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Ramasastri Kambhampati

Observed institution: Suven Life Sciences (India)
OpenAlex ID: A5086179959
Synthesis and structure–activity relationship of novel conformationally restricted analogues of serotonin as 5-HT6receptor ligands
2011 · Ramakrishna V.S. Nirogi, Ramasastri Kambhampati, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 25
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Indole-3-piperazinyl derivatives: Novel chemical class of 5-HT6 receptor antagonists
2010 · Ramakrishna V.S. Nirogi, Amol D. Deshpande, et al. · Bioorganic & Medicinal Chemistry Letters · 25
Design, Synthesis, and Pharmacological Evaluation of Piperidin-4-yl amino aryl sulfonamides: Novel, Potent, Selective, Orally Active, and Brain Penetrant 5-HT6Receptor Antagonists
2012 · Ramakrishna Nirogi, Anil Shinde, et al. · Journal of Medicinal Chemistry · 16
Design, synthesis and pharmacological evaluation of 4-(piperazin-1-yl methyl)-N1-arylsulfonyl indole derivatives as 5-HT6 receptor ligands
2012 · Ramakrishna V.S. Nirogi, Rajeshkumar Badange, et al. · Bioorganic & Medicinal Chemistry Letters · 10
Design, synthesis and pharmacological evaluation of conformationally restricted N-arylsulfonyl-3-aminoalkoxy indoles as a potential 5-HT6receptor ligands
2011 · Ramakrishna V.S. Nirogia, Ramasastri Kambhampati, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 10
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Novel and Potent 5-Piperazinyl Methyl-N1-aryl Sulfonyl Indole Derivatives as 5-HT6 Receptor Ligands
2010 · Ramakrishna V. S. Nirogi, Prabhakar Kothmirkar, et al. · ACS Medicinal Chemistry Letters · 7
P3‐451: SUVN‐502: A potent and selective 5‐HT6 antagonist, potential drug for the treatment of Alzheimer's disease
2011 · Ramakrishna Nirogi, Vishwottam Kandikere, et al. · Alzheimer s & Dementia · 3
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P1‐251: SUVN‐502: A safe, potent, selective, brain penetrant and orally active 5‐HT6 receptor antagonist ‐ first in human clinical phase‐1 study
2009 · Ramakrishna Nirogi, Ramasastri Kambhampati, et al. · Alzheimer s & Dementia · 3
Design, synthesis and preliminary screening of novel 3-(2-N,N-dimethylaminoethylthio) indole derivatives as potential 5-HT6 receptor ligands
2008 · Ramasastri Kambhampati, Jagadishbabu Konda, et al. · Journal of Enzyme Inhibition and Medicinal Chemistry · 3
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Synthesis of Novel Rigid Analogs of Tryptamine as Potential Serotonin Ligands through Pd(0)-Catalyzed Diaryl Coupling Reactions
2008 · Ramasastri Kambhampati, Prabhakar Kothmirkar, et al. · Synthetic Communications · 2
P3‐390: Effect of Gender and Food on the Single‐dose Pharmacokinetics of Suvn‐502, a Potent and Selective 5‐ht6 Receptor Antagonist
2014 · Ramakrishna Nirogi, Koteshwara Mudigonda, et al. · Alzheimer s & Dementia
P4‐235: Pro‐cognitive properties of SUVN‐G1010034, a potent selective H3 antagonist in animal models of cognition
2012 · Ramakrishna Nirogi, Vishwottam Kandikere, et al. · Alzheimer s & Dementia
P1‐263: Pro‐cognitive properties SUVN‐D1108121, a potent and selective 5‐HT4 receptor partial agonist
2012 · Ramakrishna Nirogi, Renny Abraham, et al. · Alzheimer s & Dementia
Synthesis and biological screening of 2-(4-methylpiperazin-1-yl methyl)-1-(arylsulfonyl)-1H-indole derivatives as 5-HT6 receptor ligands: Part II
2012 · Ramakrishna Nirogi, Amol D. Deshp, et al. · Der pharma chemica
Design, synthesis and biological screening of N1-arylsulfonyl (1H-indole-2-yl)-1-(piperazinyl) methanone derivatives as 5-HT6 receptor ligands: Part I
2012 · Ramakrishna Nirogi, Amol D. Deshp, et al. · Der pharma chemica
Synthesis and biological screening of 3-chloro-2-piperazinylmethyl-N-aryl sulfonamide indole derivatives as 5-HT6 receptor ligands: Part III
2012 · Ramakrishna Nirogi, Amol D. Deshp, et al. · Der pharma chemica
Design, synthesis and biological activity of novel substituted 2-Aryl sulfonyl methyl tryptamines as potential 5-HT6 Receptor ligands
2012 · Ramakrishna Nirogi, Thrinath Reddy B, et al. · Der pharma chemica
IC‐P‐107: SUVN‐90716: A Selective 5‐HT6 Antagonist for the Potential Treatment of Alzheimer's Disease
2010 · Ramakrishna Nirogi, Vishwottam Kandikere, et al. · Alzheimer s & Dementia
ChemInform Abstract: Synthesis of Novel Rigid Analogues of Tryptamine as Potential Serotonin Ligands Through Pd(0)‐Catalyzed Diaryl Coupling Reactions.
2008 · Ramasastri Kambhampati, Prabhakar Kothmirkar, et al. · ChemInform
P4‐325: A potent selective brain penetrant and orally active 5‐HT6 receptor antagonist SUVN‐502 for the symptomatic treatment of Alzheimer's disease
2008 · Ramakrishna Nirogi, Pradeep Jayarajan, et al. · Alzheimer s & Dementia
Works count: 20
Citation count: 104
H-index: 6
I10-index: 5
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