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Chahrazed Bouzriba

Stereoselective Synthesis of Fluorinated Galactopyranosides as Potential Molecular Probes for Galactophilic Proteins: Assessment of Monofluorogalactoside–LecA Interactions
2019 · Vincent Denavit, Danny Lainé, et al. · Chemistry - A European Journal · 46
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Phenyl 4-(2-oxopyrrolidin-1-yl)benzenesulfonates and phenyl 4-(2-oxopyrrolidin-1-yl)benzenesulfonamides as new antimicrotubule agents targeting the colchicine-binding site
2021 · Mathieu Gagné-Boulet, Chahrazed Bouzriba, et al. · European Journal of Medicinal Chemistry · 13
Branched alkyl of phenyl 4-(2-oxo-3-alkylimidazolidin-1-yl)benzenesulfonates as unique cytochrome P450 1A1-activated antimitotic prodrugs: Biological evaluation and mechanism of bioactivation
2021 · Chahrazed Bouzriba, Atziri Corin Chavez Alvarez, et al. · European Journal of Medicinal Chemistry · 11
4-(3-Alkyl-2-oxoimidazolidin-1-yl)-N-phenylbenzenesulfonamide salts: Novel hydrosoluble prodrugs of antimitotics selectively bioactivated by the cytochrome P450 1A1 in breast cancer cells
2023 · Vincent Ouellette, Atziri Corin Chavez Alvarez, et al. · Bioorganic Chemistry · 9
Rationale, synthesis and biological evaluation of substituted 1-(4-(phenylthio)phenyl)imidazolidin-2-one, urea, thiourea and amide analogs and derivatives designed to target the colchicine-binding site
2022 · Mathieu Gagné-Boulet, Chahrazed Bouzriba, et al. · Journal of Molecular Structure · 9
Homologation of the Alkyl Side Chain of Antimitotic Phenyl 4-(2-Oxo-3-alkylimidazolidin-1-yl)benzenesulfonate Prodrugs Selectively Targeting CYP1A1-Expressing Breast Cancers Improves Their Stability in Rodent Liver Microsomes
2023 · Atziri Corin Chavez Alvarez, Chahrazed Bouzriba, et al. · Journal of Medicinal Chemistry · 8
Preparation, characterisation and biological evaluation of new N-phenyl amidobenzenesulfonates and N-phenyl ureidobenzenesulfonates inducing DNA double-strand breaks. Part 3. Modulation of ring A
2018 · Mathieu Gagné-Boulet, Chahrazed Bouzriba, et al. · European Journal of Medicinal Chemistry · 7
N-phenyl ureidobenzenesulfonates, a novel class of promising human dihydroorotate dehydrogenase inhibitors
2020 · Chahrazed Bouzriba, Lauriane Larcher, et al. · Bioorganic & Medicinal Chemistry · 4
Diversity‐Oriented Synthesis of Diol‐Based Peptidomimetics as Potential HIV Protease Inhibitors and Antitumor Agents
2018 · Paresh M. Vadhadiya, Marc‐Alexandre Jean, et al. · ChemBioChem · 4
Design, synthesis and biological evaluation of N -pyridinyl ureidobenzenesulfonates and their hydrochloride salts as novel water-soluble dihydroorotate dehydrogenase inhibitors inducing differentiation of acute myeloid leukemia cells
2025 · Vincent Ouellette, Chahrazed Bouzriba, et al. · RSC Medicinal Chemistry · 3
Synthesis and anticancer properties of a hybrid molecule with the testosterone and estradiol head-groups
2024 · Alexis Paquin, Fayanne Nolin, et al. · Steroids · 3
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Modification of the phenyl ring B of phenyl 4-(2-oxoimidazolidin-1-yl)benzenesulfonates by pyridinyl moiety leads to novel antimitotics targeting the colchicine-binding site
2024 · Vincent Ouellette, Chahrazed Bouzriba, et al. · Bioorganic & Medicinal Chemistry Letters · 3
N-Phenyl ureidobenzenesulfonates, a novel class of human dihydroorotate dehydrogenase inhibitors inducing differentiation and apoptosis in acute myeloid leukemia cells
2024 · Chahrazed Bouzriba, Atziri Corin Chavez Alvarez, et al. · Biomedicine & Pharmacotherapy · 2
Preparation and biological evaluation of new antimicrotubule agents: Modification of the imidazolidin‐2‐one moiety of phenyl 4‐(2‐oxoimidazolidin‐1‐yl)benzenesulfonates
2021 · Mathieu Gagné‐Boulet, Chahrazed Bouzriba, et al. · Chemical Biology & Drug Design · 2
Toxicity, Half-Life and Antitumor Activity of Phenyl 4-(2-Oxo-3-alkylimidazolidin-1-yl)benzenesulfonates as Novel Antimitotic CYP1A1-Targeted Prodrugs in Female Mouse Models
2025 · Atziri Corin Chavez Alvarez, Chahrazed Bouzriba, et al. · Pharmaceutics · 1
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Development of an UHPLC-UV Method for Quantification of Three Phenyl 4-(2-oxo-3-alkylimidazolidin-1-yl)benzenesulfonates in CD-1® IGS Female Mouse Plasma
2024 · Atziri Corin Chavez Alvarez, Chahrazed Bouzriba, et al. · Journal of Analytical Chemistry · 1
Pyridinyl 4-(2-oxoalkylimidazolidin-1-yl)benzenesulfonates and their hydrochloride salts as novel water soluble antimitotic prodrugs bioactivated by cytochrome P450 1A1 in breast cancer cells
2024 · Vincent Ouellette, Chahrazed Bouzriba, et al. · RSC Medicinal Chemistry · 1
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Abstract 1359: Evaluation of the therapeutic potential of AIMZ-938 as a new cytochrome p450 1A1-selective prodrug for the treatment of breast cancers
2021 · Atziri Corin Chavez Alvarez, Chahrazed Bouzriba, et al. · Cancer Research · 1
Design, synthesis and biological evaluation of new 2,6-difluorinated phenyl 4-(2-oxoimidazolidin-1-yl)benzenesulfonates as new antimicrotubule agents
2024 · Chahrazed Bouzriba, Mathieu Gagné-Boulet, et al. · Bioorganic Chemistry
Abstract 286: Conception and preparation of new potent antimicrotubule agents
2021 · Mathieu Gagné-Boulet, Chahrazed Bouzriba, et al. · Cancer Research
Abstract 285: Development of phenyl 4-(2-oxo-3-alkylimidazolidin-1-yl)benzenesulfonates as new antimitotic cytochrome P450 1A1-activated prodrugs selective toward breast cancers: Evaluation of branched alkyl chains
2021 · Chahrazed Bouzriba, Atziri Corin Chavez Alvarez, et al. · Cancer Research
CCDC 1824899: Experimental Crystal Structure Determination
2019 · Denavit, Vincent, Lainé, Danny, et al. · The Cambridge Structural Database
CCDC 1547825: Experimental Crystal Structure Determination
2018 · Vadhadiya, Paresh M., Jean, Marc-Alexandre, et al. · The Cambridge Structural Database
Works count: 23
Citation count: 128
H-index: 7
I10-index: 3
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