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Kazuyuki Miyashita

Observed names: K. MIYASHITA, KAZUYUKI MIYASHITA, Kazuyuki MIYASHITA, Miyashita, K., Miyashita, Kazuyuki
ORCID: 0000-0002-1770-2733
Observed ORCID: 0000-0002-1770-2733
OpenAlex ID: A5102720443
Crystal Structure of 6α-(Hydroxymethyl)penicillanate Complexed to the TEM-1 β-Lactamase from Escherichia coli : Evidence on the Mechanism of Action of a Novel Inhibitor Designed by a Computer-Aided Process
1996 · Laurent Maveyraud, Irina Massova, et al. · Journal of the American Chemical Society · 122
Inhibition of the NMC-A β-Lactamase by a Penicillanic Acid Derivative and the Structural Bases for the Increase in Substrate Profile of This Antibiotic Resistance Enzyme
1998 · Lionel Mourey, Kazuyuki Miyashita, et al. · Journal of the American Chemical Society · 50
Design, Synthesis, and Evaluation of a Potent Mechanism-Based Inhibitor for the TEM .beta.-Lactamase with Implications for the Enzyme Mechanism
1995 · Kazuyuki Miyashita, Irina Massova, et al. · Journal of the American Chemical Society · 48
Total Synthesis of Leustroducsin B
2008 · Kazuyuki Miyashita, Tomoyuki Tsunemi, et al. · The Journal of Organic Chemistry · 43
Design and Concise Synthesis of a Novel Type of Green Fluorescent Protein Chromophore Analogue
2012 · Masahiro Ikejiri, Moe Tsuchino, et al. · Organic Letters · 28
Total synthesis of leustroducsin B via a convergent route
2007 · Kazuyuki Miyashita, Tomoyuki Tsunemi, et al. · Tetrahedron Letters · 27
2′,4′-BNANC: A Novel Bridged Nucleic Acid Analogue with Excellent Hybridizing and Nuclease Resistance Profiles
2007 · S. M. Abdur Rahman, Sayori Seki, et al. · Nucleosides Nucleotides & Nucleic Acids · 21
6-(Hydroxyalkyl)penicillanates as Probes for Mechanisms of .BETA.-Lactamases.
2000 · DASANTILA GOLEMI, LAURENT MAVEYRAUD, et al. · The Journal of Antibiotics · 21
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Chiral environment specifically induced by metal ion: Asymmetric α-alkylation of α-amino esters using pyridoxal derivatives having a chiral ionophore function
1999 · Kazuyuki Miyashita, Hideto Miyabe, et al. · Tetrahedron · 21
Enhanced in Vitro Percutaneous Penetration of Salicylate by Ion Pair Formation with Alkylamines.
1998 · Masanori KADONO, Kazuyoshi KUBO, et al. · Biological and Pharmaceutical Bulletin · 19
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Quantification of the extent of attenuation of the rate of turnover chemistry of the TEM-1 β-lactamase by the α-1R-hydroxyethyl group in substrates
1996 · Kazuyuki Miyashita, Irina Massova, et al. · Bioorganic & Medicinal Chemistry Letters · 18
Synthesis and fluorescence properties of 4-diarylmethylene analogues of the green fluorescent protein chromophore
2015 · Masahiro Ikejiri, Kousuke Matsumoto, et al. · Tetrahedron · 16
Studies on novel and chiral 1,4-dihydropyridines. V. Hantzsch-type 1,4-dihydropyridines having a chiral sulfinyl group: Syntheses, structures, and biological activity as a calcium channel antagonist
1997 · Kazuyuki Miyashita, Masahiro Nishimoto, et al. · Tetrahedron · 16
Design, synthesis, and evaluation of a novel bridged nucleic acid, 2′,5′-BNAON, with S-type sugar conformation fixed by N–O linkage
2008 · Tetsuya Kodama, Chieko Matsuo, et al. · Tetrahedron · 15
Studies on Novel and Chiral 1,4-Dihydropyridines. I. Synthesis and Conformational Analysis of Novel NADH Model Compounds, N-Substituted (S)-3-(p-Tolylsulfinyl)-1,4-dihydropyridines.
1996 · Takeshi IMANISHI, Satoshi OBIKA, et al. · Chemical and Pharmaceutical Bulletin · 15
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Total synthesis of (.+-.)-solavetivone and aglycone A3. Regio- and stereo-selective Birch reduction of 6,10-dimethyl-2-hydroxy-spiro[4.5]deca-6,9-dien-8-one.
1987 · CHUZO IWATA, MINORU YAMADA, et al. · Chemical and Pharmaceutical Bulletin · 15
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Stereoselective and N-terminal selective α-alkylation of peptides using a pyridoxal model compound as a chiral N-terminal activator
1998 · Kazuyuki Miyashita, Hiroshi Iwaki, et al. · Chemical Communications · 14
Syntheses of 1-Substituted (SS)-3-p-Tolylsulfinyl-1,4-dihydropyridines, Chiral NADH Model Compounds
1997 · Takeshi Imanishi, Satoshi Obika, et al. · Heterocycles · 13
Asymmetric α-alkylation of α-amino esters using pyridoxal model compounds with a chiral ionophore function; dependence of stereoselectivity on a chelated metal ion
1996 · Kazuyuki Miyashita, Hideto Miyabe, et al. · Chemical Communications · 13
Novel Indore-Ring Construction Method for the Synthesis of 2-Trifluoromethylidoles
1996 · Takeshi Imanishi, Kazuyuki Miyashita, et al. · Heterocycles · 13
A hybrid molecule of a GFP chromophore analogue and cholestene as a viscosity-dependent and cholesterol-responsive fluorescent sensor
2017 · Masahiro Ikejiri, Kenta Mori, et al. · Organic & Biomolecular Chemistry · 12
Stereoselective Reduction of α-Bromopenicillanates by Tributylphosphine
2000 · Akihiro Ishiwata, Lakshmi P. Kotra, et al. · Organic Letters · 12
A modified procedure for the synthesis of spirodienones from phenolic .ALPHA.-diazoketones.
1985 · CHUZO IWATA, KAZUYUKI MIYASHITA, et al. · Chemical and Pharmaceutical Bulletin · 12
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Synthesis and properties of 4-(diarylmethylene)imidazolinone-conjugated fluorescent nucleic acids
2016 · Takumi Okuda, Shohei Mori, et al. · Tetrahedron Letters · 11
Stereospecific 4-Hydrogen Transfer in the Asymmetric Reduction Using (SS)-3-(p-Tolylsulfinyl)-1,4-dihydropyridines, NADH Model Compounds
1996 · Satoshi Obika, Toshihiko Nishiyama, et al. · Chemistry Letters · 11
Works count: 64
Citation count: 756
H-index: 15
I10-index: 30
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