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Thomas P. Blackburn

Observed names: Blackburn, T., Blackburn, T.P., Blackburn, Thomas P, T BLACKBURN, T P Blackburn, T P. Blackburn, T. Blackburn, T. P. BLACKBURN, T. P. Blackburn, T.P BLACKBURN, T.P. BLACKBURN, T.P. Blackburn, Thomas Blackburn, Thomas P Blackburn
Observed institutions: AstraZeneca (United Kingdom), St Thomas' Hospital, University of Dundee, Pfizer (United States), GlaxoSmithKline (United Kingdom), Ninewells Hospital, Karolinska Institutet, Lundbeck (United States), Umecrine Cognition AB (Sweden)
ORCID: 0000-0001-9317-7507
Observed ORCID: 0000-0001-9317-7507
OpenAlex ID: A5083104098
SB 242084, a Selective and Brain Penetrant 5-HT 2C Receptor Antagonist
1997 · G.A. KENNETT, M.D. WOOD, et al. · Neuropharmacology · 523
Antidepressant, anxiolytic and anorectic effects of a melanin-concentrating hormone-1 receptor antagonist
2002 · Beth Borowsky, Margaret M. Durkin, et al. · Nature Medicine · 506
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Immunohistochemical localisation of the 5-HT2C receptor protein in the rat CNS
2000 · Delyth A Clemett, Taniya Punhani, et al. · Neuropharmacology · 373
In vitroandin vivoprofile of SB 206553, a potent 5‐HT2C/5‐HT2Breceptor antagonist with anxiolytic‐like properties
1996 · G.A. Kennett, M.D. Wood, et al. · British Journal of Pharmacology · 240
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The medical benefit of 5-HT research
2002 · Brian J Jones, Thomas P Blackburn · Pharmacology Biochemistry and Behavior · 227
Erratum: Antidepressant, anxiolytic and anorectic effects of a melanin-concentrating hormone-1 receptor antagonist
2002 · B. Borowsky, M.M. Durkin, et al. · Nature Medicine · 192
Anxiolytic- and antidepressant-like profiles of the galanin-3 receptor (Gal 3 ) antagonists SNAP 37889 and SNAP 398299
2005 · Chad J. Swanson, Thomas P. Blackburn, et al. · Proceedings of the National Academy of Sciences · 181
In vivoproperties of SB 200646A, a 5‐HT2C/2Breceptor antagonist
1994 · G.A. Kennett, M.D. Wood, et al. · British Journal of Pharmacology · 181
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Trace amine receptors as targets for novel therapeutics: legend, myth and fact
2003 · T BRANCHEK, T BLACKBURN · Current Opinion in Pharmacology · 163
Depressive disorders: Treatment failures and poor prognosis over the last 50 years
2019 · Thomas P. Blackburn · Pharmacology Research & Perspectives · 136
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Activation of 5-HT 2B Receptors in the Medial Amygdala causes Anxiolysis in the Social Interaction Test in the Rat
1997 · M.S DUXON, G.A KENNETT, et al. · Neuropharmacology · 103
Further characterization of 5‐hydroxytryptamine receptors (putative 5‐HT2B) in rat stomach fundus longitudinal muscle
1994 · Gordon S. Baxter, Olive E. Murphy, et al. · British Journal of Pharmacology · 100
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5-ht6 Receptors as Emerging Targets for Drug Discovery
2000 · Theresa A. Branchek, Thomas P. Blackburn · The Annual Review of Pharmacology and Toxicology · 95
6-Chloro-5-methyl-1-[[2-[(2-methyl-3- pyridyl)oxy]-5-pyridyl]carbamoyl]indoline (SB-242084): The First Selective and Brain Penetrant 5-HT2C Receptor Antagonist
1997 · Steven M. Bromidge, Malcolm Duckworth, et al. · Journal of Medicinal Chemistry · 83
Anxiolytic-like effect of paroxetine in a rat social interaction test
1994 · S. Lightowler, G.A. Kennett, et al. · Pharmacology Biochemistry and Behavior · 83
Biarylcarbamoylindolines Are Novel and Selective 5-HT2C Receptor Inverse Agonists: Identification of 5-Methyl-1-[[2-[(2-methyl-3-pyridyl)oxy]- 5-pyridyl]carbamoyl]-6-trifluoromethylindoline (SB-243213) as a Potential Antidepressant/Anxiolytic Agent
2000 · Steven M. Bromidge, Steven Dabbs, et al. · Journal of Medicinal Chemistry · 79
Evidence that 5-HT2C receptor antagonists are anxiolytic in the rat Geller-Seifter model of anxiety
1994 · G. A. Kennett, K. Pittaway, et al. · Psychopharmacology · 74
Effect of SB 200646A, a 5-HT2C/5-HT2B receptor antagonist, in two conflict models of anxiety
1995 · G. A. Kennett, F. Bailey, et al. · Psychopharmacology · 72
BRL 46470A: a highly potent, selective and long acting 5-HT3 receptor antagonist with anxiolytic-like properties
1993 · T. P. Blackburn, G. S. Baxter, et al. · Psychopharmacology · 70
Novel and Selective 5-HT2C/2B Receptor Antagonists as Potential Anxiolytic Agents: Synthesis, Quantitative Structure−Activity Relationships, and Molecular Modeling of Substituted 1-(3-Pyridylcarbamoyl)indolines
1998 · Steven M. Bromidge, Steven Dabbs, et al. · Journal of Medicinal Chemistry · 64
Anxiolytic-like Actions of the Selective 5-HT 4 Receptor Antagonists SB 204070A and SB 207266A in Rats
1997 · G.A KENNETT, F BRIGHT, et al. · Neuropharmacology · 62
5-Methyl-1-(3-pyridylcarbamoyl)-1,2,3,5-tetrahydropyrrolo[2,3-f]indole: A Novel 5-HT2C/5-HT2B Receptor Antagonist with Improved Affinity, Selectivity, and Oral Activity
1995 · Ian T. Forbes, Peter Ham, et al. · Journal of Medicinal Chemistry · 61
In vitro studies with ICI 169,369, a chemically novel 5-HT antagonist
1988 · Thomas P. Blackburn, Craig W. Thornber, et al. · European Journal of Pharmacology · 54
Pharmacological characterization of the apparent splice variants of the murine 5-HT3 R-A subunit expressed in Xenopus laevis oocytes
1994 · D.L. Downie, A.G. Hope, et al. · Neuropharmacology · 51
BRL 46470 potently antagonizes neural responses activated by 5-HT3 receptors
1993 · N NEWBERRY, C WATKINS, et al. · Neuropharmacology · 50
Works count: 94
Citation count: 4,730
H-index: 33
I10-index: 56
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