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Giuseppe Merlino
Observed names:
MERLINO, GIUSEPPE,
Merlino, Giuseppe
Observed institutions:
Mario Negri Institute for Pharmacological Research,
Menarini Group (Italy),
Fondazione IRCCS Istituto Nazionale dei Tumori
OpenAlex ID:
A5106085666
Tumor-extracellular matrix interactions: Identification of tools associated with breast cancer progression
2015
·
Marta Giussani
, Giuseppe Merlino
, et al.
·
Seminars in Cancer Biology
·
158
PDF
Complexity in the tumour microenvironment: Cancer associated fibroblast gene expression patterns identify both common and unique features of tumour-stroma crosstalk across cancer types
2015
·
Paolo Gandellini
, Francesca Andriani
, et al.
·
Seminars in Cancer Biology
·
140
Extracellular matrix proteins as diagnostic markers of breast carcinoma
2018
·
Marta Giussani
, Elena Landoni
, et al.
·
Journal of Cellular Physiology
·
77
Targeting CD205 with the antibody drug conjugate MEN1309/OBT076 is an active new therapeutic strategy in lymphoma models
2020
·
Eugenio Gaudio
, Chiara Tarantelli
, et al.
·
Haematologica
·
31
PDF
Comparative Magnetic Resonance Imaging and Histopathological Correlates in Two SOD1 Transgenic Mouse Models of Amyotrophic Lateral Sclerosis
2015
·
Ilaria Caron
, Edoardo Micotti
, et al.
·
PLoS ONE
·
27
PDF
MEN1309/OBT076, a First-In-Class Antibody–Drug Conjugate Targeting CD205 in Solid Tumors
2019
·
Giuseppe Merlino
, Alessio Fiascarelli
, et al.
·
Molecular Cancer Therapeutics
·
24
PDF
Model‐based prediction of effective target exposure for MEN1611 in combination with trastuzumab in HER2 ‐positive advanced or metastatic breast cancer patients
2023
·
Elena M. Tosca
, Elisa Borella
, et al.
·
CPT Pharmacometrics & Systems Pharmacology
·
14
PDF
Antitumor activity of the PI3K δ-sparing inhibitor MEN1611 in PIK3CA mutated, trastuzumab-resistant HER2 + breast cancer
2023
·
Alessio Fiascarelli
, Giuseppe Merlino
, et al.
·
Breast Cancer Research and Treatment
·
10
PDF
Prognostic and functional role of subtype‐specific tumor–stroma interaction in breast cancer
2017
·
Giuseppe Merlino
, Patrizia Miodini
, et al.
·
Molecular Oncology
·
10
PDF
In-depth characterization of breast cancer tumor-promoting cell transcriptome by RNA sequencing and microarrays
2015
·
Maurizio Callari
, Alessandro Guffanti
, et al.
·
Oncotarget
·
9
PDF
Stromal Activation by Tumor Cells: An in Vitro Study in Breast Cancer
2016
·
Giuseppe Merlino
, Patrizia Miodini
, et al.
·
Microarrays
·
8
PDF
Tumor Growth in the High Frequency Medulloblastoma Mouse Model Ptch1+/−/Tis21KO Has a Specific Activation Signature of the PI3K/AKT/mTOR Pathway and Is Counteracted by the PI3K Inhibitor MEN1611
2021
·
Manuela Ceccarelli
, Giorgio D’Andrea
, et al.
·
Frontiers in Oncology
·
7
PDF
The Dual PIM / FLT3 Inhibitor MEN1703 Combines Synergistically With Gilteritinib in FLT3 ‐ ITD ‐Mutant Acute Myeloid Leukaemia
2024
·
Sonia Zicari
, Giuseppe Merlino
, et al.
·
Journal of Cellular and Molecular Medicine
·
5
PDF
Abstract 2160: MEN1611, a novel α-selective PI3K inhibitor in solid tumors
2018
·
Giuseppe Merlino
, Alessio Fiascarelli
, et al.
·
Cancer Research
·
5
CD205-Shuttle study: A first-in-human trial of MEN1309/OBT076 an ADC targeting CD205 in solid tumor and NHL.
2018
·
Elena Garralda
, Josep Tabernero
, et al.
·
Journal of Clinical Oncology
·
3
The activity of a PI3K δ-sparing inhibitor, MEN1611, in non-small cell lung cancer cells with constitutive activation of the PI3K/AKT/mTOR pathway
2023
·
Giuliana Papoff
, Dario Presutti
, et al.
·
Frontiers in Oncology
·
2
Abstract 2849: The oral SERD Elacestrant in combination with the PI3K inhibitor MEN1611 inhibits tumor growth in ER+/HER2- breast cancer in vitro and in PDX models
2023
·
Giuseppe Merlino
, Alessio Fiascarelli
, et al.
·
Cancer Research
·
2
Abstract 2630: MEN1309, a novel antibody drug conjugate (ADC) targeting Ly75 antigen, induces complete responses in several xenografts of solid tumors
2017
·
Mario Bigioni
, Giuseppe Merlino
, et al.
·
Cancer Research
·
1
CD205, a target antigen for a novel antibody drug conjugate (ADC): Evaluation of antigen expression on non-Hodgkin lymphoma (NHL).
2017
·
Vincenzo Canzonieri
, Valter Gattei
, et al.
·
Journal of Clinical Oncology
·
1
MaNgROVIVIRga CUNICULI gen. nov., sp. nov., a moderately halophilic bacterium isolated from bioturbated Red Sea mangrove sediment, and proposal of the novel family MaNgROVIVIRgaCeae fam. nov.
2026
·
Sefrji, Fatmah O.
, Michoud, Grégoire
, et al.
·
The Catalogue of Life
Abstract 665: MEN1703/SEL24 exhibits promising antitumoral activity in preclinical models of myelofibrosis both as single agent and combined with ruxolitinib
2024
·
Maria Luisa Iannitto
, Diego Bisignano
, et al.
·
Cancer Research
Data from MEN1309/OBT076, a First-In-Class Antibody–Drug Conjugate Targeting CD205 in Solid Tumors
2023
·
Giuseppe Merlino
, Alessio Fiascarelli
, et al.
Supplementary Data from MEN1309/OBT076, a First-In-Class Antibody–Drug Conjugate Targeting CD205 in Solid Tumors
2023
·
Giuseppe Merlino
, Alessio Fiascarelli
, et al.
Supplementary Figure S1 from MEN1309/OBT076, a First-In-Class Antibody–Drug Conjugate Targeting CD205 in Solid Tumors
2023
·
Giuseppe Merlino
, Alessio Fiascarelli
, et al.
Supplementary Figure S2 from MEN1309/OBT076, a First-In-Class Antibody–Drug Conjugate Targeting CD205 in Solid Tumors
2023
·
Giuseppe Merlino
, Alessio Fiascarelli
, et al.
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Works count:
62
Citation count:
534
H-index:
9
I10-index:
9
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