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Yayoi Fujioka
Observed institutions:
Taiho Pharmaceutical (Japan),
Kindai University
OpenAlex ID:
A5103454927
Futibatinib Is a Novel Irreversible FGFR 1–4 Inhibitor That Shows Selective Antitumor Activity against FGFR-Deregulated Tumors
2020
·
Hiroshi Sootome
, Hidenori Fujita
, et al.
·
Cancer Research
·
215
PDF
The Novel VEGF Receptor/MET–Targeted Kinase Inhibitor TAS-115 Has Marked In Vivo Antitumor Properties and a Favorable Tolerability Profile
2013
·
Hidenori Fujita
, Kazutaka Miyadera
, et al.
·
Molecular Cancer Therapeutics
·
38
Acquired resistance to trastuzumab/pertuzumab or to T‐DM1 in vivo can be overcome by HER2 kinase inhibition with TAS0728
2020
·
Hiroki Irie
, Rumi Kawabata
, et al.
·
Cancer Science
·
36
PDF
Abstract A270: TAS-120, a highly potent and selective irreversible FGFR inhibitor, is effective in tumors harboring various FGFR gene abnormalities.
2013
·
Hiroaki Ochiiwa
, Hidenori Fujita
, et al.
·
Molecular Cancer Therapeutics
·
28
Activity of TAS4464, a novel NEDD8 activating enzyme E1 inhibitor, against multiple myeloma via inactivation of nuclear factor κB pathways
2019
·
Hiromi Muraoka
, Chihoko Yoshimura
, et al.
·
Cancer Science
·
27
PDF
High Potency VEGFRs/MET/FMS Triple Blockade by TAS-115 Concomitantly Suppresses Tumor Progression and Bone Destruction in Tumor-Induced Bone Disease Model with Lung Carcinoma Cells
2016
·
Hidenori Fujita
, Akira Gomori
, et al.
·
PLoS ONE
·
21
PDF
TAS0728, A Covalent-binding, HER2-selective Kinase Inhibitor Shows Potent Antitumor Activity in Preclinical Models
2019
·
Hiroki Irie
, Kimihiro Ito
, et al.
·
Molecular Cancer Therapeutics
·
15
Abstract A271: TAS-120, an irreversible FGFR inhibitor, was effective in tumors harboring FGFR mutations, refractory or resistant to ATP competitive inhibitors .
2013
·
Hiroshi Sootome
, Yayoi Fujioka
, et al.
·
Molecular Cancer Therapeutics
·
11
Abstract A272: Intermittent treatment with TAS-120, an irreversible FGFR inhibitor, is effective in tumors harboring a FGFR gene abnormality.
2013
·
Yoko Nakatsuru
, Hiroaki Ochiiwa
, et al.
·
Molecular Cancer Therapeutics
·
2
Abstract 3577: TAS-115: a highly potent c-Met + VEGFRs dual inhibitor with prominently safer profile
2011
·
Hidenori Fujita
, Kazutaka Miyadera
, et al.
·
Cancer Research
·
2
Abstract 3600: The prominent safety profile of TAS-115, a novel c-Met + VEGFR dual kinase inhibitor can lead to potentiate the efficacy via durable inhibition of angiogenesis
2011
·
Hiroaki Ochiiwa
, Hidenori Fujita
, et al.
·
Cancer Research
·
2
Data from Futibatinib Is a Novel Irreversible FGFR 1–4 Inhibitor That Shows Selective Antitumor Activity against FGFR-Deregulated Tumors
2023
·
Hiroshi Sootome
, Hidenori Fujita
, et al.
·
1
Abstract A126: Acquired resistance to trastuzumab/pertuzumab, or to T-DM1 in vivo can be overcome by HER2 inhibition with TAS0728
2019
·
Hiroki Irie
, Rumi Kawabata
, et al.
·
Molecular Cancer Therapeutics
·
1
Abstract 1785: MET/VEGFR dual inhibition and prominent safety profile of TAS-115 are favorable for the combination with chemotherapeutic drugs
2012
·
Hidenori Fujita
, Masanori Kato
, et al.
·
Cancer Research
·
1
Data from The Novel VEGF Receptor/MET–Targeted Kinase Inhibitor TAS-115 Has Marked In Vivo Antitumor Properties and a Favorable Tolerability Profile
2023
·
Hidenori Fujita
, Kazutaka Miyadera
, et al.
Data from The Novel VEGF Receptor/MET–Targeted Kinase Inhibitor TAS-115 Has Marked In Vivo Antitumor Properties and a Favorable Tolerability Profile
2023
·
Hidenori Fujita
, Kazutaka Miyadera
, et al.
Data from TAS0728, A Covalent-binding, HER2-selective Kinase Inhibitor Shows Potent Antitumor Activity in Preclinical Models
2023
·
Hiroki Irie
, Kimihiro Ito
, et al.
Supplementary Figures 1 through 5 and Supplementary Tables 1 through 3 from The Novel VEGF Receptor/MET–Targeted Kinase Inhibitor TAS-115 Has Marked In Vivo Antitumor Properties and a Favorable Tolerability Profile
2023
·
Hidenori Fujita
, Kazutaka Miyadera
, et al.
PDF
Table S2 from TAS0728, A Covalent-binding, HER2-selective Kinase Inhibitor Shows Potent Antitumor Activity in Preclinical Models
2023
·
Hiroki Irie
, Kimihiro Ito
, et al.
PDF
Figure S1 from TAS0728, A Covalent-binding, HER2-selective Kinase Inhibitor Shows Potent Antitumor Activity in Preclinical Models
2023
·
Hiroki Irie
, Kimihiro Ito
, et al.
PDF
Figure S2 from TAS0728, A Covalent-binding, HER2-selective Kinase Inhibitor Shows Potent Antitumor Activity in Preclinical Models
2023
·
Hiroki Irie
, Kimihiro Ito
, et al.
PDF
Table S1 from TAS0728, A Covalent-binding, HER2-selective Kinase Inhibitor Shows Potent Antitumor Activity in Preclinical Models
2023
·
Hiroki Irie
, Kimihiro Ito
, et al.
PDF
Table S1 from TAS0728, A Covalent-binding, HER2-selective Kinase Inhibitor Shows Potent Antitumor Activity in Preclinical Models
2023
·
Hiroki Irie
, Kimihiro Ito
, et al.
Table S2 from TAS0728, A Covalent-binding, HER2-selective Kinase Inhibitor Shows Potent Antitumor Activity in Preclinical Models
2023
·
Hiroki Irie
, Kimihiro Ito
, et al.
Figure S1 from TAS0728, A Covalent-binding, HER2-selective Kinase Inhibitor Shows Potent Antitumor Activity in Preclinical Models
2023
·
Hiroki Irie
, Kimihiro Ito
, et al.
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Works count:
36
Citation count:
400
H-index:
8
I10-index:
8
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