Author

Ashok V. Purandare

Observed names: A V Purandare, A. PURANDARE, A. Purandare, A. V. PURANDARE, A.V. Purandare, Ashok Purandare, Ashok V Purandare, Ashok V. Purandare

Institution: Bristol-Myers Squibb (United States)

Observed institutions: Rutgers, The State University of New Jersey, Bristol-Myers Squibb (United States)

OpenAlex ID: A5078878020

Structural basis for CARM1 inhibition by indole and pyrazole inhibitors

2011 · John S. Sack, Sandrine Thieffine, et al. · Biochemical Journal · 102

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Sensitivity of Small Cell Lung Cancer to BET Inhibition Is Mediated by Regulation of ASCL1 Gene Expression

2015 · Ryan Lenhart, Stefan Kirov, et al. · Molecular Cancer Therapeutics · 95

Pyrazole inhibitors of coactivator associated arginine methyltransferase 1 (CARM1)

2008 · Ashok V. Purandare, Zhong Chen, et al. · Bioorganic & Medicinal Chemistry Letters · 92

Optimization of pyrazole inhibitors of Coactivator Associated Arginine Methyltransferase 1 (CARM1)

2009 · Tram Huynh, Zhong Chen, et al. · Bioorganic & Medicinal Chemistry Letters · 83

Characterization of BMS-911543, a functionally selective small-molecule inhibitor of JAK2

2011 · A V Purandare, T M McDevitt, et al. · Leukemia · 77

Benzo[d]imidazole inhibitors of Coactivator Associated Arginine Methyltransferase 1 (CARM1)—Hit to Lead studies

2009 · Honghe Wan, Tram Huynh, et al. · Bioorganic & Medicinal Chemistry Letters · 62

Synthesis of chiral α- substituted β-hydroxy acid derivatives on solid support

1997 · Ashok V Purandare, Sesha Natarajan · Tetrahedron Letters · 59

Identification of chemokine receptor CCR4 antagonist

2005 · Ashok V. Purandare, Aiming Gao, et al. · Bioorganic & Medicinal Chemistry Letters · 58

A (1.fwdarw.4)-"trehazoloid" glucosidase inhibitor with aglycon selectivity

1994 · Spencer Knapp, Ashok Purandare, et al. · Journal of the American Chemical Society · 55

Inhibition of Casein Kinase 2 Disrupts Differentiation of Myeloid Cells in Cancer and Enhances the Efficacy of Immunotherapy in Mice

2018 · Ayumi Hashimoto, Chan Gao, et al. · Cancer Research · 48

Core exploration in optimization of chemokine receptor CCR4 antagonists

2006 · Ashok V. Purandare, Honghe Wan, et al. · Bioorganic & Medicinal Chemistry Letters · 44

Antagonists of CCR4 as Immunomodulatory Agents

2006 · Ashok Purandare, John Somerville · Current Topics in Medicinal Chemistry · 42

Molecular Recognition and Reactivity of Ruthenium(II) Bipyridine Barbituric Acid Guests in the Presence of Complementary Hosts: Ruthenium(II) Promoted Enolization of Barbituric Acids in Guest−Host Complexes

1997 · Teen Chin, Zhinong Gao, et al. · Journal of the American Chemical Society · 41

Discovery of a Highly Selective JAK2 Inhibitor, BMS-911543, for the Treatment of Myeloproliferative Neoplasms

2015 · Honghe Wan, Gretchen M. Schroeder, et al. · ACS Medicinal Chemistry Letters · 40

Aminotriazine 5-HT7 antagonists

2004 · Ronald J Mattson, Derek J Denhart, et al. · Bioorganic & Medicinal Chemistry Letters · 37

Kinase drug discovery approaches in chronic myeloproliferative disorders

2009 · C Kumar, A V Purandare, et al. · Oncogene · 32

Solid-phase synthesis of ‘diverse’ heterocycles

2002 · Ashok V. Purandare, Aiming Gao, et al. · Tetrahedron Letters · 22

Improved conditions for converting sterically hindered amides to 1,5-disubstituted tetrazoles

2010 · Gretchen M. Schroeder, Sydney Marshall, et al. · Tetrahedron Letters · 21

Optimization of CCR4 antagonists: Side-chain exploration

2005 · Ashok V. Purandare, Honghe Wan, et al. · Bioorganic & Medicinal Chemistry Letters · 19

Identification of a potent and rapidly reversible inhibitor of the 20S-proteasome

2004 · Ashok V. Purandare, Honghe Wan, et al. · Bioorganic & Medicinal Chemistry Letters · 17

Solid phase synthesis of unsymmetrical secondary amines—Application to the synthesis of arylethanolamines and arylpropanolamines

1998 · Ashok V Purandare, Michael A. Poss · Tetrahedron Letters · 17

Structure-Based Design of Selective Janus Kinase 2 Imidazo[4,5-d]pyrrolo[2,3-b]pyridine Inhibitors

2015 · Amy C. Hart, Gretchen M. Schroeder, et al. · ACS Medicinal Chemistry Letters · 16

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Pyrrolo[1,2-f]triazines as JAK2 inhibitors: Achieving potency and selectivity for JAK2 over JAK3

2011 · Lalgudi S. Harikrishnan, Muthoni G. Kamau, et al. · Bioorganic & Medicinal Chemistry Letters · 16

Diaminopyrimidine and diaminopyridine 5-HT7 ligands

2004 · Derek J Denhart, Ashok V Purandare, et al. · Bioorganic & Medicinal Chemistry Letters · 16

Preparation of 2,7-Diaminosubstituted-[1,2,4]triazolo[1,5-a]pyrimidine-6-Carbonitriles by Solid-Phase Synthesis

2007 · Cullen L. Cavallaro, Lalgudi S. Harikrishnan, et al. · Journal of Combinatorial Chemistry · 15

Works count: 65

Citation count: 1,179

H-index: 19

I10-index: 26