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Simona Rizzi
Institution:
Nerviano Medical Sciences
Observed institutions:
Istituto Ortopedico Rizzoli,
Nerviano Medical Sciences
ORCID:
0000-0002-1515-2096
Observed ORCID:
0000-0002-1515-2096
OpenAlex ID:
A5087080299
Covalent and allosteric inhibitors of the ATPase VCP/p97 induce cancer cell death
2013
·
Paola Magnaghi
, Roberto D'Alessio
, et al.
·
Nature Chemical Biology
·
383
NMS-P937, an Orally Available, Specific Small-Molecule Polo-like Kinase 1 Inhibitor with Antitumor Activity in Solid and Hematologic Malignancies
2012
·
Barbara Valsasina
, Italo Beria
, et al.
·
Molecular Cancer Therapeutics
·
128
Alkylsulfanyl-1,2,4-triazoles, a New Class of Allosteric Valosine Containing Protein Inhibitors. Synthesis and Structure–Activity Relationships
2012
·
Paolo Polucci
, Paola Magnaghi
, et al.
·
Journal of Medicinal Chemistry
·
95
Redundancy of autocrine loops in human osteosarcoma cells
1999
·
Stefania Benini
, Nicola Baldini
, et al.
·
International Journal of Cancer
·
88
PDF
An antibody-drug conjugate directed to the ALK receptor demonstrates efficacy in preclinical models of neuroblastoma
2019
·
Renata Sano
, Kateryna Krytska
, et al.
·
Science Translational Medicine
·
70
PDF
Phosphorylation of TCTP as a marker for polo-like kinase-1 activity in vivo.
2010
·
Ulisse Cucchi
, Laura M Gianellini
, et al.
·
PubMed
·
60
Discovery of 2-(Cyclohexylmethylamino)pyrimidines as a New Class of Reversible Valosine Containing Protein Inhibitors
2014
·
Giovanni Cervi
, Paola Magnaghi
, et al.
·
Journal of Medicinal Chemistry
·
22
Novel Thienoduocarmycin–Trastuzumab ADC Demonstrates Strong Antitumor Efficacy with Favorable Safety Profile in Preclinical Studies
2023
·
Barbara Valsasina
, Paolo Orsini
, et al.
·
Molecular Cancer Therapeutics
·
6
Abstract 734: Thienoindoles: New highly promising agents for antibody-drug conjugates generation
2018
·
Michele Caruso
, Fabio Gasparri
, et al.
·
Cancer Research
·
4
Abstract 822: Thienoindoles, a novel class of DNA minor groove alkylating agents highly suited for the generation of novel antibody drug conjugates (ADCs)
2014
·
Barbara Valsasina
, Fabio Gasparri
, et al.
·
Cancer Research
·
2
Abstract 5805: A novel platform of diversified payloads to drive ADC innovation
2024
·
Paolo Orsini
, Matteo Salsa
, et al.
·
Cancer Research
·
1
Abstract 5163: Characterization of NMS-E194, a selective and potent PERK inhibitor with efficacy in the KMS-11 multiple myeloma
2017
·
Claudia Perrera
, Maurizio Pulici
, et al.
·
Cancer Research
·
1
Abstract 2690: A novel antibody-drug conjugate directed to the ALK receptor tyrosine kinase demonstrates efficacy in models of neuroblastoma
2016
·
Renata Sano
, Kateryna Krytska
, et al.
·
Cancer Research
·
1
Abstract 2940: Identification of potent VCP/p97/CDC48 inhibitors with distinct biochemical mechanisms including a reversible, allosteric inhibitor that activates the unfolded protein response, induce autophagy and cancer cell death
2012
·
Paola Magnaghi
, Roberto D'Alessio
, et al.
·
Cancer Research
·
1
Table S5 from Novel Thienoduocarmycin–Trastuzumab ADC Demonstrates Strong Antitumor Efficacy with Favorable Safety Profile in Preclinical Studies
2023
·
Barbara Valsasina
, Paolo Orsini
, et al.
Table S6 from Novel Thienoduocarmycin–Trastuzumab ADC Demonstrates Strong Antitumor Efficacy with Favorable Safety Profile in Preclinical Studies
2023
·
Barbara Valsasina
, Paolo Orsini
, et al.
Data from Novel Thienoduocarmycin–Trastuzumab ADC Demonstrates Strong Antitumor Efficacy with Favorable Safety Profile in Preclinical Studies
2023
·
Barbara Valsasina
, Paolo Orsini
, et al.
Figure S2 from Novel Thienoduocarmycin–Trastuzumab ADC Demonstrates Strong Antitumor Efficacy with Favorable Safety Profile in Preclinical Studies
2023
·
Barbara Valsasina
, Paolo Orsini
, et al.
Figure S3 from Novel Thienoduocarmycin–Trastuzumab ADC Demonstrates Strong Antitumor Efficacy with Favorable Safety Profile in Preclinical Studies
2023
·
Barbara Valsasina
, Paolo Orsini
, et al.
Table S2 from Novel Thienoduocarmycin–Trastuzumab ADC Demonstrates Strong Antitumor Efficacy with Favorable Safety Profile in Preclinical Studies
2023
·
Barbara Valsasina
, Paolo Orsini
, et al.
Table S3 from Novel Thienoduocarmycin–Trastuzumab ADC Demonstrates Strong Antitumor Efficacy with Favorable Safety Profile in Preclinical Studies
2023
·
Barbara Valsasina
, Paolo Orsini
, et al.
Table S2 from Novel Thienoduocarmycin–Trastuzumab ADC Demonstrates Strong Antitumor Efficacy with Favorable Safety Profile in Preclinical Studies
2023
·
Barbara Valsasina
, Paolo Orsini
, et al.
Table S1 from Novel Thienoduocarmycin–Trastuzumab ADC Demonstrates Strong Antitumor Efficacy with Favorable Safety Profile in Preclinical Studies
2023
·
Barbara Valsasina
, Paolo Orsini
, et al.
Table S4 from Novel Thienoduocarmycin–Trastuzumab ADC Demonstrates Strong Antitumor Efficacy with Favorable Safety Profile in Preclinical Studies
2023
·
Barbara Valsasina
, Paolo Orsini
, et al.
Data from Novel Thienoduocarmycin–Trastuzumab ADC Demonstrates Strong Antitumor Efficacy with Favorable Safety Profile in Preclinical Studies
2023
·
Barbara Valsasina
, Paolo Orsini
, et al.
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Works count:
36
Citation count:
862
H-index:
7
I10-index:
7
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