017 · Andrew A. Wylie, Joseph Schoepfer, et al. · Nature · 615
Discovery of Asciminib (ABL001), an Allosteric Inhibitor of the Tyrosine Kinase Activity of BCR-ABL1
2018 · Joseph Schoepfer, Wolfgang Jahnke, et al. · Journal of Medicinal Chemistry · 454
Development of secondary mutations in wild-type and mutant EZH2 alleles cooperates to confer resistance to EZH2 inhibitors
2015 · V Gibaja, F Shen, et al. · Oncogene · 147
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The Novolactone Natural Product Disrupts the Allosteric Regulation of Hsp70
2014 · A. Quamrul Hassan, Christina A. Kirby, et al. · Chemistry & Biology · 64
Design and Discovery of N-(3-(2-(2-Hydroxyethoxy)-6-morpholinopyridin-4-yl)-4-methylphenyl)-2-(trifluoromethyl)isonicotinamide, a Selective, Efficacious, and Well-Tolerated RAF Inhibitor Targeting RAS Mutant Cancers: The Path to the Clinic
2019 · Savithri Ramurthy, Benjamin R. Taft, et al. · Journal of Medicinal Chemistry · 42
A Functionally Orthogonal Ligand−Receptor Pair Created by Targeting the Allosteric Mechanism of the Thyroid Hormone Receptor
2006 · A. Quamrul Hassan, John T. Koh · Journal of the American Chemical Society · 31
Allosteric inhibition of BCR-ABL
2010 · A. Quamrul Hassan, Sreenath V. Sharma, et al. · Cell Cycle · 29
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Functional Analysis of the Streptomyces coelicolor NrdR ATP-Cone Domain: Role in Nucleotide Binding, Oligomerization, and DNA Interactions
2008 · Inna Grinberg, Tatyana Shteinberg, et al. · Journal of Bacteriology · 25
Selective Chemical Rescue of a Thyroid‐Hormone‐Receptor Mutant, TRβ(H435Y), Identified in Pituitary Carcinoma and Resistance to Thyroid Hormone
2008 · A. Quamrul Hassan, John T. Koh · Angewandte Chemie International Edition · 20
Methodology To Probe Subunit Interactions in Ribonucleotide Reductases
2008 · A. Quamrul Hassan, Yongting Wang, et al. · Biochemistry · 18
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Site-Specific Incorporation of Chemical Probes into Proteins for NMR
2008 · A Quamrul Hassan · ACS Chemical Biology · 5
Mapping the subunit interface of ribonucleotide reductase (RNR) using photo cross-linking
2008 · A. Quamrul Hassan, JoAnne Stubbe · Bioorganic & Medicinal Chemistry Letters · 5
A novel allosteric means of inhibiting heat shock 70 proteins
2014 · Heather Sadlish, Asm Quamrul Hassan, et al.
Selective Chemical Rescue of a Thyroid‐Hormone‐Receptor Mutant, TRβ(H435Y), Identified in Pituitary Carcinoma and Resistance to Thyroid Hormone
2008 · A. Quamrul Hassan, John T. Koh · Angewandte Chemie
Works count: 15
Citation count: 1,455
H-index: 10
I10-index: 10
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