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Arun Kumar Gupta

Synthesis of Cyclobutane-Fused Tetracyclic Scaffolds via Visible-Light Photocatalysis for Building Molecular Complexity
2020 · Martins S. Oderinde, Edna Mao, et al. · Journal of the American Chemical Society · 165
Utilization of C(sp3)‐Carboxylic Acids and Their Redox‐Active Esters in Decarboxylative Carbon−Carbon Bond Formation
2021 · Sukhen Karmakar, Arundutt Silamkoti, et al. · Advanced Synthesis & Catalysis · 146
1-(2-Iodophenyl)-1H-tetrazole as a ligand for Pd(II) catalyzed Heck reaction
2004 · Arun Kumar Gupta, Chung Hyun Song, et al. · Tetrahedron Letters · 114
Rhodium-catalyzed tandem cyclization–cycloaddition reactions of enynebenzaldehydes: construction of polycyclic ring systems
2005 · Seunghoon Shin, Arun Kumar Gupta, et al. · Chemical Communications · 96
Highly efficient [2 + 2] intramolecular cyclizations of allenynes under microwave irradiation: construction of fused bicyclic compounds
2005 · Chang Ho Oh, Arun Kumar Gupta, et al. · Chemical Communications · 67
Novel [6 + 2] Cycloaddition of Fulvenes with Alkenes: A Facile Synthesis of the Anislactone and Hirsutane Framework
2002 · Bor-Cherng Hong, Yeong-Jou Shr, et al. · Organic Letters · 65
Hetero [6+3] Cycloaddition of Fulvenes with N-Alkylidene Glycine Esters: A Facile Synthesis of the Delavayine and Incarvillateine Framework
2003 · Bor-Cherng Hong, Arun Kumar Gupta, et al. · Organic Letters · 50
Gold nanoparticle-catalysed [3 + 2]dipolar cycloaddition of 1,6-allenynebenzaldehydes: construction of polycyclic ring systems
2005 · Arun Kumar Gupta, Chul Yun Rhim, et al. · Green Chemistry · 42
Identification of bicyclic hexafluoroisopropyl alcohol sulfonamides as retinoic acid receptor-related orphan receptor gamma (RORγ/RORc) inverse agonists. Employing structure-based drug design to improve pregnane X receptor (PXR) selectivity
2017 · Hua Gong, David S. Weinstein, et al. · Bioorganic & Medicinal Chemistry Letters · 40
Regioselective Pd-catalyzed alkylative lactonizations of 4-hydroxy-2-alkynecarboxylates with organoboronic acids
2004 · Chang Ho Oh, Su Jin Park, et al. · Tetrahedron Letters · 40
Azadiene Diels−Alder Cycloaddition of Fulvenes: A Facile Approach to the [1]Pyrindine System
2004 · Bor-Cherng Hong, Jian-Lin Wu, et al. · Organic Letters · 38
Rationally Designed, Conformationally Constrained Inverse Agonists of RORγt—Identification of a Potent, Selective Series with Biologic-Like in Vivo Efficacy
2019 · David Marcoux, James J.-W. Duan, et al. · Journal of Medicinal Chemistry · 37
Chemodiversity in the Palladium-Catalyzed Cyclizations of Allenynecarboxylates
2005 · Chang Ho Oh, Dai In Park, et al. · Synlett · 33
Formal [6+3] cycloaddition of fulvenes with 2H-azirine: a facile approach to the [2]pyrindines system
2004 · Bor-Cherng Hong, Arun Kumar Gupta, et al. · Tetrahedron Letters · 30
Selective IKur Inhibitors for the Potential Treatment of Atrial Fibrillation: Optimization of the Phenyl Quinazoline Series Leading to Clinical Candidate 5-[5-Phenyl-4-(pyridin-2-ylmethylamino)quinazolin-2-yl]pyridine-3-sulfonamide
2017 · Prashantha Gunaga, John Lloyd, et al. · Journal of Medicinal Chemistry · 25
Unprecedented carbocyclization of 1,6-allenynes on addition of organoboronic acids under Pd-catalysis
2005 · Arun Kumar Gupta, Chul Yun Rhim, et al. · Tetrahedron Letters · 25
Structural models in the assessment of protein druggability based on HTS data
2009 · Anvita Gupta, Arun Kumar Gupta, et al. · Journal of Computer-Aided Molecular Design · 22
Tertiary-butoxycarbonyl (Boc) – A strategic group for N-protection/deprotection in the synthesis of various natural/unnatural N-unprotected aminoacid cyanomethyl esters
2018 · Ananta Karmakar, Mushkin Basha, et al. · Tetrahedron Letters · 18
Tricyclic-Carbocyclic RORγt Inverse Agonists—Discovery of BMS-986313
2021 · Michael G. Yang, Myra Beaudoin-Bertrand, et al. · Journal of Medicinal Chemistry · 16
The exclusive formation of cyclopentenones from molybdenum hexacarbonyl-catalyzed Pauson–Khand reactions of 5-allenyl-1-ynes
2005 · Arun Kumar Gupta, Dai In Park, et al. · Tetrahedron Letters · 15
Identification of potent, selective and orally bioavailable phenyl ((R)-3-phenylpyrrolidin-3-yl)sulfone analogues as RORγt inverse agonists
2019 · Zhonghui Lu, James J.-W. Duan, et al. · Bioorganic & Medicinal Chemistry Letters · 13
Development of a Scalable Synthesis for the Potent Kinase Inhibitor BMS-986236; 1-(5-(4-(3-Hydroxy-3-methylbutyl)-1H-1,2,3-triazol-1-yl)-4-(isopropylamino)pyridin-2-yl)-1H-pyrazolo[3,4-b]pyridine-5-carbonitrile
2019 · Pirama Nayagam Arunachalam, Prakasam Kuppusamy, et al. · Organic Process Research & Development · 11
Practical Synthesis of (3aR, 9bR)-8-Fluoro-7-(perfluoropropan-2-yl)-9b-(phenylsulfonyl)-2,3,3a,4,5,9b-hexahydro-1H-benzo[e]indole: An Advanced Intermediate to Access the RORγt Inverse Agonist BMT-362265
2021 · Ananta Karmakar, Roshan Y. Nimje, et al. · Organic Process Research & Development · 10
Discovery of (3S,4S)-3-methyl-3-(4-fluorophenyl)-4-(4-(1,1,1,3,3,3-hexafluoro-2-hydroxyprop-2-yl)phenyl)pyrrolidines as novel RORγt inverse agonists
2020 · Bin Jiang, James J.-W. Duan, et al. · Bioorganic & Medicinal Chemistry Letters · 10
Study of physicochemical properties-antitubercular activity relationship of naphthalene-1,4-dione analogs: A QSAR approach
2009 · Revathi Gupta, Arun Gupta, et al. · Chemical Papers · 10
Works count: 68
Citation count: 1,190
H-index: 18
I10-index: 25
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