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Mateusz Daśko

Observed names: Daśko, Mateusz, Mateusz Dasko
ORCID: 0000-0002-3367-6491
Observed ORCID: 0000-0002-3367-6491
OpenAlex ID: A5083666138
Selected organophosphorus compounds with biological activity. Applications in medicine
2016 · Sebastian Demkowicz, Janusz Rachon, et al. · RSC Advances · 288
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Novel 1,2,4-Oxadiazole Derivatives in Drug Discovery
2020 · Karol Biernacki, Mateusz Daśko, et al. · Pharmaceuticals · 198
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HDAC Inhibitors: Innovative Strategies for Their Design and Applications
2022 · Mateusz Daśko, Beatriz de Pascual-Teresa, et al. · Molecules · 85
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Synthesis and biological evaluation of fluorinated N -benzoyl and N -phenylacetoyl derivatives of 3-(4-aminophenyl)-coumarin-7- O -sulfamate as steroid sulfatase inhibitors
2017 · Mateusz Daśko, Maja Przybyłowska, et al. · European Journal of Medicinal Chemistry · 26
Selected Methods for the Chemical Phosphorylation and Thiophosphorylation of Phenols
2017 · Witold Kozak, Janusz Rachon, et al. · Asian Journal of Organic Chemistry · 23
Recent progress in the development of steroid sulphatase inhibitors – examples of the novel and most promising compounds from the last decade
2020 · Mateusz Daśko, Sebastian Demkowicz, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 22
Steroid Sulfatase Inhibitors Based on Phosphate and Thiophosphate Flavone Analogs
2015 · Witold Kozak, Mateusz Daśko, et al. · Drug Development Research · 21
Phosphate tricyclic coumarin analogs as steroid sulfatase inhibitors: synthesis and biological activity
2014 · Witold Kozak, Mateusz Daśko, et al. · RSC Advances · 21
Synthesis and Biological Evaluation of Fluorinated 3‐Phenylcoumarin‐7‐O‐Sulfamate Derivatives as Steroid Sulfatase Inhibitors
2015 · Sebastian Demkowicz, Mateusz Daśko, et al. · Chemical Biology & Drug Design · 20
Evaluation of Tyrosinase Inhibitory Activity of Carbathioamidopyrazoles and Their Potential Application in Cosmetic Products and Melanoma Treatment
2025 · Ewelina Namiecińska, Jan Jaszczak, et al. · International Journal of Molecular Sciences · 19
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Design, synthesis and biological evaluation of novel N -phosphorylated and O -phosphorylated tacrine derivatives as potential drugs against Alzheimer’s disease
2022 · Maja Przybyłowska, Krystyna Dzierzbicka, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 19
Development of Sulfamoylated 4-(1-Phenyl-1H-1,2,3-triazol-4-yl)phenol Derivatives as Potent Steroid Sulfatase Inhibitors for Efficient Treatment of Breast Cancer
2022 · Karol Biernacki, Olga Ciupak, et al. · Journal of Medicinal Chemistry · 18
Synthesis of bicoumarin thiophosphate derivatives as steroid sulfatase inhibitors
2015 · Sebastian Demkowicz, Witold Kozak, et al. · European Journal of Medicinal Chemistry · 18
Thermodynamic Studies of Interactions between Sertraline Hydrochloride and Randomly Methylated β-Cyclodextrin Molecules Supported by Circular Dichroism Spectroscopy and Molecular Docking Results
2021 · Sylwia Belica-Pacha, Mateusz Daśko, et al. · International Journal of Molecular Sciences · 17
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Modifications at the C(5) position of pyrimidine nucleosides
2019 · Witold Kozak, Sebastian Demkowicz, et al. · Russian Chemical Reviews · 16
Geometry optimization of steroid sulfatase inhibitors - the influence on the free binding energy with STS
2017 · Karolina Jagiello, Anita Sosnowska, et al. · Structural Chemistry · 12
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Synthesis and biological evaluation of N‐acylated tyramine sulfamates containing C–F bonds as steroid sulfatase inhibitors
2016 · Mateusz Daśko, Janusz Rachon, et al. · Chemical Biology & Drug Design · 11
Synthesis and biological evaluation of thiophosphate tricyclic coumarin derivatives as steroid sulfatase inhibitors
2015 · Witold Kozak, Mateusz Daśko, et al. · Journal of Asian Natural Products Research · 11
Development of potent and effective SARS-CoV-2 main protease inhibitors based on maleimide analogs for the potential treatment of COVID-19
2023 · Karol Biernacki, Olga Ciupak, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 10
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Novel steroid sulfatase inhibitors based on N‐thiophosphorylated 3‐(4‐aminophenyl)‐coumarin‐7‐O‐sulfamates
2019 · Mateusz Daśko, Sebastian Demkowicz, et al. · Drug Development Research · 10
Novel 1,2,3-Triazole Derivatives as Mimics of Steroidal System—Synthesis, Crystal Structures Determination, Hirshfeld Surfaces Analysis and Molecular Docking
2021 · Mateusz Daśko, Anna Dołęga, et al. · Molecules · 9
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Synthesis and steroid sulfatase inhibitory activities of N-alkanoyl tyramine phosphates and thiophosphates
2015 · Witold Kozak, Mateusz Daśko, et al. · RSC Advances · 9
Novel amides of mycophenolic acid and some heterocyclic derivatives as immunosuppressive agents
2022 · Juliusz Maksymilian Walczak, Dorota Iwaszkiewicz-Grześ, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 8
New potent steroid sulphatase inhibitors based on 6-(1-phenyl-1H-1,2,3-triazol-4-yl)naphthalen-2-yl sulphamate derivatives
2020 · Olga Ciupak, Mateusz Daśko, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 8
New potent STS inhibitors based on fluorinated 4-(1-phenyl-1H-[1,2,3]triazol-4-yl)-phenyl sulfamates
2019 · Mateusz Daśko, Sebastian Demkowicz, et al. · Journal of Asian Natural Products Research · 8
Works count: 66
Citation count: 948
H-index: 15
I10-index: 20
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