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Wayne Jackson

Observed names: Jackson, W., W. Jackson
OpenAlex ID: A5108495886
2-Anilino-4-(thiazol-5-yl)pyrimidine CDK Inhibitors: Synthesis, SAR Analysis, X-ray Crystallography, and Biological Activity
2004 · Shudong Wang, Christopher Meades, et al. · Journal of Medicinal Chemistry · 154
Discovery and Characterization of 2-Anilino-4- (Thiazol-5-yl)Pyrimidine Transcriptional CDK Inhibitors as Anticancer Agents
2010 · Shudong Wang, Gary Griffiths, et al. · Chemistry & Biology · 107
Discovery ofN-Phenyl-4-(thiazol-5-yl)pyrimidin-2-amine Aurora Kinase Inhibitors
2010 · Shudong Wang, Carol A. Midgley, et al. · Journal of Medicinal Chemistry · 102
Structural Determinants of CDK4 Inhibition and Design of Selective ATP Competitive Inhibitors
2004 · Campbell McInnes, Shudong Wang, et al. · Chemistry & Biology · 63
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Synthesis and biological activity of 2-anilino-4-(1H-pyrrol-3-yl) pyrimidine CDK inhibitors
2004 · Shudong Wang, Gavin Wood, et al. · Bioorganic & Medicinal Chemistry Letters · 61
Molecular profiling and combinatorial activity of CCT 068127: a potent CDK 2 and CDK 9 inhibitor
2017 · Steven R. Whittaker, Clare Barlow, et al. · Molecular Oncology · 41
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Design, synthesis and biological evaluation of 6-pyridylmethylaminopurines as CDK inhibitors
2011 · Stuart C. Wilson, Butrus Atrash, et al. · Bioorganic & Medicinal Chemistry · 35
Design, Synthesis, and Evaluation of 2-Methyl- and 2-Amino-N-aryl-4,5-dihydrothiazolo[4,5-h]quinazolin-8-amines as Ring-Constrained 2-Anilino-4-(thiazol-5-yl)pyrimidine Cyclin-Dependent Kinase Inhibitors
2010 · Neil A. McIntyre, Campbell McInnes, et al. · Journal of Medicinal Chemistry · 35
Novel cyclin dependent kinase (CDK) inhibitors induce down regulation of Mcl-1 and apoptosis in multiple myeloma cells
2006 · David E. MacCallum, Jean Melville, et al. · Cancer Research · 1
CCDC 818968: Experimental Crystal Structure Determination
2011 · McIntyre, N.A., McInnes, C., et al. · The Cambridge Structural Database
HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE INHIBITOR N-[4-(2,4-Dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-N',N'-dimethyl-benzene-1,4-diamine
2003 · S. Wang, C. Meades, et al. · Worldwide Protein Data Bank
HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE INHIBITOR 4-[4-(4-Methyl-2-methylamino-thiazol-5-yl)-pyrimidin-2-ylamino]-phenol
2003 · S. Wang, C. Meades, et al. · Worldwide Protein Data Bank
Works count: 13
Citation count: 599
H-index: 8
I10-index: 8
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