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Jacek Olczak
Observed names:
J Olczak,
J. Olczak,
Olczak, J.,
Olczak, Jacek
Institution:
Molecure SA (Poland)
Observed institutions:
Lodz University of Technology,
Washington University in St. Louis,
Medical University of Lodz,
OncoArendi Therapeutics (Poland),
Centrum Badań Molekularnych i Makromolekularnych Polskiej Akademii Nauk,
Molecure SA (Poland),
Polish Academy of Sciences
show all 7
ORCID:
0000-0001-9932-2373
Observed ORCID:
0000-0001-9932-2373
OpenAlex ID:
A5081028300
cis-peptide bond mimetic tetrazole analogs of the insect kinins identify the active conformation
2002
·
Ronald J Nachman
, Janusz Zabrocki
, et al.
·
Peptides
·
62
Chitinases and Chitinase-Like Proteins as Therapeutic Targets in Inflammatory Diseases, with a Special Focus on Inflammatory Bowel Diseases
2021
·
Marzena Mazur
, Anna Zielińska
, et al.
·
International Journal of Molecular Sciences
·
56
PDF
Synthesis of quaternary α-amino acid-based arginase inhibitors via the Ugi reaction
2013
·
Adam Golebiowski
, Darren Whitehouse
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
48
Discovery and Pharmacokinetics of Sulfamides and Guanidines as Potent Human Arginase 1 Inhibitors
2020
·
Roman Blaszczyk
, Joanna Brzezinska
, et al.
·
ACS Medicinal Chemistry Letters
·
46
Arginase 1/2 Inhibitor OATD-02: From Discovery to First-in-man Setup in Cancer Immunotherapy
2023
·
Bartlomiej Borek
, Julita Nowicka
, et al.
·
Molecular Cancer Therapeutics
·
44
PDF
OATD-02 Validates the Benefits of Pharmacological Inhibition of Arginase 1 and 2 in Cancer
2022
·
Marcin Mikołaj Grzybowski
, Paulina Seweryna Stańczak
, et al.
·
Cancers
·
44
PDF
Targeting Acidic Mammalian chitinase Is Effective in Animal Model of Asthma
2017
·
Marzena Mazur
, Jacek Olczak
, et al.
·
Journal of Medicinal Chemistry
·
35
Constrained Peptidomimetics for TRH: cis-Peptide Bond Analogs
2000
·
Yunsong Tong
, Jacek Olczak
, et al.
·
Tetrahedron
·
35
Discovery of OATD-01, a First-in-Class Chitinase Inhibitor as Potential New Therapeutics for Idiopathic Pulmonary Fibrosis
2020
·
Robert Koralewski
, Barbara Dymek
, et al.
·
Journal of Medicinal Chemistry
·
32
Development of Dual Chitinase Inhibitors as Potential New Treatment for Respiratory System Diseases
2019
·
Marzena Mazur
, Barbara Dymek
, et al.
·
Journal of Medicinal Chemistry
·
26
X-ray and Nuclear Magnetic Resonance (NMR) Studies of Signalizing the Tripeptide Sequence (Tyr-D-Ala-Phe) of Dermorphin and Deltorphins I and II. Comparative Analysis in the Liquid and Solid Phases
2004
·
Mikołaj M. Słabicki
, Marek J. Potrzebowski
, et al.
·
The Journal of Physical Chemistry B
·
24
Antarctic, cold-adapted β-galactosidase of Pseudoalteromonas sp. 22b as an effective tool for alkyl galactopyranosides synthesis
2008
·
K. Makowski
, A. Białkowska
, et al.
·
Enzyme and Microbial Technology
·
23
Structure-Based Discovery of High-Affinity Small Molecule Ligands and Development of Tool Probes to Study the Role of Chitinase-3-Like Protein 1
2024
·
Wojciech Czestkowski
, Łukasz Krzemiński
, et al.
·
Journal of Medicinal Chemistry
·
22
Specific interactions of bovine and human β-casomorphin-7 with Cu(II) ions
1998
·
Elżbieta Chruścińska
, Jacek Olczak
, et al.
·
Journal of Inorganic Biochemistry
·
16
Antinociceptive and antidepressant-like action of endomorphin-2 analogs with proline surrogates in position 2
2014
·
Renata Perlikowska
, Justyna Piekielna
, et al.
·
Bioorganic & Medicinal Chemistry
·
15
Novel glycosylated endomorphin-2 analog produces potent centrally-mediated antinociception in mice after peripheral administration
2013
·
Jakub Fichna
, Marzena Mazur
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
15
Impact of 1,5-disubstituted tetrazole ring on chelating ability of δ-selective opioid peptide
2003
·
Elżbieta Łodyga-Chruścińska
, Stanisław Ołdziej
, et al.
·
Journal of Inorganic Biochemistry
·
14
Novel orally bioavailable piperidine derivatives as extracellular arginase inhibitors developed by a ring expansion
2023
·
Anna Gzik
, Bartlomiej Borek
, et al.
·
European Journal of Medicinal Chemistry
·
13
Benzoxazepine-Derived Selective, Orally Bioavailable Inhibitor of Human Acidic Mammalian Chitinase
2020
·
Gleb Andryianau
, Michal Kowalski
, et al.
·
ACS Medicinal Chemistry Letters
·
13
Discovery of selective, orally bioavailable inhibitor of mouse chitotriosidase
2017
·
Marzena Mazur
, Agnieszka Bartoszewicz
, et al.
·
Bioorganic & Medicinal Chemistry Letters
·
13
Cyclic side-chain-linked opioid analogs utilizing cis- and trans-4-aminocyclohexyl-d-alanine
2014
·
Justyna Piekielna
, Luca Gentilucci
, et al.
·
Bioorganic & Medicinal Chemistry
·
12
Can the 1,5-disubstituted tetrazole ring modify the co-ordinating ability and biological activity of opiate-like peptides?
2000
·
Elzbieta Lodyga-Chruscinska
, Ewa Brzezinska-Blaszczyk
, et al.
·
Journal of Inorganic Biochemistry
·
12
Binding ability of Cu2+ ions by opiate-like fragments of bovine casein
1997
·
Elz̊bieta Chruścińska
, Marcin Dyba
, et al.
·
Journal of Inorganic Biochemistry
·
12
The Anti-Inflammatory Effect of Acidic Mammalian Chitinase Inhibitor OAT-177 in DSS-Induced Mouse Model of Colitis
2022
·
Marzena Mazur
, Jakub Włodarczyk
, et al.
·
International Journal of Molecular Sciences
·
10
PDF
Effect of the tetrazole cis-amide bond surrogate on the complexing ability of some enkephalin analogues toward Cu(II) ions
1999
·
Elzbieta Lodyga-Chruscinska
, Giovanni Micera
, et al.
·
Journal of Inorganic Biochemistry
·
10
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Works count:
100
Citation count:
705
H-index:
15
I10-index:
25
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