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Peter Nußbaumer

Observed names: Nussbaumer, Peter, P A NUSSBAUMER, P. NUSSBAUMER, P. Nussbaumer, Peter Nussbaumer
Observed institutions: Novartis (Switzerland), TU Wien, Lead Discovery Center (Germany), Novartis (Austria), Sandoz Group AG (Switzerland), Novartis Institutes for BioMedical Research
ORCID: 0000-0002-2761-629X
Observed ORCID: 0000-0002-2761-629X
OpenAlex ID: A5103171217
Gasdermin D plays a vital role in the generation of neutrophil extracellular traps
2018 · Gabriel Sollberger, Axel Choidas, et al. · Science Immunology · 784
Small-molecule inhibitors of human mitochondrial DNA transcription
2020 · Nina A. Bonekamp, Bradley Peter, et al. · Nature · 275
Identification of Atuveciclib (BAY 1143572), the First Highly Selective, Clinical PTEFb/CDK9 Inhibitor for the Treatment of Cancer
2017 · Ulrich Lücking, Arne Scholz, et al. · ChemMedChem · 197
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Identification of pyrazolopyridazinones as PDEδ inhibitors
2016 · Björn Papke, Sandip Murarka, et al. · Nature Communications · 164
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Picomolar, selective, and subtype-specific small-molecule inhibition of TRPC1/4/5 channels
2017 · Hussein N. Rubaiy, Melanie J. Ludlow, et al. · Journal of Biological Chemistry · 122
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Regulation and Traffic of Ceramide 1-Phosphate Produced by Ceramide Kinase
2007 · Alistair Boath, Christine Graf, et al. · Journal of Biological Chemistry · 115
2-Substituted 4-(Thio)chromenone 6-O-Sulfamates: Potent Inhibitors of Human Steroid Sulfatase
2002 · Peter Nussbaumer, Philipp Lehr, et al. · Journal of Medicinal Chemistry · 112
Steroid sulfatase inhibitors
2004 · Peter Nussbaumer, Andreas Billich · Medicinal Research Reviews · 108
Synthesis and Structure-Activity Relationships of Side-Chain-Substituted Analogs of the Allylamine Antimycotic Terbinafine Lacking the Central Amino Function
1995 · Peter Nussbaumer, Ingrid Leitner, et al. · Journal of Medicinal Chemistry · 105
Synthesis of Borondipyrromethene (BODIPY)-Labeled Sphingosine Derivatives by Cross-metathesis Reaction
2007 · Carsten Peters, Andreas Billich, et al. · The Journal of Organic Chemistry · 98
Stimulation of MCF-7 breast cancer cell proliferation by estrone sulfate and dehydroepiandrosterone sulfate: inhibition by novel non-steroidal steroid sulfatase inhibitors
2000 · Andreas Billich, Peter Nussbaumer, et al. · The Journal of Steroid Biochemistry and Molecular Biology · 97
Dynarrestin, a Novel Inhibitor of Cytoplasmic Dynein
2018 · Susanne Höing, Ting-Yu Yeh, et al. · Cell chemical biology · 85
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Structure Guided Design and Kinetic Analysis of Highly Potent Benzimidazole Inhibitors Targeting the PDEδ Prenyl Binding Site
2014 · Gunther Zimmermann, Carsten Schultz-Fademrecht, et al. · Journal of Medicinal Chemistry · 65
Dual Inhibition of GSK3β and CDK5 Protects the Cytoskeleton of Neurons from Neuroinflammatory-Mediated Degeneration In Vitro and In Vivo
2019 · Lydia Reinhardt, Susanne Kordes, et al. · Stem Cell Reports · 64
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Synthesis and structure-activity relationships of benzo[b]thienylallylamine antimycotics
1991 · Peter Nussbaumer, Gabor Petranyi, et al. · Journal of Medicinal Chemistry · 61
Inhibitors of vitamin D hydroxylases: Structure–activity relationships
2003 · Inge Schuster, Helmut Egger, et al. · Journal of Cellular Biochemistry · 60
Design, synthesis and biological evaluation of 3,5-disubstituted 2-amino thiophene derivatives as a novel class of antitumor agents
2013 · Romeo Romagnoli, Pier Giovanni Baraldi, et al. · Bioorganic & Medicinal Chemistry · 47
Identification of Two Secondary Ligand Binding Sites in 14-3-3 Proteins Using Fragment Screening
2017 · Eline Sijbesma, Lukasz Skora, et al. · Biochemistry · 46
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2-(1-Adamantyl)-4-(thio)chromenone-6-carboxylic Acids: Potent Reversible Inhibitors of Human Steroid Sulfatase
2004 · Amarylla Horvath, Peter Nussbaumer, et al. · Journal of Medicinal Chemistry · 40
Synthesis and structure-activity relationships of phenyl-substituted benzylamine antimycotics: a novel benzylbenzylamine antifungal agent for systemic treatment
1993 · Peter Nussbaumer, Gerhard Dorfstaetter, et al. · Journal of Medicinal Chemistry · 40
Na+ entry through heteromeric TRPC4/C1 channels mediates (−)Englerin A-induced cytotoxicity in synovial sarcoma cells
2017 · Katsuhiko Muraki, Kaori Ohnishi, et al. · Scientific Reports · 37
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Estrogenic Potential of 2-Alkyl-4-(thio)chromenone 6-O-Sulfamates: Potent Inhibitors of Human Steroid Sulfatase
2003 · Peter Nussbaumer, Anthony P. Winiski, et al. · Journal of Medicinal Chemistry · 37
Fluorescence-labeled sphingosines as substrates of sphingosine kinases 1 and 2
2004 · Peter Ettmayer, Andreas Billich, et al. · Bioorganic & Medicinal Chemistry Letters · 35
Steroid sulfatase inhibitors
2003 · Peter Nussbaumer, Andreas Billich · Expert Opinion on Therapeutic Patents · 35
Development of Pyridazinone Chemotypes Targeting the PDEδ Prenyl Binding Site
2016 · Sandip Murarka, Pablo Martín‐Gago, et al. · Chemistry - A European Journal · 34
Works count: 112
Citation count: 3,602
H-index: 29
I10-index: 57
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